FI59590C - Foerfarande foer framstaellning av terapeutiskt aktiva substituerade bensimidazoler eller syraadditionssalter daerav - Google Patents

Foerfarande foer framstaellning av terapeutiskt aktiva substituerade bensimidazoler eller syraadditionssalter daerav Download PDF

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Publication number
FI59590C
FI59590C FI750421A FI750421A FI59590C FI 59590 C FI59590 C FI 59590C FI 750421 A FI750421 A FI 750421A FI 750421 A FI750421 A FI 750421A FI 59590 C FI59590 C FI 59590C
Authority
FI
Finland
Prior art keywords
group
het
compound
general formula
alkanoyl
Prior art date
Application number
FI750421A
Other languages
English (en)
Finnish (fi)
Other versions
FI750421A (xx
FI59590B (fi
Inventor
Peder Bernhard Berntsson
Stig Aoke Ingemar Carlsson
Lars Erik Garberg
Ulf Krister Junggren
Sven Erik Sjoestrand
Sundell Gunhild Wika V Wittken
Original Assignee
Haessle Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Haessle Ab filed Critical Haessle Ab
Publication of FI750421A publication Critical patent/FI750421A/fi
Publication of FI59590B publication Critical patent/FI59590B/fi
Application granted granted Critical
Publication of FI59590C publication Critical patent/FI59590C/fi

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
FI750421A 1974-02-18 1975-02-14 Foerfarande foer framstaellning av terapeutiskt aktiva substituerade bensimidazoler eller syraadditionssalter daerav FI59590C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE7402101 1974-02-18
SE7402101A SE418966B (sv) 1974-02-18 1974-02-18 Analogiforfarande for framstellning av foreningar med magsyrasekretionsinhiberande verkan

Publications (3)

Publication Number Publication Date
FI750421A FI750421A (xx) 1975-08-19
FI59590B FI59590B (fi) 1981-05-29
FI59590C true FI59590C (fi) 1981-09-10

Family

ID=20320233

Family Applications (1)

Application Number Title Priority Date Filing Date
FI750421A FI59590C (fi) 1974-02-18 1975-02-14 Foerfarande foer framstaellning av terapeutiskt aktiva substituerade bensimidazoler eller syraadditionssalter daerav

Country Status (23)

Country Link
JP (1) JPS5924157B2 (xx)
AT (1) AT343659B (xx)
AU (1) AU499639B2 (xx)
BE (1) BE825655A (xx)
CA (1) CA1060448A (xx)
CH (1) CH616160A5 (xx)
CS (1) CS194715B2 (xx)
DD (1) DD119422A5 (xx)
DE (1) DE2504252A1 (xx)
DK (1) DK141122B (xx)
FI (1) FI59590C (xx)
FR (1) FR2261007B1 (xx)
GB (1) GB1500043A (xx)
HK (1) HK67080A (xx)
HU (1) HU172141B (xx)
IE (1) IE40858B1 (xx)
LU (1) LU71872A1 (xx)
MY (1) MY8100208A (xx)
NL (1) NL7501917A (xx)
NO (1) NO142401C (xx)
SE (1) SE418966B (xx)
SU (1) SU795476A3 (xx)
ZA (1) ZA75558B (xx)

Families Citing this family (42)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE416649B (sv) * 1974-05-16 1981-01-26 Haessle Ab Forfarande for framstellning av foreningar som paverkar magsyrasekretionen
JPS5364103A (en) * 1976-09-24 1978-06-08 Hitachi Ltd Waste heat recovery boiler
IN148930B (xx) 1977-09-19 1981-07-25 Hoffmann La Roche
SE7804231L (sv) * 1978-04-14 1979-10-15 Haessle Ab Magsyrasekretionsmedel
US4343805A (en) * 1978-12-16 1982-08-10 John Wyeth & Brother Limited Heterocyclic compounds
CH644116A5 (de) * 1980-08-21 1984-07-13 Hoffmann La Roche Imidazolderivate.
DE3047388A1 (de) * 1980-12-16 1982-07-15 Basf Ag, 6700 Ludwigshafen Isatogenderivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide
IL66340A (en) * 1981-08-13 1986-08-31 Haessle Ab Pharmaceutical compositions comprising pyridylmethyl-thiobenzimidazole derivatives,certain such novel derivatives and their preparation
DE3216843C2 (de) * 1982-05-05 1986-10-23 Ludwig Heumann & Co GmbH, 8500 Nürnberg 3-Thiomethyl-pyridin-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
US4552886A (en) * 1982-06-07 1985-11-12 Eli Lilly And Company Fungicidal pyridylmethyl-amines
SE8300736D0 (sv) * 1983-02-11 1983-02-11 Haessle Ab Novel pharmacologically active compounds
GB8307865D0 (en) * 1983-03-22 1983-04-27 Fujisawa Pharmaceutical Co Benzimidazole derivatives
US4503139A (en) * 1983-05-09 1985-03-05 Polaroid Corporation Photographic products and processes and novel compounds
US4575554A (en) * 1983-12-05 1986-03-11 The Upjohn Company Substituted 2-pyridylmethylthio- and sulfinyl-benzimidazoles as gastric antisecretory agents
US4767770A (en) * 1984-06-18 1988-08-30 Eli Lilly And Company Method of inhibiting aromatase
SE8505112D0 (sv) * 1985-10-29 1985-10-29 Haessle Ab Novel pharmacological compounds
FR2593178B1 (fr) * 1986-01-20 1988-04-29 Esteve Labor Dr Derives de 2-benzimidazolylalkylthio (ou sulfinyle ou sulfonyle) leur preparation et leur application en tant que medicaments.
SE8600658D0 (sv) * 1986-02-14 1986-02-14 Haessle Ab Novel composition of matter
SE8604566D0 (sv) * 1986-10-27 1986-10-27 Haessle Ab Novel compunds
SE8604998D0 (sv) 1986-11-21 1986-11-21 Haessle Ab Novel pharmacological compounds
NZ234564A (en) 1986-11-21 1991-04-26 Haessle Ab 1-substituted benzimidazoles and pharmaceutical compositions
WO1989005643A1 (en) * 1987-12-18 1989-06-29 Pfizer Inc. Heterocyclic-substituted quinoline-carboxylic acids
JPH021280U (xx) * 1988-06-14 1990-01-08
KR920003928B1 (ko) * 1988-09-20 1992-05-18 히사미쯔세이야꾸 가부시기가이샤 신규의 디벤즈[b,e]옥세핀유도체
SE8804629D0 (sv) 1988-12-22 1988-12-22 Ab Haessle New therapeutically active compounds
IE64199B1 (en) * 1988-12-22 1995-07-12 Haessle Ab Compound with gastric acid inhibitory effect and process for its preparation
SE8804628D0 (sv) 1988-12-22 1988-12-22 Ab Haessle New compounds
JP2679745B2 (ja) * 1989-06-29 1997-11-19 明治製菓株式会社 アゾール誘導体及びそれらを有効成分とする抗潰瘍剤
JPH0347053U (xx) * 1989-09-16 1991-04-30
US5049674A (en) 1989-12-20 1991-09-17 Aktiebolaget Hassle Therapeutically active fluoro substituted benzimidazoles
US5274099A (en) * 1989-12-20 1993-12-28 Aktiebolaget Hassle Therapeutically active fluoro substituted benzimidazoles
US4965269A (en) * 1989-12-20 1990-10-23 Ab Hassle Therapeutically active chloro substituted benzimidazoles
SE9002206D0 (sv) 1990-06-20 1990-06-20 Haessle Ab New compounds
PL372409A1 (en) 2002-03-27 2005-07-25 Altana Pharma Ag Novel alkoxypyridine-derivatives
CN1751043A (zh) 2003-02-25 2006-03-22 奥坦纳医药公司 咪唑并(4,5－b)喹啉衍生物及其作为no－合酶抑制剂的应用
ATE399168T1 (de) 2003-10-01 2008-07-15 Nycomed Gmbh Imidazopyridin-derivate und ihre verwendung als induzierbare no-synthase inhibitoren
KR20060092221A (ko) 2003-10-01 2006-08-22 알타나 파마 아게 유도성 ｎｏ-신타제 억제제로서의이미다조（4,5-ｂ）피리딘 유도체
EA010261B1 (ru) * 2003-10-01 2008-06-30 Алтана Фарма Аг Производные имидазопиридина как ингибиторы индуцируемой no - синтазы
US20080125460A1 (en) * 2003-10-01 2008-05-29 Altana Pharma Ag Imidazopyridine-Derivatives As Inducible No-Synthase Inhibitors
NZ546394A (en) * 2003-10-01 2009-08-28 Altana Pharma Ag Aminopyridine derivatives as inductible NO-synthase inhibitors
EP2070923A1 (de) 2007-12-11 2009-06-17 Bayer CropScience AG Insektizide Iminoheterocyclen
JP5911476B2 (ja) * 2010-05-26 2016-04-27 スノビオン プハルマセウトイカルス インコーポレイテッド ヘテロアリール化合物及びその使用方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1234058A (xx) * 1968-10-21 1971-06-03

Also Published As

Publication number Publication date
DE2504252C2 (xx) 1989-02-02
DK141122C (xx) 1980-07-07
FI750421A (xx) 1975-08-19
JPS5924157B2 (ja) 1984-06-07
FI59590B (fi) 1981-05-29
DD119422A5 (xx) 1976-04-20
DK141122B (da) 1980-01-21
DK54075A (xx) 1975-10-20
HK67080A (en) 1980-12-05
ZA75558B (en) 1976-01-28
AU499639B2 (en) 1979-04-26
SE418966B (sv) 1981-07-06
NO142401C (no) 1980-08-13
NO142401B (no) 1980-05-05
CA1060448A (en) 1979-08-14
ATA113775A (de) 1977-10-15
LU71872A1 (xx) 1975-12-09
CS194715B2 (en) 1979-12-31
SU795476A3 (ru) 1981-01-07
IE40858B1 (en) 1979-08-29
GB1500043A (en) 1978-02-08
IE40858L (en) 1975-08-18
AT343659B (de) 1978-06-12
AU7820675A (en) 1976-08-19
FR2261007A1 (xx) 1975-09-12
SE7402101L (xx) 1975-08-19
FR2261007B1 (xx) 1978-11-24
BE825655A (fr) 1975-08-18
DE2504252A1 (de) 1975-08-21
HU172141B (hu) 1978-06-28
NO750541L (xx) 1975-08-19
JPS50116474A (en) 1975-09-11
MY8100208A (en) 1981-12-31
CH616160A5 (en) 1980-03-14
NL7501917A (nl) 1975-08-20

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MM Patent lapsed

Owner name: AB HAESSLE