AR218500A1 - Procedimiento para la obtencion de derivados de 1,5-dihidro-imidazo(2,1-b)quinazolin-2(3h)-ona 3-sustituidos - Google Patents

Procedimiento para la obtencion de derivados de 1,5-dihidro-imidazo(2,1-b)quinazolin-2(3h)-ona 3-sustituidos

Info

Publication number
AR218500A1
AR218500A1 AR273064A AR27306478A AR218500A1 AR 218500 A1 AR218500 A1 AR 218500A1 AR 273064 A AR273064 A AR 273064A AR 27306478 A AR27306478 A AR 27306478A AR 218500 A1 AR218500 A1 AR 218500A1
Authority
AR
Argentina
Prior art keywords
quinazolin
ona
imidazo
dihydro
substituted
Prior art date
Application number
AR273064A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of AR218500A1 publication Critical patent/AR218500A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
AR273064A 1977-07-25 1978-07-25 Procedimiento para la obtencion de derivados de 1,5-dihidro-imidazo(2,1-b)quinazolin-2(3h)-ona 3-sustituidos AR218500A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
LU77829 1977-07-25
CH577678 1978-05-26

Publications (1)

Publication Number Publication Date
AR218500A1 true AR218500A1 (es) 1980-06-13

Family

ID=25698353

Family Applications (1)

Application Number Title Priority Date Filing Date
AR273064A AR218500A1 (es) 1977-07-25 1978-07-25 Procedimiento para la obtencion de derivados de 1,5-dihidro-imidazo(2,1-b)quinazolin-2(3h)-ona 3-sustituidos

Country Status (29)

Country Link
US (1) US4256748A (es)
EP (1) EP0000718B1 (es)
JP (1) JPS5441894A (es)
AR (1) AR218500A1 (es)
AT (1) AT363479B (es)
AU (1) AU519688B2 (es)
BR (1) BR7804763A (es)
CA (1) CA1094555A (es)
CS (1) CS203014B2 (es)
DE (2) DE2832138A1 (es)
DK (1) DK144128C (es)
ES (2) ES471981A1 (es)
FI (1) FI63409C (es)
FR (1) FR2398748A1 (es)
GB (1) GB2001638B (es)
GR (1) GR72968B (es)
HU (1) HU177643B (es)
IE (1) IE47280B1 (es)
IL (1) IL55183A (es)
IT (1) IT1097337B (es)
MC (1) MC1199A1 (es)
MY (1) MY8500249A (es)
NL (1) NL7807507A (es)
NO (1) NO150800C (es)
NZ (1) NZ187921A (es)
PH (1) PH14642A (es)
PT (1) PT68342A (es)
SE (1) SE7808111L (es)
YU (1) YU177578A (es)

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US5158958A (en) * 1992-04-03 1992-10-27 Bristol-Myers Squibb Company Imidazo[4,5-b]quinolinyl oxy alkyl sulfonyl piperidine derivatives
US5208237A (en) * 1992-04-03 1993-05-04 Bristol-Meyers Squibb Company 7-oxypropylsulfonamido-imidazo[4,5-b]quinolin-2-ones
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US7910597B2 (en) 2006-11-28 2011-03-22 Shire Llc Substituted quinazolines
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
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JP5935843B2 (ja) * 2014-08-08 2016-06-15 Ｊｆｅスチール株式会社 スポット溶接性に優れた冷延鋼板およびその製造方法
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DE1645917A1 (de) 1962-10-26 1970-09-24 American Home Prod Verfahren zur Herstellung von 5-Aryl-3-acyloxy-1,2-dihydro-3H-1,4-benzodiazepin-2-onen
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NL7807507A (nl) 1977-07-25 1979-01-29 Hoffmann La Roche Tricyclische verbindingen.

Also Published As

Publication number Publication date
EP0000718A3 (en) 1979-06-13
CS203014B2 (en) 1981-02-27
ATA535178A (de) 1981-01-15
DE2861688D1 (en) 1982-04-29
HU177643B (en) 1981-11-28
NO782541L (no) 1979-01-26
FI63409B (fi) 1983-02-28
DK144128B (da) 1981-12-14
FI782248A (fi) 1979-01-26
NO150800B (no) 1984-09-10
US4256748A (en) 1981-03-17
DK328978A (da) 1979-01-26
IE781478L (en) 1979-01-25
GB2001638A (en) 1979-02-07
IE47280B1 (en) 1984-02-08
IT7826019A0 (it) 1978-07-24
EP0000718A2 (de) 1979-02-21
PH14642A (en) 1981-10-12
IL55183A (en) 1981-11-30
SE7808111L (sv) 1979-01-26
ES471981A1 (es) 1979-10-16
YU177578A (en) 1983-01-21
PT68342A (en) 1978-08-01
FI63409C (fi) 1983-06-10
CA1094555A (en) 1981-01-27
MY8500249A (en) 1985-12-31
AU3812778A (en) 1980-01-24
JPS5441894A (en) 1979-04-03
GB2001638B (en) 1982-02-10
IL55183A0 (en) 1978-09-29
AT363479B (de) 1981-08-10
AU519688B2 (en) 1981-12-17
FR2398748A1 (fr) 1979-02-23
MC1199A1 (fr) 1979-03-19
NL7807507A (nl) 1979-01-29
NO150800C (no) 1984-12-27
FR2398748B1 (es) 1981-09-04
NZ187921A (en) 1981-03-16
DK144128C (da) 1982-05-17
IT1097337B (it) 1985-08-31
DE2832138A1 (de) 1979-02-08
ES476955A1 (es) 1979-10-16
GR72968B (es) 1984-01-20
BR7804763A (pt) 1979-04-10
EP0000718B1 (de) 1982-03-24

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