FI63409C - Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 1,5-dihydro-imidazo(2,1-b)kinazolin-2(3h)-onderivat - Google Patents

Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 1,5-dihydro-imidazo(2,1-b)kinazolin-2(3h)-onderivat Download PDF

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Publication number
FI63409C
FI63409C FI782248A FI782248A FI63409C FI 63409 C FI63409 C FI 63409C FI 782248 A FI782248 A FI 782248A FI 782248 A FI782248 A FI 782248A FI 63409 C FI63409 C FI 63409C
Authority
FI
Finland
Prior art keywords
quinazolin
dihydro
chloro
formula
ethyl ester
Prior art date
Application number
FI782248A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI63409B (fi
FI782248A (fi
Inventor
Madhukar Subraya Chodnekar
Ado Kaiser
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of FI782248A publication Critical patent/FI782248A/fi
Publication of FI63409B publication Critical patent/FI63409B/fi
Application granted granted Critical
Publication of FI63409C publication Critical patent/FI63409C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
FI782248A 1977-07-25 1978-07-14 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 1,5-dihydro-imidazo(2,1-b)kinazolin-2(3h)-onderivat FI63409C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
LU77829 1977-07-25
LU77829 1977-07-25
CH577678 1978-05-26
CH577678 1978-05-26

Publications (3)

Publication Number Publication Date
FI782248A FI782248A (fi) 1979-01-26
FI63409B FI63409B (fi) 1983-02-28
FI63409C true FI63409C (fi) 1983-06-10

Family

ID=25698353

Family Applications (1)

Application Number Title Priority Date Filing Date
FI782248A FI63409C (fi) 1977-07-25 1978-07-14 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 1,5-dihydro-imidazo(2,1-b)kinazolin-2(3h)-onderivat

Country Status (29)

Country Link
US (1) US4256748A (nl)
EP (1) EP0000718B1 (nl)
JP (1) JPS5441894A (nl)
AR (1) AR218500A1 (nl)
AT (1) AT363479B (nl)
AU (1) AU519688B2 (nl)
BR (1) BR7804763A (nl)
CA (1) CA1094555A (nl)
CS (1) CS203014B2 (nl)
DE (2) DE2832138A1 (nl)
DK (1) DK144128C (nl)
ES (2) ES471981A1 (nl)
FI (1) FI63409C (nl)
FR (1) FR2398748A1 (nl)
GB (1) GB2001638B (nl)
GR (1) GR72968B (nl)
HU (1) HU177643B (nl)
IE (1) IE47280B1 (nl)
IL (1) IL55183A (nl)
IT (1) IT1097337B (nl)
MC (1) MC1199A1 (nl)
MY (1) MY8500249A (nl)
NL (1) NL7807507A (nl)
NO (1) NO150800C (nl)
NZ (1) NZ187921A (nl)
PH (1) PH14642A (nl)
PT (1) PT68342A (nl)
SE (1) SE7808111L (nl)
YU (1) YU177578A (nl)

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US4775674A (en) * 1986-05-23 1988-10-04 Bristol-Myers Company Imidazoquinolinylether derivatives useful as phosphodiesterase and blood aggregation inhibitors
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US5208237A (en) * 1992-04-03 1993-05-04 Bristol-Meyers Squibb Company 7-oxypropylsulfonamido-imidazo[4,5-b]quinolin-2-ones
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JPH06167328A (ja) * 1992-05-26 1994-06-14 Mayekawa Mfg Co Ltd 氷厚測定装置
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US6388073B1 (en) * 2000-07-26 2002-05-14 Shire Us Inc. Method for the manufacture of anagrelide
BRPI0406634A (pt) * 2003-01-23 2005-12-06 Shire Holding Ag Uso de um anagrelìdeo, anagrelìdeo na forma de base, ou um sal farmaceuticamente aceitável do anagrelìdeo, composição farmacêutica não-oral, e dispositivo médido para administração transdérmica
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US20060030574A1 (en) * 2004-08-04 2006-02-09 Shire Holdings Ag Quinazoline derivatives useful for the treatment of peripheral arterial disease and as phosphodiesterase inhibitors
US7700608B2 (en) * 2004-08-04 2010-04-20 Shire Holdings Ag Quinazoline derivatives and their use in the treatment of thrombocythemia
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US8436006B2 (en) * 2004-08-06 2013-05-07 Jansssen Pharmaceutica N.V. 2-amino-quinazoline derivatives useful as inhibitors of β-secretase (BACE)
US8383637B2 (en) 2004-08-06 2013-02-26 Jansssen Pharmaceutica N.V. 2-amino-quinazoline derivatives useful as inhibitors of β-secretase (BACE)
US8304420B2 (en) 2006-11-28 2012-11-06 Shire Llc Substituted quinazolines for reducing platelet count
US7910597B2 (en) 2006-11-28 2011-03-22 Shire Llc Substituted quinazolines
GB0623750D0 (en) * 2006-11-28 2007-01-10 Shire Llc Substituted quinazolines
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KR102272746B1 (ko) 2013-06-05 2021-07-08 보슈 헬스 아일랜드 리미티드 구아닐레이트 사이클라제 c의 초순수 작용제, 및 이의 제조 및 사용 방법
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JP5935843B2 (ja) * 2014-08-08 2016-06-15 Ｊｆｅスチール株式会社 スポット溶接性に優れた冷延鋼板およびその製造方法
CN114340631A (zh) 2019-05-21 2022-04-12 阿德利克斯股份有限公司 用于降低患者的血清磷酸盐的组合
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NL7807507A (nl) 1977-07-25 1979-01-29 Hoffmann La Roche Tricyclische verbindingen.

Also Published As

Publication number Publication date
IL55183A (en) 1981-11-30
EP0000718A3 (en) 1979-06-13
AU3812778A (en) 1980-01-24
CA1094555A (en) 1981-01-27
ATA535178A (de) 1981-01-15
EP0000718A2 (de) 1979-02-21
IT7826019A0 (it) 1978-07-24
IT1097337B (it) 1985-08-31
FR2398748A1 (fr) 1979-02-23
DE2832138A1 (de) 1979-02-08
AT363479B (de) 1981-08-10
NO782541L (no) 1979-01-26
DK328978A (da) 1979-01-26
FR2398748B1 (nl) 1981-09-04
MC1199A1 (fr) 1979-03-19
NO150800B (no) 1984-09-10
FI63409B (fi) 1983-02-28
AU519688B2 (en) 1981-12-17
AR218500A1 (es) 1980-06-13
DK144128B (da) 1981-12-14
DK144128C (da) 1982-05-17
GB2001638A (en) 1979-02-07
CS203014B2 (en) 1981-02-27
MY8500249A (en) 1985-12-31
PT68342A (en) 1978-08-01
ES471981A1 (es) 1979-10-16
IL55183A0 (en) 1978-09-29
NZ187921A (en) 1981-03-16
ES476955A1 (es) 1979-10-16
IE47280B1 (en) 1984-02-08
GB2001638B (en) 1982-02-10
DE2861688D1 (en) 1982-04-29
EP0000718B1 (de) 1982-03-24
FI782248A (fi) 1979-01-26
PH14642A (en) 1981-10-12
NO150800C (no) 1984-12-27
GR72968B (nl) 1984-01-20
NL7807507A (nl) 1979-01-29
YU177578A (en) 1983-01-21
JPS5441894A (en) 1979-04-03
SE7808111L (sv) 1979-01-26
US4256748A (en) 1981-03-17
BR7804763A (pt) 1979-04-10
HU177643B (en) 1981-11-28
IE781478L (en) 1979-01-25

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Owner name: F. HOFFMANN-LA ROCHE & CO.