FR2400511A1 - N-(4-pyrazolidinyl) benzamides, presentant notamment des proprietes antiemetiques et de vidage gastrique - Google Patents

N-(4-pyrazolidinyl) benzamides, presentant notamment des proprietes antiemetiques et de vidage gastrique

Info

Publication number
FR2400511A1
FR2400511A1 FR7824138A FR7824138A FR2400511A1 FR 2400511 A1 FR2400511 A1 FR 2400511A1 FR 7824138 A FR7824138 A FR 7824138A FR 7824138 A FR7824138 A FR 7824138A FR 2400511 A1 FR2400511 A1 FR 2400511A1
Authority
FR
France
Prior art keywords
benzamides
pyrazolidinyl
antiemetic
presenting
gastric emptying
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7824138A
Other languages
English (en)
Other versions
FR2400511B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AH Robins Co Inc
Original Assignee
AH Robins Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by AH Robins Co Inc filed Critical AH Robins Co Inc
Publication of FR2400511A1 publication Critical patent/FR2400511A1/fr
Application granted granted Critical
Publication of FR2400511B1 publication Critical patent/FR2400511B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/04—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Hospice & Palliative Care (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Otolaryngology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La présente invention concerne des N-(4-pyrazolidinyl-benzamides de formules :
FR7824138A 1977-08-19 1978-08-18 N-(4-pyrazolidinyl) benzamides, presentant notamment des proprietes antiemetiques et de vidage gastrique Granted FR2400511A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US82603177A 1977-08-19 1977-08-19
US90036978A 1978-04-26 1978-04-26
US93012578A 1978-08-01 1978-08-01

Publications (2)

Publication Number Publication Date
FR2400511A1 true FR2400511A1 (fr) 1979-03-16
FR2400511B1 FR2400511B1 (fr) 1981-09-04

Family

ID=27420183

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7824138A Granted FR2400511A1 (fr) 1977-08-19 1978-08-18 N-(4-pyrazolidinyl) benzamides, presentant notamment des proprietes antiemetiques et de vidage gastrique

Country Status (21)

Country Link
JP (1) JPS5441873A (fr)
AU (1) AU521421B2 (fr)
BR (1) BR7805288A (fr)
CA (1) CA1105037A (fr)
CH (2) CH639374A5 (fr)
DE (1) DE2836062A1 (fr)
DK (1) DK152361C (fr)
ES (1) ES472686A1 (fr)
FI (1) FI68044C (fr)
FR (1) FR2400511A1 (fr)
GB (2) GB2017678B (fr)
HK (1) HK42282A (fr)
IE (1) IE47430B1 (fr)
MX (1) MX5469E (fr)
NL (1) NL7808596A (fr)
NO (1) NO149107C (fr)
NZ (1) NZ188189A (fr)
PH (1) PH13331A (fr)
PT (1) PT68442A (fr)
SE (2) SE444434B (fr)
YU (1) YU41116B (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2490639A1 (fr) * 1980-08-07 1982-03-26 Robins Co Inc A H Nouveau procede pour la synthese de 4-amino-1,2-dihydrocarbylpyrazolidines par l'intermediaire des analogues 4-nitro

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5126343A (en) * 1989-09-11 1992-06-30 G. D. Searle & Co. N-azabicyclo [3.3.0]octane amides of aromatic acids
JP3065506B2 (ja) * 1995-04-03 2000-07-17 株式会社資生堂 ピラゾリジン誘導体及びラジカルスカベンジャー、脳梗塞抑制剤、脳浮腫抑制剤
UY34104A (es) 2011-05-31 2013-01-03 Syngenta Participations Ag ?compuestos derivados benzamídicos heterocíclicos, procesos e intermedios para su preparación, composiciones y métodos para su uso?.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3966957A (en) * 1972-04-03 1976-06-29 A. H. Robins Company, Incorporated Method for controlling emesis with N-(1-substituted-3-pyrrolidinyl)benzamides and thiobenzamides

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2490639A1 (fr) * 1980-08-07 1982-03-26 Robins Co Inc A H Nouveau procede pour la synthese de 4-amino-1,2-dihydrocarbylpyrazolidines par l'intermediaire des analogues 4-nitro
FR2491065A1 (fr) * 1980-08-07 1982-04-02 Robins Co Inc A H Nouveau procede pour la synthese de 4-nitro-1,2-dihydrocarbyl-pyrazolidines, et produits obtenus

Also Published As

Publication number Publication date
GB2003153B (en) 1982-02-24
YU41116B (en) 1986-12-31
CH639374A5 (fr) 1983-11-15
SE444434B (sv) 1986-04-14
SE8303564D0 (sv) 1983-06-21
FI68044C (fi) 1985-07-10
CH645356A5 (fr) 1984-09-28
GB2017678B (en) 1982-03-10
JPS6315273B2 (fr) 1988-04-04
PT68442A (en) 1978-09-01
FI68044B (fi) 1985-03-29
NO149107B (no) 1983-11-07
NO782812L (no) 1979-02-20
IE781682L (en) 1979-02-19
SE8303564L (sv) 1983-06-21
FI782507A (fi) 1979-02-20
YU198678A (en) 1983-01-21
HK42282A (en) 1982-10-08
BR7805288A (pt) 1979-04-10
GB2003153A (en) 1979-03-07
DK152361C (da) 1988-07-25
AU521421B2 (en) 1982-04-01
ES472686A1 (es) 1979-03-16
DK366978A (da) 1979-02-20
MX5469E (es) 1983-08-16
PH13331A (en) 1980-03-13
AU3906178A (en) 1980-02-21
DK152361B (da) 1988-02-22
FR2400511B1 (fr) 1981-09-04
NZ188189A (en) 1984-07-06
GB2017678A (en) 1979-10-10
JPS5441873A (en) 1979-04-03
IE47430B1 (en) 1984-03-21
SE7808694L (sv) 1979-02-20
NL7808596A (nl) 1979-02-21
DE2836062A1 (de) 1979-03-01
NO149107C (no) 1984-02-22
SE451723B (sv) 1987-10-26
CA1105037A (fr) 1981-07-14

Similar Documents

Publication Publication Date Title
FR2400517A1 (fr) Triazolo-2,4-benzodiazepines et leur utilisation therapeutique
FR2417500A1 (fr) Derives d'amino-acides cycliques dehydrogenes et leur utilisation therapeutique
FR2446832A1 (fr) Octahydro-pyrazolo(3,4-g)quinoleines et leur utilisation therapeutique
FR2416891A1 (fr) 6-n-propyl-8-methoxymethyl ou methylmercaptomethylergolines et composes apparentes, et leur utilisation therapeutique
FR2430411A1 (fr) Phenethanolamines et leur utilisation therapeutique
FR2417510A1 (fr) 9-amino- et imino-dibenzopyrannes et leur utilisation therapeutique
FR2442845A1 (fr) Derives amines spiranniques, leur preparation et leur utilisation comme medicaments
FR2442836A1 (fr) 1,2,4,5-tetra-alkyl-4-arylpiperidines, leur preparation et leur utilisation therapeutique
FR2385682A1 (fr) Nouveaux 1-amino-indanes et leur utilisation comme medicaments
FR2430408A1 (fr) Phenethanolamines optiquement actives et leur utilisation therapeutique
FR2381762A1 (fr) Dibenzodiazepines utilisables comme antischizophreniques
TR20232A (tr) Cis-9-trikosen ve metomil'den olusan ensektisit bilesim
IT1079395B (it) Alchilammidi n-alchinil-(fenossi-sostituite)composizioni che le contengono e procedimento per produrle
FR2387989A1 (fr) Analogues des alcaloides de l'ergot
FR2378016A1 (fr) 1-alkylthiophenyl-2,3,4,5-tetrahydro-1h-3-benzazepine substituees et leur application en therapeutique
BR8004481A (pt) Composicoes de aclaradores oticos,sua obtencao e utilizacao
FR2400511A1 (fr) N-(4-pyrazolidinyl) benzamides, presentant notamment des proprietes antiemetiques et de vidage gastrique
FR2421613A1 (fr) Compositions contenant des benzamides de 3-aminopyrrolidines et leur utilisation therapeutique pour le traitement des allergies
FR2363541A1 (fr) Acyloxy-n,n' diacylmalonamides et leur mode de preparation
FR2399406A1 (fr) Derives de perhydronaphtalenepentol et leur utilisation therapeutique
FR2446833A1 (fr) Octahydro-2h-pyrrolo(3,4-g)quinoleines et leur utilisation therapeutiques
FR2428047A1 (fr) Arylalkyl- et aryloxyalkyl- phosphonates, leur preparation et leur utilisation therapeutique
IT1156188B (it) Composizioni furificate di urochinasi e procedimento per ottenerle
JO1120B1 (en) N- (1-night-2-pyrrolidinyl-methyl) 2-methoxy-4-amino-5-methylsulfamoyil benzamide, method of preparation and use as a drug
FR2360305A1 (fr) Nouveaux 2,3-alkylene bis (oxy)benzamides substitues, leurs derives et leurs procedes de preparation

Legal Events

Date Code Title Description
ST Notification of lapse