FI68044C - Foerfarande foer framstaellning av terapeutiskt aktiva n-(4-pyrazolidinyl)bensamider - Google Patents

Foerfarande foer framstaellning av terapeutiskt aktiva n-(4-pyrazolidinyl)bensamider Download PDF

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Publication number
FI68044C
FI68044C FI782507A FI782507A FI68044C FI 68044 C FI68044 C FI 68044C FI 782507 A FI782507 A FI 782507A FI 782507 A FI782507 A FI 782507A FI 68044 C FI68044 C FI 68044C
Authority
FI
Finland
Prior art keywords
amino
formula
substituted
pyrazolidine
pyrazolidinyl
Prior art date
Application number
FI782507A
Other languages
English (en)
Finnish (fi)
Other versions
FI68044B (fi
FI782507A (fi
Inventor
Carl Dalton Lunsford
Jr Albert Duncan Cale
Original Assignee
Robins Co Inc A H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robins Co Inc A H filed Critical Robins Co Inc A H
Publication of FI782507A publication Critical patent/FI782507A/fi
Priority to FI832671A priority Critical patent/FI70706C/fi
Publication of FI68044B publication Critical patent/FI68044B/fi
Application granted granted Critical
Publication of FI68044C publication Critical patent/FI68044C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/04Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Hospice & Palliative Care (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Otolaryngology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI782507A 1977-08-19 1978-08-16 Foerfarande foer framstaellning av terapeutiskt aktiva n-(4-pyrazolidinyl)bensamider FI68044C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI832671A FI70706C (fi) 1977-08-19 1983-07-22 4-aminopyrazolidinderivat till anvaendning som mellanprodukt vid framstaellning av n-(4-pyrazolidinyl)bensamider

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US82603177A 1977-08-19 1977-08-19
US82603177 1977-08-19
US90036978A 1978-04-26 1978-04-26
US90036978 1978-04-26
US93012578A 1978-08-01 1978-08-01
US93012578 1978-08-01

Publications (3)

Publication Number Publication Date
FI782507A FI782507A (fi) 1979-02-20
FI68044B FI68044B (fi) 1985-03-29
FI68044C true FI68044C (fi) 1985-07-10

Family

ID=27420183

Family Applications (1)

Application Number Title Priority Date Filing Date
FI782507A FI68044C (fi) 1977-08-19 1978-08-16 Foerfarande foer framstaellning av terapeutiskt aktiva n-(4-pyrazolidinyl)bensamider

Country Status (21)

Country Link
JP (1) JPS5441873A (cs)
AU (1) AU521421B2 (cs)
BR (1) BR7805288A (cs)
CA (1) CA1105037A (cs)
CH (2) CH639374A5 (cs)
DE (1) DE2836062A1 (cs)
DK (1) DK152361C (cs)
ES (1) ES472686A1 (cs)
FI (1) FI68044C (cs)
FR (1) FR2400511A1 (cs)
GB (2) GB2017678B (cs)
HK (1) HK42282A (cs)
IE (1) IE47430B1 (cs)
MX (1) MX5469E (cs)
NL (1) NL7808596A (cs)
NO (1) NO149107C (cs)
NZ (1) NZ188189A (cs)
PH (1) PH13331A (cs)
PT (1) PT68442A (cs)
SE (2) SE444434B (cs)
YU (1) YU41116B (cs)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4309552A (en) * 1980-08-07 1982-01-05 A. H. Robins Company, Inc. Synthesis of 4-nitro-1,2-hydrocarbyl pyrazolidines and process for preparation thereof
US5126343A (en) * 1989-09-11 1992-06-30 G. D. Searle & Co. N-azabicyclo [3.3.0]octane amides of aromatic acids
JP3065506B2 (ja) * 1995-04-03 2000-07-17 株式会社資生堂 ピラゾリジン誘導体及びラジカルスカベンジャー、脳梗塞抑制剤、脳浮腫抑制剤
AR086587A1 (es) 2011-05-31 2014-01-08 Syngenta Participations Ag Compuestos insecticidas

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3966957A (en) * 1972-04-03 1976-06-29 A. H. Robins Company, Incorporated Method for controlling emesis with N-(1-substituted-3-pyrrolidinyl)benzamides and thiobenzamides

Also Published As

Publication number Publication date
NO782812L (no) 1979-02-20
YU41116B (en) 1986-12-31
ES472686A1 (es) 1979-03-16
PH13331A (en) 1980-03-13
SE8303564D0 (sv) 1983-06-21
PT68442A (en) 1978-09-01
CA1105037A (en) 1981-07-14
IE47430B1 (en) 1984-03-21
NO149107C (no) 1984-02-22
IE781682L (en) 1979-02-19
AU521421B2 (en) 1982-04-01
FR2400511A1 (fr) 1979-03-16
AU3906178A (en) 1980-02-21
FI68044B (fi) 1985-03-29
GB2017678B (en) 1982-03-10
HK42282A (en) 1982-10-08
GB2003153B (en) 1982-02-24
FR2400511B1 (cs) 1981-09-04
MX5469E (es) 1983-08-16
GB2017678A (en) 1979-10-10
YU198678A (en) 1983-01-21
JPS5441873A (en) 1979-04-03
GB2003153A (en) 1979-03-07
SE8303564L (sv) 1983-06-21
DK366978A (da) 1979-02-20
JPS6315273B2 (cs) 1988-04-04
NO149107B (no) 1983-11-07
DK152361B (da) 1988-02-22
CH645356A5 (fr) 1984-09-28
SE444434B (sv) 1986-04-14
SE451723B (sv) 1987-10-26
FI782507A (fi) 1979-02-20
NZ188189A (en) 1984-07-06
DE2836062A1 (de) 1979-03-01
SE7808694L (sv) 1979-02-20
BR7805288A (pt) 1979-04-10
CH639374A5 (fr) 1983-11-15
DK152361C (da) 1988-07-25
NL7808596A (nl) 1979-02-21

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Legal Events

Date Code Title Description
BB Publication of examined application
BB Publication of examined application
MM Patent lapsed

Owner name: A.H. ROBINS COMPANY, INCORPORATED