FI110000B - Menetelmä 3-{2-[4-(6-fluori-bentso[d]-isoksatsol-3-yyli)piperidin-1-yyli]-etyyli}-2-metyyli-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-onin saamiseksi - Google Patents

Menetelmä 3-{2-[4-(6-fluori-bentso[d]-isoksatsol-3-yyli)piperidin-1-yyli]-etyyli}-2-metyyli-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-onin saamiseksi Download PDF

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Publication number
FI110000B
FI110000B FI950579A FI950579A FI110000B FI 110000 B FI110000 B FI 110000B FI 950579 A FI950579 A FI 950579A FI 950579 A FI950579 A FI 950579A FI 110000 B FI110000 B FI 110000B
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FI
Finland
Prior art keywords
tetrahydro
methyl
pyrido
pyrimidin
fluoro
Prior art date
Application number
FI950579A
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English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI950579A0 (fi
FI950579A (fi
Inventor
Barjoan Pere Dalmases
Olondriz Francisco Marquillas
Clotet Joan Huguet
Rovira Ana Bosch
Castillo Nieto Juan Carlos Del
Ges Jose Maria Caldero
Original Assignee
Vita Invest Sa
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Publication date
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Publication of FI950579A0 publication Critical patent/FI950579A0/fi
Publication of FI950579A publication Critical patent/FI950579A/fi
Application granted granted Critical
Publication of FI110000B publication Critical patent/FI110000B/fi

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI950579A 1994-02-11 1995-02-10 Menetelmä 3-{2-[4-(6-fluori-bentso[d]-isoksatsol-3-yyli)piperidin-1-yyli]-etyyli}-2-metyyli-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-onin saamiseksi FI110000B (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES9400252 1994-02-11
ES09400252A ES2074966B1 (es) 1994-02-11 1994-02-11 Procedimiento para la obtencion de 3-(2-(4-(6-fluoro-benzo(d)isoxazol-3-il)piperidin-1-il)-etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido-(1,2-a)pirimidin-4-ona.

Publications (3)

Publication Number Publication Date
FI950579A0 FI950579A0 (fi) 1995-02-10
FI950579A FI950579A (fi) 1995-08-12
FI110000B true FI110000B (fi) 2002-11-15

Family

ID=8285178

Family Applications (1)

Application Number Title Priority Date Filing Date
FI950579A FI110000B (fi) 1994-02-11 1995-02-10 Menetelmä 3-{2-[4-(6-fluori-bentso[d]-isoksatsol-3-yyli)piperidin-1-yyli]-etyyli}-2-metyyli-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-onin saamiseksi

Country Status (14)

Country Link
KR (1) KR100221108B1 (ru)
AT (1) AT405401B (ru)
CZ (1) CZ286398B6 (ru)
EG (1) EG20877A (ru)
ES (1) ES2074966B1 (ru)
FI (1) FI110000B (ru)
GR (1) GR1002344B (ru)
HU (1) HU222110B1 (ru)
IS (1) IS1766B (ru)
NO (1) NO306022B1 (ru)
PL (1) PL181420B1 (ru)
PT (1) PT101654B (ru)
RU (1) RU2123004C1 (ru)
SK (1) SK281752B6 (ru)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2101646B1 (es) * 1995-04-12 1998-04-01 Ferrer Int Nuevo compuesto derivado del cromeno.
ES2144355B1 (es) * 1997-12-30 2001-01-01 Ferrer Int Compuestos derivados del cromeno.
EP1280804B1 (en) * 2000-05-05 2004-04-14 RPG Life Sciences Limited A process for the preparation of anti-psychotic 3- 2- 4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4h-pyrido 1,2,-a]pyrimidin-4-one
EP1317434A4 (en) 2000-08-14 2005-06-22 Teva Pharma PREPARATION OF RISPERIDONE
KR20040034996A (ko) 2002-10-18 2004-04-29 한미약품 주식회사 리스페리돈의 개선된 제조방법
EP1560814A1 (en) 2002-11-13 2005-08-10 Synthon B.V. Process for making risperidone and intermediates therefor
JP5315336B2 (ja) * 2007-04-19 2013-10-16 又欣 李 精神疾患治療用の新規化合物とその調剤及び使用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4352811A (en) * 1981-11-12 1982-10-05 Hoechst-Roussel Pharmaceuticals Inc. 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4980365A (en) * 1987-07-13 1990-12-25 Hoechst-Roussel Pharmaceuticals Inc. N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents

Also Published As

Publication number Publication date
FI950579A0 (fi) 1995-02-10
RU95101859A (ru) 1997-03-20
HU9500418D0 (en) 1995-03-28
NO950501D0 (no) 1995-02-09
SK15695A3 (en) 1995-10-11
KR100221108B1 (ko) 1999-09-15
PT101654A (pt) 1995-09-12
PL307200A1 (en) 1995-08-21
CZ32995A3 (en) 1995-09-13
ATA24995A (de) 1998-12-15
SK281752B6 (sk) 2001-07-10
EG20877A (en) 2000-05-31
ES2074966B1 (es) 1996-06-16
NO950501L (no) 1995-08-14
HUT70169A (en) 1995-09-28
AT405401B (de) 1999-08-25
CZ286398B6 (en) 2000-04-12
RU2123004C1 (ru) 1998-12-10
PL181420B1 (pl) 2001-07-31
KR950032196A (ko) 1995-12-20
GR1002344B (el) 1996-05-24
HU222110B1 (hu) 2003-04-28
NO306022B1 (no) 1999-09-06
ES2074966A1 (es) 1995-09-16
FI950579A (fi) 1995-08-12
IS1766B (is) 2001-03-15
IS4259A (is) 1995-08-12
PT101654B (pt) 2002-01-30

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