RU93045711A - Нейролептические пергидро-1h-пиридо(1,2-a)пиразины, способ их получения, фармацевтическая композиция, способ лечения - Google Patents
Нейролептические пергидро-1h-пиридо(1,2-a)пиразины, способ их получения, фармацевтическая композиция, способ леченияInfo
- Publication number
- RU93045711A RU93045711A RU93045711/04A RU93045711A RU93045711A RU 93045711 A RU93045711 A RU 93045711A RU 93045711/04 A RU93045711/04 A RU 93045711/04A RU 93045711 A RU93045711 A RU 93045711A RU 93045711 A RU93045711 A RU 93045711A
- Authority
- RU
- Russia
- Prior art keywords
- pirasins
- pyrido
- treatment
- production
- pharmaceutical composition
- Prior art date
Links
- 230000000701 neuroleptic Effects 0.000 title 1
- 239000003176 neuroleptic agent Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- -1 cyclic imides Chemical class 0.000 claims 3
- 229940093912 Gynecological Sulfonamides Drugs 0.000 claims 1
- 230000000561 anti-psychotic Effects 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 229940079867 intestinal antiinfectives Sulfonamides Drugs 0.000 claims 1
- 229940005938 ophthalmologic antiinfectives Sulfonamides Drugs 0.000 claims 1
- 229940026752 topical Sulfonamides Drugs 0.000 claims 1
Claims (1)
- Антипсихотические соединения, имеющие формулу I, приведенную в описании, образуют циклические имиды, 4-замещенные пиперидины или циклические сульфонамиды.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US661.791 | 1991-02-27 | ||
US07/661,791 US5157034A (en) | 1991-02-27 | 1991-02-27 | Neuroleptic perhydro-1H-pyrido[1,2-a]pyrazines |
US661791 | 1991-02-27 | ||
PCT/US1991/008378 WO1992015580A1 (en) | 1991-02-27 | 1991-11-18 | NEUROLEPTIC PERHYDRO-1H-PYRIDO[1,2-a]PYRAZINES |
Publications (2)
Publication Number | Publication Date |
---|---|
RU93045711A true RU93045711A (ru) | 1996-06-20 |
RU2090565C1 RU2090565C1 (ru) | 1997-09-20 |
Family
ID=24655130
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU9193045711A RU2090565C1 (ru) | 1991-02-27 | 1991-11-18 | Рацемические или оптически активные пергидро-1h-пиридо(1,2-а) пиразины или их фармацевтически приемлемые соли и способ их получения |
Country Status (24)
Country | Link |
---|---|
US (1) | US5157034A (ru) |
EP (1) | EP0573467B1 (ru) |
JP (1) | JP2546770B2 (ru) |
KR (1) | KR0163413B1 (ru) |
AT (1) | ATE123284T1 (ru) |
AU (1) | AU652422B2 (ru) |
CA (2) | CA2101518C (ru) |
DE (2) | DE69110135T2 (ru) |
DK (1) | DK0573467T3 (ru) |
ES (1) | ES2073914T3 (ru) |
FI (3) | FI105030B (ru) |
HU (1) | HU216637B (ru) |
IE (1) | IE67190B1 (ru) |
IL (2) | IL101021A (ru) |
MX (1) | MX9200803A (ru) |
MY (1) | MY108185A (ru) |
NO (1) | NO300847B1 (ru) |
NZ (1) | NZ241739A (ru) |
PT (1) | PT100160B (ru) |
RU (1) | RU2090565C1 (ru) |
TW (1) | TW207540B (ru) |
WO (1) | WO1992015580A1 (ru) |
YU (1) | YU48311B (ru) |
ZA (1) | ZA921405B (ru) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5326874A (en) * | 1991-02-27 | 1994-07-05 | Pfizer Inc. | Process for preparing trans-piperidine-2,5-dicarboxylates |
JP2753146B2 (ja) * | 1992-06-16 | 1998-05-18 | ファイザー・インコーポレーテッド | ビス−アザー二環式抗不安薬の製法および中間体 |
WO1996010570A1 (en) * | 1994-09-30 | 1996-04-11 | Pfizer Inc. | NEUROLEPTIC 2,7-DISUBSTITUTED PERHYDRO-1H-PYRIDO[1,2-a]PYRAZINES |
US6231833B1 (en) | 1999-08-05 | 2001-05-15 | Pfizer Inc | 2,7-substituted octahydro-1H-pyrido[1,2-A]pyrazine derivatives as ligands for serotonin receptors |
CZ285090B6 (cs) * | 1994-09-30 | 1999-05-12 | Pfizer Inc. | 2,7-Disubstituovaný oktahydro-1H-pyrido-[1,2-a]pyrazinové deriváty a farmaceutické prostředky na jejich bázi |
PA8469101A1 (es) * | 1998-04-09 | 2000-09-29 | Pfizer Prod Inc | Ligandos azabiciclicos de receptores 5ht1 |
UA62015C2 (en) * | 1998-12-28 | 2003-12-15 | Pfizer Prod Inc | Benzoizoxazol derivatives, a pharmaceutical composition (variants) based thereon (variants) and a method for treatment (variants) |
EP1608648B1 (en) * | 2003-03-12 | 2012-07-18 | Pfizer Products Inc. | Pyridyloxymethyl and benzisoxazole azabicyclic derivatives |
PL217630B1 (pl) | 2003-04-24 | 2014-08-29 | Incyte Corp | Pochodne azaspiroalkanów, kompozycja farmaceutyczna oraz zastosowanie związku |
US7910108B2 (en) * | 2006-06-05 | 2011-03-22 | Incyte Corporation | Sheddase inhibitors combined with CD30-binding immunotherapeutics for the treatment of CD30 positive diseases |
CA2891122C (en) | 2012-11-14 | 2021-07-20 | The Johns Hopkins University | Methods and compositions for treating schizophrenia |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4681938A (en) * | 1984-08-27 | 1987-07-21 | Ciba-Geigy Corporation | Novel polycyclic hydrazones of rifamycins, their manufacture, and their pharmaceutical compositions for treating tuberculosis |
US4831031A (en) * | 1988-01-22 | 1989-05-16 | Pfizer Inc. | Aryl piperazinyl-(C2 or C4) alkylene heterocyclic compounds having neuroleptic activity |
US4957916A (en) * | 1988-08-05 | 1990-09-18 | Janssen Pharmaceutica N.V. | Antipsychotic 3-piperazinylbenzazole derivatives |
WO1990008148A1 (en) * | 1989-01-23 | 1990-07-26 | Pfizer Inc. | Bis-aza-bicyclic anxiolytic agents |
-
1991
- 1991-02-27 US US07/661,791 patent/US5157034A/en not_active Expired - Lifetime
- 1991-11-18 AT AT92904861T patent/ATE123284T1/de not_active IP Right Cessation
- 1991-11-18 DE DE69110135T patent/DE69110135T2/de not_active Expired - Fee Related
- 1991-11-18 HU HU9302427A patent/HU216637B/hu unknown
- 1991-11-18 KR KR1019930702554A patent/KR0163413B1/ko not_active IP Right Cessation
- 1991-11-18 DK DK92904861.9T patent/DK0573467T3/da active
- 1991-11-18 EP EP92904861A patent/EP0573467B1/en not_active Expired - Lifetime
- 1991-11-18 CA CA002101518A patent/CA2101518C/en not_active Expired - Fee Related
- 1991-11-18 JP JP4505183A patent/JP2546770B2/ja not_active Expired - Fee Related
- 1991-11-18 RU RU9193045711A patent/RU2090565C1/ru not_active IP Right Cessation
- 1991-11-18 DE DE9190206U patent/DE9190206U1/de not_active Expired - Lifetime
- 1991-11-18 ES ES92904861T patent/ES2073914T3/es not_active Expired - Lifetime
- 1991-11-18 WO PCT/US1991/008378 patent/WO1992015580A1/en active IP Right Grant
- 1991-11-18 AU AU12599/92A patent/AU652422B2/en not_active Ceased
- 1991-11-18 CA CA002163274A patent/CA2163274C/en not_active Expired - Fee Related
-
1992
- 1992-01-21 TW TW081100420A patent/TW207540B/zh active
- 1992-02-20 IL IL10102192A patent/IL101021A/en not_active IP Right Cessation
- 1992-02-20 IL IL11232595A patent/IL112325A/xx not_active IP Right Cessation
- 1992-02-25 MX MX9200803A patent/MX9200803A/es not_active IP Right Cessation
- 1992-02-25 PT PT100160A patent/PT100160B/pt not_active IP Right Cessation
- 1992-02-26 IE IE920601A patent/IE67190B1/en not_active IP Right Cessation
- 1992-02-26 NZ NZ24173992A patent/NZ241739A/en not_active IP Right Cessation
- 1992-02-26 YU YU19892A patent/YU48311B/sh unknown
- 1992-02-26 MY MYPI92000318A patent/MY108185A/en unknown
- 1992-02-26 ZA ZA921405A patent/ZA921405B/xx unknown
-
1993
- 1993-08-26 FI FI933753A patent/FI105030B/fi not_active IP Right Cessation
- 1993-08-26 NO NO933049A patent/NO300847B1/no unknown
-
2000
- 2000-02-17 FI FI20000354A patent/FI112865B/fi not_active IP Right Cessation
-
2003
- 2003-03-11 FI FI20030361A patent/FI114214B/fi not_active IP Right Cessation
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