FI60010C - Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 4-(2-imidazolin-2-ylamino)-2,1,3-bensotiadiazoler - Google Patents

Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 4-(2-imidazolin-2-ylamino)-2,1,3-bensotiadiazoler Download PDF

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Publication number
FI60010C
FI60010C FI1393/73A FI139373A FI60010C FI 60010 C FI60010 C FI 60010C FI 1393/73 A FI1393/73 A FI 1393/73A FI 139373 A FI139373 A FI 139373A FI 60010 C FI60010 C FI 60010C
Authority
FI
Finland
Prior art keywords
formula
benzothiadiazole
ylamino
imidazolin
methyl
Prior art date
Application number
FI1393/73A
Other languages
English (en)
Finnish (fi)
Other versions
FI60010B (fi
Inventor
Peter Neumann
Original Assignee
Wander Ag Dr A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wander Ag Dr A filed Critical Wander Ag Dr A
Application granted granted Critical
Publication of FI60010B publication Critical patent/FI60010B/fi
Publication of FI60010C publication Critical patent/FI60010C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/14—Thiadiazoles; Hydrogenated thiadiazoles condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
FI1393/73A 1972-05-09 1973-05-02 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 4-(2-imidazolin-2-ylamino)-2,1,3-bensotiadiazoler FI60010C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH686572 1972-05-09
CH686572A CH570401A5 (cs) 1972-05-09 1972-05-09

Publications (2)

Publication Number Publication Date
FI60010B FI60010B (fi) 1981-07-31
FI60010C true FI60010C (fi) 1981-11-10

Family

ID=4316243

Family Applications (1)

Application Number Title Priority Date Filing Date
FI1393/73A FI60010C (fi) 1972-05-09 1973-05-02 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 4-(2-imidazolin-2-ylamino)-2,1,3-bensotiadiazoler

Country Status (26)

Country Link
US (1) US3843668A (cs)
JP (3) JPS5533718B2 (cs)
AT (1) AT336006B (cs)
BE (1) BE799332A (cs)
CH (1) CH570401A5 (cs)
CS (2) CS202052B2 (cs)
CY (1) CY989A (cs)
DD (1) DD106180A5 (cs)
DE (1) DE2322880C2 (cs)
DK (1) DK135454B (cs)
ES (3) ES414470A1 (cs)
FI (1) FI60010C (cs)
FR (1) FR2183930B1 (cs)
GB (2) GB1429683A (cs)
HK (1) HK11179A (cs)
HU (1) HU166329B (cs)
IE (1) IE38012B1 (cs)
IL (2) IL49205A (cs)
MY (1) MY7900117A (cs)
NL (1) NL161445C (cs)
NO (1) NO138566C (cs)
PL (1) PL89214B1 (cs)
SE (1) SE386445B (cs)
SU (1) SU493966A3 (cs)
YU (4) YU36174B (cs)
ZA (1) ZA733143B (cs)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5930899B2 (ja) * 1973-02-01 1984-07-30 隆弘 上野 内燃機関の制動方法及びその装置
GB1559811A (en) * 1975-07-28 1980-01-30 Sandoz Ltd Pharmaceutically active benzothiadiazole derivatives
US4217356A (en) * 1975-08-22 1980-08-12 Sandoz Ltd. 2-Imidazolinylamino-2,1,3-benzothiadiazoles
CH613966A5 (en) * 1975-08-22 1979-10-31 Sandoz Ag Process for the preparation of novel 5-(2-imidazolin-2-ylamino)-2,1,3-benzothiadiazoles
CH632268A5 (de) * 1977-01-14 1982-09-30 Sandoz Ag Verfahren zur herstellung von neuen heterocyclylaminoderivaten.
FR2499991A1 (fr) * 1981-02-19 1982-08-20 Sandoz Sa Nouveaux 2,1,3-benzothiadiazoles et 2,1,3-benzoxadiazoles, leur preparation et leur application comme medicaments
FR2502951B1 (fr) * 1981-04-06 1985-12-06 Sandoz Sa Compositions pharmaceutiques topiques sous forme d'une micro-emulsion
JPS61268828A (ja) * 1985-05-22 1986-11-28 Kubota Ltd 圧縮空気取出装置付き容積形内燃機関
JPH0622121Y2 (ja) * 1988-01-18 1994-06-08 川崎重工業株式会社 空気圧縮機兼用多気筒エンジン
JP2668816B2 (ja) * 1993-09-09 1997-10-27 株式会社パーマケム・アジア ベンゾチアジアゾール誘導体の製法
US6455557B1 (en) 2001-11-28 2002-09-24 Elan Pharmaceuticals, Inc. Method of reducing somnolence in patients treated with tizanidine
US20040220240A1 (en) * 2001-11-28 2004-11-04 Pellegrini Cara A. Method of increasing the extent of absorption of tizanidine
EP2316468A1 (en) 2002-02-22 2011-05-04 Shire LLC Delivery system and methods for protecting and administering dextroamphetamine
GB0224198D0 (en) * 2002-10-17 2002-11-27 Novartis Ag Organic compounds
RU2234506C1 (ru) * 2003-06-05 2004-08-20 Федеральное государственное унитарное предприятие "Государственный научный центр "Научно-исследовательский институт органических полупродуктов и красителей" Способ получения 5-хлор-4-/(2-имидазолин-2-ил)амино/-2,1,3-бензотиадиазола хлоргидрата
TWI435729B (zh) 2005-11-09 2014-05-01 Combinatorx Inc 治療病症之方法，組合物及套組
WO2008008394A1 (en) * 2006-07-12 2008-01-17 Transform Pharmaceuticals, Inc. Tizanidine succinate salt forms and methods of making and using the same
US8524749B2 (en) * 2007-02-09 2013-09-03 Alza Corporation Controlled release compositions of tizanidine
CZ301889B6 (cs) 2008-12-18 2010-07-21 Farmak, A. S. Zpusob prípravy tizanidinu hydrochloridu
US8980298B2 (en) * 2011-10-24 2015-03-17 Braeburn Pharmaceuticals Bvba Sprl Implantable tizanidine compositions and methods of treatment thereof
CN106946874A (zh) * 2017-04-07 2017-07-14 四川智强医药科技开发有限公司 替扎尼定的脱色方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1211341A (fr) * 1955-12-19 1960-03-15 A Wander Dr Procédé pour la préparation de 2-amino-imidazolines
BE754832A (fr) * 1969-08-14 1971-02-15 Beecham Group Ltd Iminazolines

Also Published As

Publication number Publication date
ZA733143B (en) 1975-01-29
JPS5543081A (en) 1980-03-26
CS208788B2 (en) 1981-09-15
DK135454C (cs) 1977-10-17
HU166329B (cs) 1975-02-28
YU36025B (en) 1981-11-13
ES440599A1 (es) 1977-05-16
JPS5350168A (en) 1978-05-08
YU36024B (en) 1981-11-13
NO138566C (no) 1978-09-27
JPS5533718B2 (cs) 1980-09-02
CH570401A5 (cs) 1975-12-15
GB1429926A (en) 1976-03-31
CY989A (en) 1979-08-02
DK135454B (da) 1977-05-02
YU50579A (en) 1981-04-30
NL7306228A (cs) 1973-11-13
DD106180A5 (cs) 1974-06-05
FI60010B (fi) 1981-07-31
YU36174B (en) 1982-02-25
JPS562071B2 (cs) 1981-01-17
AT336006B (de) 1977-04-12
IE38012B1 (en) 1977-12-07
JPS5442983B2 (cs) 1979-12-17
YU36026B (en) 1981-11-13
HK11179A (en) 1979-03-16
JPS4954370A (cs) 1974-05-27
FR2183930B1 (cs) 1976-03-05
ES414470A1 (es) 1976-05-01
IL49205A (en) 1977-05-31
YU119673A (en) 1981-06-30
MY7900117A (en) 1979-12-31
DE2322880C2 (de) 1982-09-23
SE386445B (sv) 1976-08-09
FR2183930A1 (cs) 1973-12-21
NL161445B (nl) 1979-09-17
NO138566B (no) 1978-06-19
SU493966A3 (ru) 1975-11-28
GB1429683A (en) 1976-03-24
BE799332A (fr) 1973-11-09
ES440598A1 (es) 1977-05-16
PL89214B1 (cs) 1976-11-30
ATA403273A (de) 1976-08-15
US3843668A (en) 1974-10-22
YU50479A (en) 1981-04-30
DE2322880A1 (de) 1973-11-22
AU5540873A (en) 1974-11-14
NL161445C (nl) 1980-02-15
IL49205A0 (en) 1976-05-31
IL42231A0 (en) 1973-07-30
IL42231A (en) 1977-06-30
CS202052B2 (en) 1980-12-31
IE38013L (en) 1973-11-09
YU50679A (en) 1981-04-30

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