ES8401478A1 - "procedimiento de preparacion de 2-isopropilamino-pirimidina-n-oxido". - Google Patents

"procedimiento de preparacion de 2-isopropilamino-pirimidina-n-oxido".

Info

Publication number
ES8401478A1
ES8401478A1 ES516534A ES516534A ES8401478A1 ES 8401478 A1 ES8401478 A1 ES 8401478A1 ES 516534 A ES516534 A ES 516534A ES 516534 A ES516534 A ES 516534A ES 8401478 A1 ES8401478 A1 ES 8401478A1
Authority
ES
Spain
Prior art keywords
preparation
same
compositions containing
isopropylamino
therapeutic compositions
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES516534A
Other languages
English (en)
Other versions
ES516534A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Ipsen Pharma SAS
Original Assignee
Societe de Conseils de Recherches et dApplications Scientifiques SCRAS SAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Societe de Conseils de Recherches et dApplications Scientifiques SCRAS SAS filed Critical Societe de Conseils de Recherches et dApplications Scientifiques SCRAS SAS
Publication of ES8401478A1 publication Critical patent/ES8401478A1/es
Publication of ES516534A0 publication Critical patent/ES516534A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/42One nitrogen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE 2-ISOPROPILAMINOPIRIMI DINA-N-OXIDO.CONSISTE EN LA REACCION DE OXIDACION SUAVE DE 2-ISOPROPILAMINOPORIMIDINA CON UNA CANTIDAD ESTEQUIOMETRICA O UN EXCESO DE HASTA 10 DE UN AGENTE OXIDANTE, TAL COMO PEROXIDO DE HIDROGENO, ACIDO M-CLOROPEROXIBENZOICO, ACIDO CROMICO, ETC. LA REACCION SE LLEVA A CABO EN UN DISOLVENTE INERTE A UNA TEMPERATURA ENTRE 15JC Y 45JC.ESTE COMPUESTOS TIENE APLICACIONES FARMACOLOGICAS PARA LA REGENERACION NERVIOSA Y PARA EL TRATAMIENTO DE DISTROFIA MUSCULAR.
ES516534A 1981-10-16 1982-10-15 "procedimiento de preparacion de 2-isopropilamino-pirimidina-n-oxido". Granted ES516534A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8131201 1981-10-16

Publications (2)

Publication Number Publication Date
ES8401478A1 true ES8401478A1 (es) 1983-12-01
ES516534A0 ES516534A0 (es) 1983-12-01

Family

ID=10525194

Family Applications (1)

Application Number Title Priority Date Filing Date
ES516534A Granted ES516534A0 (es) 1981-10-16 1982-10-15 "procedimiento de preparacion de 2-isopropilamino-pirimidina-n-oxido".

Country Status (36)

Country Link
US (1) US4492701A (es)
JP (1) JPS58131971A (es)
KR (1) KR860001468B1 (es)
AR (1) AR230439A1 (es)
AT (1) AT383119B (es)
AU (1) AU554162B2 (es)
BE (1) BE894517A (es)
CA (1) CA1198434A (es)
CH (1) CH654834A5 (es)
DE (1) DE3238305A1 (es)
DK (1) DK156393C (es)
EG (1) EG16015A (es)
ES (1) ES516534A0 (es)
FI (1) FI76788C (es)
FR (2) FR2514645A1 (es)
GR (1) GR77344B (es)
HK (1) HK22585A (es)
HU (1) HU189185B (es)
IE (1) IE54028B1 (es)
IL (1) IL66894A (es)
IN (1) IN158958B (es)
IT (1) IT1152718B (es)
LU (1) LU84403A1 (es)
MA (1) MA19623A1 (es)
MX (1) MX7057E (es)
MY (1) MY8600124A (es)
NL (1) NL8203991A (es)
NO (1) NO157737C (es)
NZ (1) NZ202102A (es)
OA (1) OA07230A (es)
PL (1) PL135808B1 (es)
PT (1) PT75663B (es)
SE (1) SE461276B (es)
SG (1) SG91584G (es)
YU (1) YU225382A (es)
ZA (1) ZA827137B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0282637U (es) * 1988-12-15 1990-06-26
DE19930960A1 (de) * 1999-07-05 2001-01-18 Bayer Ag Verfahren zur Oxidation von organischen Verbindungen

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1249282B (es) * 1960-11-01
BE788648A (fr) * 1971-10-09 1973-01-02 Soc D Etudes Prod Chimique Derives de l'isopropylamino pyrimidine, leur preparation leur composition et leur utilisation therapeutique
US3984414A (en) * 1971-10-09 1976-10-05 Societe D'etudes De Produits Chimiques Dichloroacetate salt of 2-isopropylamino pyrimidine
GB1525995A (en) * 1976-02-18 1978-09-27 Soc D Etudes Prod Chimique Aminopyrimidine salt
IN153791B (es) * 1979-03-10 1984-08-18 Soc D Etudes Prod Chimique
BE882836A (fr) * 1979-05-15 1980-08-18 Soc D Etudes Prod Chimique Nouveaux derives halogenes de l'isopropylamino pyrimidine, leur preparation et leur utilisaton therapeutique

Also Published As

Publication number Publication date
ZA827137B (en) 1983-08-31
AU8939982A (en) 1983-04-21
MY8600124A (en) 1986-12-31
DK156393C (da) 1990-01-08
OA07230A (fr) 1984-04-30
PT75663A (en) 1982-11-01
DE3238305C2 (es) 1989-02-09
DK156393B (da) 1989-08-14
CH654834A5 (fr) 1986-03-14
DE3238305A1 (de) 1983-04-28
FI76788B (fi) 1988-08-31
FI823445A0 (fi) 1982-10-11
SE461276B (sv) 1990-01-29
FI76788C (fi) 1988-12-12
IE54028B1 (en) 1989-05-24
IE822504L (en) 1983-04-16
US4492701A (en) 1985-01-08
NO157737C (no) 1988-05-11
NO823440L (no) 1983-04-18
ATA382482A (de) 1986-10-15
IN158958B (es) 1987-02-28
IL66894A (en) 1985-12-31
SG91584G (en) 1985-06-14
EG16015A (en) 1986-12-30
YU225382A (en) 1985-03-20
NO157737B (no) 1988-02-01
MA19623A1 (fr) 1983-07-01
FR2514645A1 (fr) 1983-04-22
KR840001957A (ko) 1984-06-07
DK458082A (da) 1983-04-17
IL66894A0 (en) 1982-12-31
IT1152718B (it) 1987-01-07
BE894517A (fr) 1983-01-17
PL135808B1 (en) 1985-12-31
LU84403A1 (fr) 1983-06-13
NL8203991A (nl) 1983-05-16
CA1198434A (en) 1985-12-24
FR2514645B1 (es) 1984-05-18
FR2514764B1 (es) 1984-05-18
AT383119B (de) 1987-05-25
AU554162B2 (en) 1986-08-07
ES516534A0 (es) 1983-12-01
KR860001468B1 (ko) 1986-09-26
PL238643A1 (en) 1983-06-20
PT75663B (en) 1985-01-11
HU189185B (en) 1986-06-30
FR2514764A1 (fr) 1983-04-22
AR230439A1 (es) 1984-04-30
HK22585A (en) 1985-03-29
GR77344B (es) 1984-09-11
MX7057E (es) 1987-04-08
JPS6148831B2 (es) 1986-10-25
SE8205837D0 (sv) 1982-10-14
JPS58131971A (ja) 1983-08-06
FI823445L (fi) 1983-04-17
NZ202102A (en) 1984-11-09
IT8223733A0 (it) 1982-10-13
SE8205837L (sv) 1983-04-17

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