ES2550319T3 - Moduladores selectivos del receptor de andrógenos - Google Patents

Moduladores selectivos del receptor de andrógenos Download PDF

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Publication number
ES2550319T3
ES2550319T3 ES11767355.8T ES11767355T ES2550319T3 ES 2550319 T3 ES2550319 T3 ES 2550319T3 ES 11767355 T ES11767355 T ES 11767355T ES 2550319 T3 ES2550319 T3 ES 2550319T3
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methyl
trifluoro
hydroxyethyl
benzonitrile
mmol
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Spanish (es)
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Chris P. Miller
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Radius Health Inc
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Radius Health Inc
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    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
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    • C07D263/16Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18Oxygen atoms
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    • GPHYSICS
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    • G01N33/48Biological material, e.g. blood, urine; Haemocytometers
    • G01N33/50Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
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    • G01N2333/705Assays involving receptors, cell surface antigens or cell surface determinants
    • G01N2333/70567Nuclear receptors, e.g. retinoic acid receptor [RAR], RXR, nuclear orphan receptors

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ES11767355.8T 2010-09-28 2011-09-27 Moduladores selectivos del receptor de andrógenos Active ES2550319T3 (es)

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Application Number Priority Date Filing Date Title
US387440P 2002-06-11
US38744010P 2010-09-28 2010-09-28
PCT/US2011/053375 WO2012047617A1 (en) 2010-09-28 2011-09-27 Selective androgen receptor modulators

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ES2550319T3 true ES2550319T3 (es) 2015-11-06

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US (2) US9133182B2 (enExample)
EP (1) EP2621901B1 (enExample)
JP (1) JP5965909B2 (enExample)
AU (1) AU2011312490B2 (enExample)
BR (1) BR112013007685B1 (enExample)
ES (1) ES2550319T3 (enExample)
WO (1) WO2012047617A1 (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2531029B1 (en) 2010-02-04 2016-10-19 Radius Health, Inc. Selective androgen receptor modulators
US20130053448A1 (en) 2010-05-12 2013-02-28 Louis O'Dea Therapeutic Regimens
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