FI65238C - Foerfarande foer framstaellning av terapeutiskt anvaendbara teracykliska foereningar - Google Patents

Foerfarande foer framstaellning av terapeutiskt anvaendbara teracykliska foereningar Download PDF

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Publication number
FI65238C
FI65238C FI771635A FI771635A FI65238C FI 65238 C FI65238 C FI 65238C FI 771635 A FI771635 A FI 771635A FI 771635 A FI771635 A FI 771635A FI 65238 C FI65238 C FI 65238C
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FI
Finland
Prior art keywords
formula
compounds
alkyl
compound
test
Prior art date
Application number
FI771635A
Other languages
English (en)
Finnish (fi)
Other versions
FI65238B (fi
FI771635A (xx
Inventor
Willem Jacob Van Der Burg
Original Assignee
Akzo Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nv filed Critical Akzo Nv
Publication of FI771635A publication Critical patent/FI771635A/fi
Priority to FI832085A priority Critical patent/FI67701C/fi
Application granted granted Critical
Publication of FI65238B publication Critical patent/FI65238B/fi
Publication of FI65238C publication Critical patent/FI65238C/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/58[b]- or [c]-condensed
    • C07D209/70[b]- or [c]-condensed containing carbocyclic rings other than six-membered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04Ortho- or peri-condensed ring systems
    • C07D221/18Ring systems of four or more rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
FI771635A 1976-05-24 1977-05-23 Foerfarande foer framstaellning av terapeutiskt anvaendbara teracykliska foereningar FI65238C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI832085A FI67701C (fi) 1976-05-24 1983-06-09 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara tetracykliska foereningar

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
NL7605526A NL7605526A (nl) 1976-05-24 1976-05-24 Nieuwe tetracyclische derivaten.
NL7605526 1976-05-24

Publications (3)

Publication Number Publication Date
FI771635A FI771635A (xx) 1977-11-25
FI65238B FI65238B (fi) 1983-12-30
FI65238C true FI65238C (fi) 1984-04-10

Family

ID=19826245

Family Applications (1)

Application Number Title Priority Date Filing Date
FI771635A FI65238C (fi) 1976-05-24 1977-05-23 Foerfarande foer framstaellning av terapeutiskt anvaendbara teracykliska foereningar

Country Status (18)

Country Link
US (1) US4145434A (xx)
JP (2) JPS532465A (xx)
AU (1) AU509073B2 (xx)
BE (1) BE854915A (xx)
CA (1) CA1122976A (xx)
CH (2) CH633536A5 (xx)
DE (2) DE2723209A1 (xx)
DK (1) DK157868C (xx)
ES (3) ES459024A1 (xx)
FI (1) FI65238C (xx)
FR (1) FR2352800A1 (xx)
GB (1) GB1567862A (xx)
HU (1) HU173795B (xx)
IE (1) IE45419B1 (xx)
LU (1) LU77387A1 (xx)
NL (1) NL7605526A (xx)
SE (1) SE436202B (xx)
ZA (1) ZA772752B (xx)

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ATE9159T1 (de) * 1979-12-10 1984-09-15 Ciba-Geigy Ag Azatetracyclische carbonitrile.
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JPS62101941U (xx) * 1985-12-16 1987-06-29
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ATE233765T1 (de) * 1993-04-06 2003-03-15 Abbott Lab Tetracyclische verbindungen als dopamin-agonisten
KR100330942B1 (ko) * 1994-03-02 2002-11-16 악조 노벨 엔.브이. 설하또는협측투여용약학조성물
JP3274579B2 (ja) * 1995-01-12 2002-04-15 住友製薬株式会社 脳血管障害に伴う精神症候治療剤
KR100389298B1 (ko) * 1996-04-12 2003-10-30 얀센 파마슈티카 엔.브이. 치환된테트라사이클릭테트라하이드로퓨란유도체
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HRP20030959A2 (xx) * 2003-11-21 2005-10-31 Pliva-Istra�iva�ki institut d.o.o.
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CN103113379A (zh) * 2013-03-12 2013-05-22 盛世泰科生物医药技术(苏州)有限公司 阿塞那平马来酸盐的合成工艺
CN103351393B (zh) * 2013-07-03 2016-04-06 华裕(无锡)制药有限公司 用于制备阿森那平之还原剂及阿森那平之制备方法
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Also Published As

Publication number Publication date
IE45419B1 (en) 1982-08-25
CH633536A5 (de) 1982-12-15
CA1122976A (en) 1982-05-04
BE854915A (fr) 1977-11-23
FI65238B (fi) 1983-12-30
AU509073B2 (en) 1980-04-17
HU173795B (hu) 1979-08-28
DK157868B (da) 1990-02-26
CH637382A5 (de) 1983-07-29
JPS6238348B2 (xx) 1987-08-17
SE436202B (sv) 1984-11-19
FR2352800B1 (xx) 1980-02-01
FR2352800A1 (fr) 1977-12-23
ES470407A1 (es) 1979-01-01
DE2760372C2 (xx) 1991-05-29
US4145434A (en) 1979-03-20
SE7705957L (sv) 1977-11-25
JPS61178965A (ja) 1986-08-11
JPS6134426B2 (xx) 1986-08-07
LU77387A1 (xx) 1977-08-29
JPS532465A (en) 1978-01-11
ZA772752B (en) 1978-04-26
GB1567862A (en) 1980-05-21
AU2533177A (en) 1978-11-23
NL7605526A (nl) 1977-11-28
DE2723209A1 (de) 1977-12-15
IE45419L (en) 1977-11-24
ES459024A1 (es) 1978-11-01
DK157868C (da) 1990-07-30
FI771635A (xx) 1977-11-25
DK227477A (da) 1977-11-25
ES470408A1 (es) 1979-01-01

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