FI64366C - Analogifoerfarande foer framstaellning av antihypertensiva kinazolinderivat - Google Patents

Analogifoerfarande foer framstaellning av antihypertensiva kinazolinderivat Download PDF

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Publication number
FI64366C
FI64366C FI783347A FI783347A FI64366C FI 64366 C FI64366 C FI 64366C FI 783347 A FI783347 A FI 783347A FI 783347 A FI783347 A FI 783347A FI 64366 C FI64366 C FI 64366C
Authority
FI
Finland
Prior art keywords
formula
benzodioxane
quinazoline
mixture
group
Prior art date
Application number
FI783347A
Other languages
English (en)
Finnish (fi)
Other versions
FI783347A (fi
FI64366B (fi
Inventor
Simon Fraser Campbell
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI783347A publication Critical patent/FI783347A/fi
Application granted granted Critical
Publication of FI64366B publication Critical patent/FI64366B/fi
Publication of FI64366C publication Critical patent/FI64366C/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D319/00Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/101,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/141,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/161,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/201,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
FI783347A 1977-11-05 1978-11-02 Analogifoerfarande foer framstaellning av antihypertensiva kinazolinderivat FI64366C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB4612877 1977-11-05
GB4612877 1977-11-05

Publications (3)

Publication Number Publication Date
FI783347A FI783347A (fi) 1979-05-06
FI64366B FI64366B (fi) 1983-07-29
FI64366C true FI64366C (fi) 1983-11-10

Family

ID=10439957

Family Applications (1)

Application Number Title Priority Date Filing Date
FI783347A FI64366C (fi) 1977-11-05 1978-11-02 Analogifoerfarande foer framstaellning av antihypertensiva kinazolinderivat

Country Status (36)

Country Link
JP (1) JPS5498792A (el)
AR (2) AR219562A1 (el)
AT (1) AT365186B (el)
AU (1) AU509329B2 (el)
BE (1) BE871771A (el)
CA (1) CA1088059A (el)
CH (1) CH643255A5 (el)
CS (2) CS207671B2 (el)
DD (1) DD139850A5 (el)
DE (1) DE2847623C2 (el)
DK (1) DK154082C (el)
EG (1) EG13594A (el)
ES (2) ES474805A1 (el)
FI (1) FI64366C (el)
FR (1) FR2407929A1 (el)
GR (1) GR81514B (el)
HK (1) HK94284A (el)
HU (1) HU176306B (el)
IE (1) IE47888B1 (el)
IL (1) IL55857A (el)
IN (1) IN148828B (el)
IT (1) IT1100919B (el)
KE (1) KE3350A (el)
LU (2) LU80470A1 (el)
MY (1) MY8500286A (el)
NL (2) NL174549C (el)
NO (1) NO150158C (el)
NZ (1) NZ188813A (el)
PH (1) PH13966A (el)
PL (2) PL119419B1 (el)
PT (1) PT68735A (el)
SE (1) SE437518B (el)
SU (1) SU816403A3 (el)
UA (1) UA8324A1 (el)
YU (2) YU40204B (el)
ZA (1) ZA786184B (el)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1986002644A1 (en) * 1984-11-01 1986-05-09 Takeda Chemical Industries, Ltd. 1,5-benzoxathiepin derivatives and process for their preparation
WO1985004658A1 (en) * 1984-04-04 1985-10-24 Takeda Chemical Industries, Ltd. 1,5-benzoxathiepine derivatives and their preparation
WO1985002617A1 (en) * 1983-12-14 1985-06-20 Takeda Chemical Industries. Ltd. 1,5-benzoxathiepin derivatives and process for their preparation
PT849266E (pt) * 1996-12-20 2007-03-30 Heumann Pcs Gmbh Nova forma polimorfa de mesilato de doxazosina (forma iii)
EP0849265A1 (de) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Neue polymorphe Form von Doxazosin-Mesylat (Form II)
EP0849264A1 (de) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Neue polymorphe Form von doxazosinmesylat (Form I)
TW448155B (en) * 1999-03-29 2001-08-01 Dev Center Biotechnology Method for producing amide compounds and quinazolin derivatives
EP1403263B1 (en) * 2002-09-27 2005-06-22 Council of Scientific and Industrial Research Process for the preparation of N-(2,3-dihydrobenzo 1,4 dioxin-2-carbonyl) piperazine

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3663706A (en) * 1969-09-29 1972-05-16 Pfizer Use of 2,4-diaminoquinazolines as hypotensive agents
US3669968A (en) * 1970-05-21 1972-06-13 Pfizer Trialkoxy quinazolines

Also Published As

Publication number Publication date
DK154082C (da) 1989-02-27
NL7810909A (nl) 1979-05-08
YU255378A (en) 1983-06-30
AR223015A1 (es) 1981-07-15
FR2407929B1 (el) 1981-02-27
CS207671B2 (en) 1981-08-31
FR2407929A1 (fr) 1979-06-01
NL174549C (nl) 1984-07-02
IL55857A0 (en) 1979-01-31
ES8308559A1 (es) 1980-07-16
SE7811382L (sv) 1979-05-06
YU40204B (en) 1985-08-31
NL174549B (nl) 1984-02-01
AU509329B2 (en) 1980-05-08
YU38683A (en) 1983-06-30
ES480121A0 (es) 1980-07-16
MY8500286A (en) 1985-12-31
NO150158B (no) 1984-05-21
NZ188813A (en) 1980-10-08
PL119419B1 (en) 1981-12-31
AU4132278A (en) 1979-05-17
JPS5498792A (en) 1979-08-03
UA8324A1 (uk) 1996-03-29
IL55857A (en) 1982-07-30
FI783347A (fi) 1979-05-06
EG13594A (en) 1982-03-31
ATA784378A (de) 1981-05-15
CS354491A3 (en) 1992-06-17
YU40419B (en) 1985-12-31
NO783705L (no) 1979-05-08
NL930062I1 (nl) 1993-09-01
DE2847623C2 (de) 1983-06-01
FI64366B (fi) 1983-07-29
GR81514B (el) 1984-12-11
PH13966A (en) 1980-11-12
SE437518B (sv) 1985-03-04
DD139850A5 (de) 1980-01-23
KE3350A (en) 1983-12-16
AT365186B (de) 1981-12-28
IN148828B (el) 1981-06-27
CH643255A5 (en) 1984-05-30
IE782179L (en) 1979-05-05
LU80470A1 (fr) 1980-06-05
AR219562A1 (es) 1980-08-29
SU816403A3 (ru) 1981-03-23
IT7829434A0 (it) 1978-11-03
JPS5625233B2 (el) 1981-06-11
CA1088059A (en) 1980-10-21
HU176306B (en) 1981-01-28
DK428678A (da) 1979-05-06
ZA786184B (en) 1979-10-31
ES474805A1 (es) 1980-01-16
NL930062I2 (nl) 1993-11-16
IT1100919B (it) 1985-09-28
PT68735A (en) 1978-12-01
PL119586B1 (en) 1982-01-30
IE47888B1 (en) 1984-07-11
PL210681A1 (el) 1979-11-05
DK154082B (da) 1988-10-10
DE2847623A1 (de) 1979-05-23
HK94284A (en) 1984-12-07
NO150158C (no) 1984-08-29
LU88331I2 (fr) 1994-05-04
BE871771A (fr) 1979-05-03

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Owner name: PFIZER CORPORATION