FI950579A - Menetelmä valmistaa 3-(2-(4-(6-fluori-bentso/D/-isoksatsol-3-yyli)piperidiini-1-iili/-etyyli)-2-metyyli-6,7,8,9-tetrahydro-4H-pyrido/1,2-A/pyrimidin-4-onia - Google Patents

Menetelmä valmistaa 3-(2-(4-(6-fluori-bentso/D/-isoksatsol-3-yyli)piperidiini-1-iili/-etyyli)-2-metyyli-6,7,8,9-tetrahydro-4H-pyrido/1,2-A/pyrimidin-4-onia Download PDF

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Publication number
FI950579A
FI950579A FI950579A FI950579A FI950579A FI 950579 A FI950579 A FI 950579A FI 950579 A FI950579 A FI 950579A FI 950579 A FI950579 A FI 950579A FI 950579 A FI950579 A FI 950579A
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FI
Finland
Prior art keywords
fluorobenzo
isoxazol
pyrido
pyrimidin
piperidin
Prior art date
Application number
FI950579A
Other languages
English (en)
Swedish (sv)
Other versions
FI950579A0 (fi
FI110000B (fi
Inventor
Barjoan Pere Dalmases
Olondriz Francisco Marquillas
Clotet Joan Huguet
Rovira Ana Bosch
Castillo Nieto Juan Carlos Del
Ges Jose Maria Caldero
Original Assignee
Vita Invest Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Vita Invest Sa filed Critical Vita Invest Sa
Publication of FI950579A0 publication Critical patent/FI950579A0/fi
Publication of FI950579A publication Critical patent/FI950579A/fi
Application granted granted Critical
Publication of FI110000B publication Critical patent/FI110000B/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI950579A 1994-02-11 1995-02-10 Menetelmä 3-{2-[4-(6-fluori-bentso[d]-isoksatsol-3-yyli)piperidin-1-yyli]-etyyli}-2-metyyli-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-onin saamiseksi FI110000B (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES9400252 1994-02-11
ES09400252A ES2074966B1 (es) 1994-02-11 1994-02-11 Procedimiento para la obtencion de 3-(2-(4-(6-fluoro-benzo(d)isoxazol-3-il)piperidin-1-il)-etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido-(1,2-a)pirimidin-4-ona.

Publications (3)

Publication Number Publication Date
FI950579A0 FI950579A0 (fi) 1995-02-10
FI950579A true FI950579A (fi) 1995-08-12
FI110000B FI110000B (fi) 2002-11-15

Family

ID=8285178

Family Applications (1)

Application Number Title Priority Date Filing Date
FI950579A FI110000B (fi) 1994-02-11 1995-02-10 Menetelmä 3-{2-[4-(6-fluori-bentso[d]-isoksatsol-3-yyli)piperidin-1-yyli]-etyyli}-2-metyyli-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-onin saamiseksi

Country Status (14)

Country Link
KR (1) KR100221108B1 (fi)
AT (1) AT405401B (fi)
CZ (1) CZ286398B6 (fi)
EG (1) EG20877A (fi)
ES (1) ES2074966B1 (fi)
FI (1) FI110000B (fi)
GR (1) GR1002344B (fi)
HU (1) HU222110B1 (fi)
IS (1) IS1766B (fi)
NO (1) NO306022B1 (fi)
PL (1) PL181420B1 (fi)
PT (1) PT101654B (fi)
RU (1) RU2123004C1 (fi)
SK (1) SK281752B6 (fi)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2101646B1 (es) * 1995-04-12 1998-04-01 Ferrer Int Nuevo compuesto derivado del cromeno.
ES2144355B1 (es) * 1997-12-30 2001-01-01 Ferrer Int Compuestos derivados del cromeno.
EP1280804B1 (en) * 2000-05-05 2004-04-14 RPG Life Sciences Limited A process for the preparation of anti-psychotic 3- 2- 4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4h-pyrido 1,2,-a]pyrimidin-4-one
ATE401313T1 (de) 2000-08-14 2008-08-15 Teva Pharma Herstellung von risperidon
KR20040034996A (ko) 2002-10-18 2004-04-29 한미약품 주식회사 리스페리돈의 개선된 제조방법
WO2004043923A1 (en) 2002-11-13 2004-05-27 Synthon B.V. Process for making risperidone and intermediates therefor
RU2459824C2 (ru) * 2007-04-19 2012-08-27 Юсинь ЛИ Новые соединения для лечения психических расстройств, их получение и применение

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4352811A (en) * 1981-11-12 1982-10-05 Hoechst-Roussel Pharmaceuticals Inc. 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4980365A (en) * 1987-07-13 1990-12-25 Hoechst-Roussel Pharmaceuticals Inc. N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents

Also Published As

Publication number Publication date
NO950501D0 (no) 1995-02-09
KR100221108B1 (ko) 1999-09-15
PL181420B1 (pl) 2001-07-31
FI950579A0 (fi) 1995-02-10
PT101654A (pt) 1995-09-12
HU9500418D0 (en) 1995-03-28
RU2123004C1 (ru) 1998-12-10
ATA24995A (de) 1998-12-15
PT101654B (pt) 2002-01-30
CZ286398B6 (en) 2000-04-12
RU95101859A (ru) 1997-03-20
NO950501L (no) 1995-08-14
HU222110B1 (hu) 2003-04-28
NO306022B1 (no) 1999-09-06
KR950032196A (ko) 1995-12-20
GR1002344B (el) 1996-05-24
SK15695A3 (en) 1995-10-11
IS4259A (is) 1995-08-12
IS1766B (is) 2001-03-15
SK281752B6 (sk) 2001-07-10
FI110000B (fi) 2002-11-15
EG20877A (en) 2000-05-31
PL307200A1 (en) 1995-08-21
HUT70169A (en) 1995-09-28
ES2074966A1 (es) 1995-09-16
ES2074966B1 (es) 1996-06-16
CZ32995A3 (en) 1995-09-13
AT405401B (de) 1999-08-25

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