ES472686A1 - Procedimiento para preparar n-(4-pirazolidinil) benzamidas. - Google Patents

Procedimiento para preparar n-(4-pirazolidinil) benzamidas.

Info

Publication number
ES472686A1
ES472686A1 ES472686A ES472686A ES472686A1 ES 472686 A1 ES472686 A1 ES 472686A1 ES 472686 A ES472686 A ES 472686A ES 472686 A ES472686 A ES 472686A ES 472686 A1 ES472686 A1 ES 472686A1
Authority
ES
Spain
Prior art keywords
alkyl
benzamides
lower alkyl
pyrzaolidinyl
phenyllower
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES472686A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AH Robins Co Inc
Original Assignee
AH Robins Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by AH Robins Co Inc filed Critical AH Robins Co Inc
Publication of ES472686A1 publication Critical patent/ES472686A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/04—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Hospice & Palliative Care (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Otolaryngology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La presente invención se refiere a compuestos heterocíclicos que tienen propiedades antieméticas y de vaciado gástrico, y se refiere particularmente a ciertas N-(4-pirazolidinil) benzamidas, a composiciones de las mismas y a métodos para emplear las composiciones para controlar las propiedades de emesis y de vaciado gástrico en animales de sangre caliente, con efectos secundarios mínimos.
ES472686A 1977-08-19 1978-08-18 Procedimiento para preparar n-(4-pirazolidinil) benzamidas. Expired ES472686A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US82603177A 1977-08-19 1977-08-19
US90036978A 1978-04-26 1978-04-26
US93012578A 1978-08-01 1978-08-01

Publications (1)

Publication Number Publication Date
ES472686A1 true ES472686A1 (es) 1979-03-16

Family

ID=27420183

Family Applications (1)

Application Number Title Priority Date Filing Date
ES472686A Expired ES472686A1 (es) 1977-08-19 1978-08-18 Procedimiento para preparar n-(4-pirazolidinil) benzamidas.

Country Status (21)

Country Link
JP (1) JPS5441873A (es)
AU (1) AU521421B2 (es)
BR (1) BR7805288A (es)
CA (1) CA1105037A (es)
CH (2) CH639374A5 (es)
DE (1) DE2836062A1 (es)
DK (1) DK152361C (es)
ES (1) ES472686A1 (es)
FI (1) FI68044C (es)
FR (1) FR2400511A1 (es)
GB (2) GB2017678B (es)
HK (1) HK42282A (es)
IE (1) IE47430B1 (es)
MX (1) MX5469E (es)
NL (1) NL7808596A (es)
NO (1) NO149107C (es)
NZ (1) NZ188189A (es)
PH (1) PH13331A (es)
PT (1) PT68442A (es)
SE (2) SE444434B (es)
YU (1) YU41116B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4309552A (en) * 1980-08-07 1982-01-05 A. H. Robins Company, Inc. Synthesis of 4-nitro-1,2-hydrocarbyl pyrazolidines and process for preparation thereof
US5126343A (en) * 1989-09-11 1992-06-30 G. D. Searle & Co. N-azabicyclo [3.3.0]octane amides of aromatic acids
JP3065506B2 (ja) 1995-04-03 2000-07-17 株式会社資生堂 ピラゾリジン誘導体及びラジカルスカベンジャー、脳梗塞抑制剤、脳浮腫抑制剤
TW201311677A (zh) * 2011-05-31 2013-03-16 Syngenta Participations Ag 殺蟲化合物

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3966957A (en) * 1972-04-03 1976-06-29 A. H. Robins Company, Incorporated Method for controlling emesis with N-(1-substituted-3-pyrrolidinyl)benzamides and thiobenzamides

Also Published As

Publication number Publication date
GB2017678B (en) 1982-03-10
DE2836062A1 (de) 1979-03-01
DK152361B (da) 1988-02-22
SE451723B (sv) 1987-10-26
SE8303564L (sv) 1983-06-21
YU41116B (en) 1986-12-31
DK152361C (da) 1988-07-25
GB2003153B (en) 1982-02-24
FI782507A (fi) 1979-02-20
NZ188189A (en) 1984-07-06
BR7805288A (pt) 1979-04-10
PT68442A (en) 1978-09-01
AU3906178A (en) 1980-02-21
MX5469E (es) 1983-08-16
FI68044C (fi) 1985-07-10
HK42282A (en) 1982-10-08
YU198678A (en) 1983-01-21
NO782812L (no) 1979-02-20
CA1105037A (en) 1981-07-14
NO149107C (no) 1984-02-22
CH645356A5 (fr) 1984-09-28
JPS6315273B2 (es) 1988-04-04
NO149107B (no) 1983-11-07
SE444434B (sv) 1986-04-14
SE8303564D0 (sv) 1983-06-21
PH13331A (en) 1980-03-13
IE781682L (en) 1979-02-19
CH639374A5 (fr) 1983-11-15
DK366978A (da) 1979-02-20
AU521421B2 (en) 1982-04-01
FI68044B (fi) 1985-03-29
IE47430B1 (en) 1984-03-21
FR2400511B1 (es) 1981-09-04
NL7808596A (nl) 1979-02-21
GB2017678A (en) 1979-10-10
FR2400511A1 (fr) 1979-03-16
GB2003153A (en) 1979-03-07
JPS5441873A (en) 1979-04-03
SE7808694L (sv) 1979-02-20

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19971103