ES8502114A1 - Un procedimiento para preparar una beta-lactama. - Google Patents
Un procedimiento para preparar una beta-lactama.Info
- Publication number
- ES8502114A1 ES8502114A1 ES524698A ES524698A ES8502114A1 ES 8502114 A1 ES8502114 A1 ES 8502114A1 ES 524698 A ES524698 A ES 524698A ES 524698 A ES524698 A ES 524698A ES 8502114 A1 ES8502114 A1 ES 8502114A1
- Authority
- ES
- Spain
- Prior art keywords
- oxoazetidin
- analogs
- substitute
- acetic acids
- lactam
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- SNRSSOXPZDUYHU-UHFFFAOYSA-N 2-(2-oxoazetidin-1-yl)oxyacetic acid Chemical class OC(=O)CON1CCC1=O SNRSSOXPZDUYHU-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- -1 HYDROXYL GROUP Chemical group 0.000 abstract 2
- 150000003952 β-lactams Chemical class 0.000 abstract 2
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 230000001681 protective effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Cephalosporin Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US40494582A | 1982-08-04 | 1982-08-04 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8502114A1 true ES8502114A1 (es) | 1984-12-16 |
| ES524698A0 ES524698A0 (es) | 1984-12-16 |
Family
ID=23601669
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES524698A Granted ES524698A0 (es) | 1982-08-04 | 1983-08-03 | Un procedimiento para preparar una beta-lactama. |
Country Status (33)
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4939253A (en) * | 1982-08-04 | 1990-07-03 | E. R. Squibb & Sons, Inc. | 2-oxoazetidin-1-yloxy acetic acids and analogs |
| US4548747A (en) * | 1983-05-02 | 1985-10-22 | E. R. Squibb & Sons, Inc. | 3-Acylamino-1-sulfonylaminocarbonylmethoxy-2-azetidinones |
| EP0127177B1 (en) * | 1983-05-31 | 1988-12-21 | E.R. Squibb & Sons, Inc. | [[(3-Acylamino-2-oxo-1-azetidinyl)oxy]methyl]phosphinic acids |
| US4534896A (en) * | 1983-06-13 | 1985-08-13 | E. R. Squibb & Sons, Inc. | 3-Acylamino-2-oxoazetidine-1-(β-oxopropionic acid) |
| US4548751A (en) * | 1983-08-03 | 1985-10-22 | E. R. Squibb & Sons, Inc. | (2-Oxo-1-azetidinyloxy)-2-propenoic acid |
| AU581180B2 (en) * | 1983-08-26 | 1989-02-16 | E.R. Squibb & Sons, Inc. | 1-(1h-tetrazol-5-ylalkoxy)-2-azetidinones |
| CA1243679A (en) * | 1983-09-14 | 1988-10-25 | Henner Straub | 3-ACYLAMINO-2-OXO-1-AZETIDINYL-.beta.-OXYPROPIONATES |
| WO1985004876A1 (en) * | 1984-04-24 | 1985-11-07 | Takeda Chemical Industries, Ltd. | 2-azetidinone derivatives and process for their preparation |
| EP0135194A1 (en) * | 1983-09-16 | 1985-03-27 | Takeda Chemical Industries, Ltd. | Azetidinones and their production |
| US4576749A (en) * | 1983-10-03 | 1986-03-18 | E. R. Squibb & Sons, Inc. | 3-Acylamino-1-carboxymethylaminocarbonyl-2-azetidinones |
| US4559335A (en) * | 1983-10-03 | 1985-12-17 | E. R. Squibb & Sons, Inc. | 3-Acylamino-1-carboxymethyloxy (or thio) carbonyl-2-azetidinones |
| US4551277A (en) * | 1983-11-09 | 1985-11-05 | E. R. Squibb & Sons, Inc. | 4-(3-Acylamino-2-oxo-1-azetidinyl)-4-oxo-2-butenoic acid |
| US4581170A (en) * | 1984-08-03 | 1986-04-08 | E. R. Squibb & Sons, Inc. | N-hydroxyl protecting groups and process and intermediates for the preparation of 3-acylamino-1-hydroxy-2-azetidinones |
| EG18314A (en) * | 1985-09-26 | 1993-02-28 | Squibb & Sons Inc | Process for preparing of 2-oxo-1((substituted sulfonyl)amino)carbonyl)-azitidines |
| US5112968A (en) * | 1989-07-28 | 1992-05-12 | E. R. Squibb & Sons, Inc. | Monobactam hydrazide derivatives |
| EP1827449A4 (en) * | 2004-11-17 | 2008-01-23 | Smithkline Beecham Corp | USE OF NOVEL ANTIBACTERIAL COMPOUNDS |
| DK2308874T3 (da) | 2005-12-07 | 2013-04-15 | Basilea Pharmaceutica Ag | Brokoblede monobactamer nyttige som beta-lactamase-inhibitorer |
| WO2014164526A1 (en) * | 2013-03-13 | 2014-10-09 | Rempex Pharmaceuticals, Inc. | Oxamazin antibiotics |
| US20140275007A1 (en) * | 2013-03-14 | 2014-09-18 | Rempex Pharmaceuticals, Inc. | Oxamazin antibiotics |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ196202A (en) * | 1980-02-07 | 1984-07-31 | Squibb & Sons Inc | Beta-lactam antibiotics (of azetidine-sulphonic acid type) |
| EP0048953B1 (en) * | 1980-09-29 | 1988-03-09 | E.R. Squibb & Sons, Inc. | Beta-lactam antibiotics |
| US4337197A (en) * | 1980-10-31 | 1982-06-29 | E. R. Squibb & Sons, Inc. | O-sulfated β-lactam hydroxamic acids and intermediates |
| WO1982001873A1 (en) * | 1980-12-05 | 1982-06-10 | Takeda Chemical Industries Ltd | 1-sulfo-2-oxoazetidine derivatives and process for their preparation |
| US4939253A (en) * | 1982-08-04 | 1990-07-03 | E. R. Squibb & Sons, Inc. | 2-oxoazetidin-1-yloxy acetic acids and analogs |
-
1983
- 1983-07-21 US US06/515,727 patent/US4939253A/en not_active Expired - Fee Related
- 1983-07-22 FI FI832675A patent/FI832675A7/fi not_active Application Discontinuation
- 1983-07-22 HU HU832602A patent/HU191058B/hu not_active IP Right Cessation
- 1983-07-26 ZA ZA835470A patent/ZA835470B/xx unknown
- 1983-07-28 GR GR72076A patent/GR79368B/el unknown
- 1983-07-29 GB GB08320497A patent/GB2125794B/en not_active Expired
- 1983-08-01 IL IL69381A patent/IL69381A/xx unknown
- 1983-08-02 NZ NZ205111A patent/NZ205111A/en unknown
- 1983-08-03 KR KR1019830003626A patent/KR900001211B1/ko not_active Expired
- 1983-08-03 DK DK354683A patent/DK354683A/da not_active Application Discontinuation
- 1983-08-03 NL NL8302746A patent/NL8302746A/nl unknown
- 1983-08-03 CS CS835759A patent/CS243474B2/cs unknown
- 1983-08-03 PT PT77155A patent/PT77155B/pt not_active IP Right Cessation
- 1983-08-03 CS CS83267A patent/CS26783A2/cs unknown
- 1983-08-03 SU SU833635150A patent/SU1329617A3/ru active
- 1983-08-03 CS CS85267A patent/CS243498B2/cs unknown
- 1983-08-03 AT AT0281283A patent/AT382367B/de not_active IP Right Cessation
- 1983-08-03 DE DE19833328047 patent/DE3328047A1/de not_active Ceased
- 1983-08-03 IE IE1830/83A patent/IE55839B1/en not_active IP Right Cessation
- 1983-08-03 ES ES524698A patent/ES524698A0/es active Granted
- 1983-08-03 SE SE8304256A patent/SE8304256L/xx not_active Application Discontinuation
- 1983-08-03 CS CS85268A patent/CS243499B2/cs unknown
- 1983-08-03 NO NO832801A patent/NO832801L/no unknown
- 1983-08-03 AU AU17556/83A patent/AU568086B2/en not_active Ceased
- 1983-08-04 IT IT22430/83A patent/IT1224129B/it active
- 1983-08-04 JP JP58143603A patent/JPS5993046A/ja active Pending
- 1983-08-04 FR FR8312862A patent/FR2531427A1/fr active Granted
- 1983-08-04 DD DD83253715A patent/DD213919A5/de not_active IP Right Cessation
- 1983-08-04 CH CH4244/83A patent/CH655309A5/fr not_active IP Right Cessation
- 1983-08-04 PL PL24330883A patent/PL243308A1/xx unknown
- 1983-08-04 AR AR293815A patent/AR241158A1/es active
- 1983-08-04 PL PL25744183A patent/PL257441A1/xx unknown
- 1983-08-04 PL PL25744083A patent/PL257440A1/xx unknown
- 1983-08-04 LU LU84947A patent/LU84947A1/fr unknown
- 1983-08-04 YU YU1627/83A patent/YU43324B/xx unknown
- 1983-08-04 RO RO111814A patent/RO86511B/ro unknown
- 1983-08-04 BE BE0/211304A patent/BE897466A/fr not_active IP Right Cessation
- 1983-08-11 IN IN525/DEL/83A patent/IN160955B/en unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ES8502114A1 (es) | Un procedimiento para preparar una beta-lactama. | |
| ES8602022A1 (es) | Un procedimiento para preparar un derivado de 4'-dimetil-4-epipodofilotoxina | |
| ES8102131A1 (es) | Procedimiento para preparar una composicion oral que com- prende un compuesto de 2-penem | |
| FI931031A0 (fi) | Mometasonfuroatmonohydrat, foerfarande foer dess framstaellning och farmaceutiska sammansaettningar | |
| ES8800186A1 (es) | Un metodo para preparar derivados de tiazol | |
| SE7803805L (sv) | Forfarande for framstellning av sellskapsdjursfoda av torr typ och dess sammansettning | |
| ES2060883T3 (es) | Procedimiento de obtencion del acido carnosico. | |
| ES2067022T3 (es) | Complejos estabilizados de oxido nitrico y aminas primarias utiles como agentes cardiovasculares. | |
| FI880163A0 (fi) | Menetelmä lääkeaineena käytettävän liuoksen valmistamiseksi | |
| ES2089199T3 (es) | Composicion curable. | |
| SE7601755L (sv) | Anvendning av perfluoralkansulfonamider och/eller ammoniumsalter av perfluoralkansulfonsyror och/eller cyklimmoniumsalter av perfluoralkansulfonsyror som formsleppmedel for termoplastiska, hogmolekyllera, m m | |
| LV12443A (en) | 7-(2-Aminoethyl)-benzothiazolones | |
| DE3580124D1 (de) | Pyridobenzothiazinderivate mit hoch antimikrobieller wirkung. | |
| ES2062375T3 (es) | Composiciones farmaceuticas que contienen un complejo de zinc. | |
| BE883616A (fr) | Compositions d'organopolysiloxane durcissables inhibees, exemptes de solvant | |
| ES2062215T3 (es) | Derivados aminoalcoxibencenicos sustituidos. | |
| DE68928174D1 (de) | Verfahren zur Herstellung von Cephemderivaten | |
| DE3686022D1 (de) | Monosaccharide enthaltende zusammensetzung zum heilen von wunden. | |
| MA19882A1 (fr) | Derives d'acides w-amines, leur preparation et utilisation ainsi que les compositions contenant ces acides. | |
| BE738104A (fr) | Procédé de préparation d'esters d'éthyléne glycol. | |
| ES388884A1 (es) | Procedimiento para la preparacion de 1-(2-nitrilofenoxi)-2-hidroxi-3-etilaminopropano racemicos u opticamente activo. | |
| UY24009A1 (es) | Compuestos ariltio útiles como agentes antivirales y antibacteriales | |
| BE779277A (fr) | Agents de protection contre l'hydrolyse pour matieres plastiques contenant des groupes ester | |
| ES8707550A1 (es) | Un procedimiento para preparar compuestos peptidicos sustituidos. | |
| ES2054833T3 (es) | Derivados tioformamida. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19970303 |