ES482330A1 - Un procedimiento para producir derivados de acido (dl)-16- fenoxi, y 16-fenoxi-sustituido-9-ceto-prostatrienoico. - Google Patents

Un procedimiento para producir derivados de acido (dl)-16- fenoxi, y 16-fenoxi-sustituido-9-ceto-prostatrienoico.

Info

Publication number
ES482330A1
ES482330A1 ES482330A ES482330A ES482330A1 ES 482330 A1 ES482330 A1 ES 482330A1 ES 482330 A ES482330 A ES 482330A ES 482330 A ES482330 A ES 482330A ES 482330 A1 ES482330 A1 ES 482330A1
Authority
ES
Spain
Prior art keywords
phenoxy
formula
hydrogen
keto
carboxylic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES482330A
Other languages
English (en)
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Syntex USA LLC
Original Assignee
Syntex USA LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex USA LLC filed Critical Syntex USA LLC
Publication of ES482330A1 publication Critical patent/ES482330A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/06Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08Systems containing only non-condensed rings with a five-membered ring the ring being saturated
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/582Recycling of unreacted starting or intermediate materials

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ES482330A 1978-07-10 1979-07-09 Un procedimiento para producir derivados de acido (dl)-16- fenoxi, y 16-fenoxi-sustituido-9-ceto-prostatrienoico. Expired ES482330A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/922,957 US4178457A (en) 1978-07-10 1978-07-10 (dl)-16-Phenoxy- and 16-substituted phenoxy-9-keto prostatrienoic acid derivatives and processes for the production thereof

Publications (1)

Publication Number Publication Date
ES482330A1 true ES482330A1 (es) 1980-08-16

Family

ID=25447871

Family Applications (1)

Application Number Title Priority Date Filing Date
ES482330A Expired ES482330A1 (es) 1978-07-10 1979-07-09 Un procedimiento para producir derivados de acido (dl)-16- fenoxi, y 16-fenoxi-sustituido-9-ceto-prostatrienoico.

Country Status (26)

Country Link
US (1) US4178457A (en, 2012)
EP (1) EP0008003B1 (en, 2012)
JP (1) JPS5513282A (en, 2012)
KR (1) KR890002773B1 (en, 2012)
AT (1) ATE2427T1 (en, 2012)
AU (1) AU527516B2 (en, 2012)
CA (1) CA1149802A (en, 2012)
CS (1) CS209927B2 (en, 2012)
DD (1) DD146179A5 (en, 2012)
DE (2) DE2964709D1 (en, 2012)
DK (1) DK157753C (en, 2012)
ES (1) ES482330A1 (en, 2012)
FI (1) FI69061C (en, 2012)
FR (1) FR2430939A1 (en, 2012)
GB (1) GB2025413B (en, 2012)
HK (1) HK41384A (en, 2012)
HU (1) HU184185B (en, 2012)
IT (1) IT1121462B (en, 2012)
MY (1) MY8500576A (en, 2012)
NO (4) NO150836C (en, 2012)
NZ (1) NZ190924A (en, 2012)
PL (4) PL120632B1 (en, 2012)
SG (1) SG82483G (en, 2012)
SU (1) SU1031407A3 (en, 2012)
YU (3) YU41870B (en, 2012)
ZA (1) ZA793293B (en, 2012)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4328245A (en) * 1981-02-13 1982-05-04 Syntex (U.S.A.) Inc. Carbonate diester solutions of PGE-type compounds
US4358603A (en) * 1981-04-16 1982-11-09 Syntex (U.S.A.) Inc. Acetal stabilized prostaglandin compositions
US4409239A (en) * 1982-01-21 1983-10-11 Syntex (U.S.A.) Inc. Propylene glycol diester solutions of PGE-type compounds
US4600785A (en) * 1983-12-22 1986-07-15 Syntex (U.S.A.) Inc. Processes and intermediates for making 16-phenoxy and 16-substituted phenoxy-prostatrienoic acid derivatives
US4804787A (en) * 1983-12-22 1989-02-14 Syntex (U.S.A.) Inc. Processes and intermediates for making 16-phenoxy and 16-substituted phenoxy-prostatrienoic acid derivatives
US4912235A (en) * 1983-12-22 1990-03-27 Syntex (U.S.A.) Inc. Processes and intermediates for making 16-phenoxy- and 16-substituted phenoxy-prostatrienoic acid derivatives and their stereoisomers
DE3414509A1 (de) * 1984-04-13 1985-10-24 Schering AG, 1000 Berlin und 4709 Bergkamen Neue 9-halogen-prostaglandine
US4618696A (en) * 1984-07-31 1986-10-21 Syntex (U.S.A.) Inc. 9-oxo-15α-hydroxy-16-phenoxy and 16-substituted phenoxy 17,18,19,20-tetranorprosta-4,5,13,(E)-trienoates
US5057621A (en) * 1984-07-31 1991-10-15 Syntex (U.S.A.) Inc. 11-substituted-16-phenoxy and 16-substituted phenoxy-prostatrienoic acid derivatives
US4792617A (en) * 1984-07-31 1988-12-20 Syntex (U.S.A.) Inc. 11-substituted-16-phenoxy and 16-substituted phenoxy-prostatrienioc acid derivatives
ES8607921A1 (es) * 1984-07-31 1986-06-16 Syntex Inc Procedimiento para preparar derivados de acidos 11-sustitui-dos-16-fenoxi y 16-fenoxi sustituido-prostatrienoicos
US4778904A (en) * 1985-09-13 1988-10-18 Syntex (U.S.A.) Inc. Intermediates for making 16-phenoxy- and 16-(substituted phenoxy)-prostatrienoic acid derivatives
EP0248999A3 (en) * 1986-04-11 1988-03-16 Syntex (U.S.A.) Inc. Uses of enprostil-type prostaglandins in regulating fat and carbohydrate metabolism
US4755531A (en) * 1986-08-11 1988-07-05 Syntex (U.S.A.) Inc. Thiol esters of 4,5-allenyl prostaglandins and use thereof as antigastric secretion agents
GB8625321D0 (en) * 1986-10-22 1986-11-26 Glaxo Group Ltd Chemical compounds
US4689419A (en) * 1986-11-14 1987-08-25 G. D. Searle & Co. Novel intermediate compounds in a process for producing 16-phenoxy- and 16-substituted phenoxy-9-keto-prostatrienoic acid derivatives
US6103765A (en) * 1997-07-09 2000-08-15 Androsolutions, Inc. Methods for treating male erectile dysfunction
AU742787B2 (en) 1997-07-09 2002-01-10 Androsolutions, Inc. Improved methods and compositions for treating male erectile dysfunction
US20020172693A1 (en) 2000-03-31 2002-11-21 Delong Michell Anthony Compositions and methods for treating hair loss using non-naturally occurring prostaglandins
US20020037914A1 (en) 2000-03-31 2002-03-28 Delong Mitchell Anthony Compositions and methods for treating hair loss using C16-C20 aromatic tetrahydro prostaglandins
US20020013294A1 (en) 2000-03-31 2002-01-31 Delong Mitchell Anthony Cosmetic and pharmaceutical compositions and methods using 2-decarboxy-2-phosphinico derivatives
US8966971B2 (en) * 2008-07-28 2015-03-03 Ford Global Technologies, Llc Vehicle engine with fluid measuring system
US8623918B2 (en) 2008-10-29 2014-01-07 Novaer Holdings, Inc. Amino acid salts of prostaglandins
EP2349242B1 (en) * 2008-10-29 2018-12-05 Novaer Holdings, Inc. Amino acid salts of prostaglandins
US8722739B2 (en) 2008-10-29 2014-05-13 Novaer Holdings, Inc. Amino acid salts of prostaglandins
US20110293549A1 (en) 2009-02-03 2011-12-01 Athena Cosmetics, Inc. Composition, method and kit for enhancing hair

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES449162A1 (es) * 1975-06-23 1977-12-16 Syntex Inc Un procedimiento para la preparacion de un compuesto racemi-co u 8r-antimerico.

Also Published As

Publication number Publication date
NO152212B (no) 1985-05-13
YU168579A (en) 1983-02-28
IT7968428A0 (it) 1979-07-09
MY8500576A (en) 1985-12-31
DE2927715C2 (en, 2012) 1987-08-27
NO792283L (no) 1980-01-11
JPS5513282A (en) 1980-01-30
PL121778B1 (en) 1982-05-31
AU4864179A (en) 1980-02-07
GB2025413B (en) 1982-07-28
FI792149A7 (fi) 1980-01-11
YU44553B (en) 1990-08-31
HU184185B (en) 1984-07-30
EP0008003B1 (en) 1983-02-09
YU44554B (en) 1990-08-31
SG82483G (en) 1984-08-03
YU73686A (en) 1986-12-31
NO840258L (no) 1980-01-11
PL120633B1 (en) 1982-03-31
GB2025413A (en) 1980-01-23
DE2964709D1 (en) 1983-03-17
FR2430939A1 (fr) 1980-02-08
YU73586A (en) 1986-12-31
CA1149802A (en) 1983-07-12
AU527516B2 (en) 1983-03-10
NO152211B (no) 1985-05-13
DE2927715A1 (de) 1980-01-24
EP0008003A1 (en) 1980-02-20
ATE2427T1 (de) 1983-03-15
FI69061B (fi) 1985-08-30
DK157753C (da) 1990-07-09
NO152211C (no) 1985-08-21
NO152296C (no) 1985-09-04
NO840256L (no) 1980-01-11
NO150836C (no) 1985-01-09
FR2430939B1 (en, 2012) 1981-08-14
NO150836B (no) 1984-09-17
NO152296B (no) 1985-05-28
NO840257L (no) 1980-01-11
NZ190924A (en) 1980-11-28
US4178457A (en) 1979-12-11
FI69061C (fi) 1985-12-10
CS209927B2 (en) 1981-12-31
PL217001A1 (en, 2012) 1980-03-24
PL120632B1 (en) 1982-03-31
NO152212C (no) 1985-08-21
HK41384A (en) 1984-05-18
DK288879A (da) 1980-01-11
KR890002773B1 (ko) 1989-07-28
DK157753B (da) 1990-02-12
IT1121462B (it) 1986-04-02
ZA793293B (en) 1981-02-25
SU1031407A3 (ru) 1983-07-23
PL120604B1 (en) 1982-03-31
JPS6210227B2 (en, 2012) 1987-03-05
YU41870B (en) 1988-02-29
DD146179A5 (de) 1981-01-28

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970203