ES2400687T3 - Formulaciones de liberación sostenida - Google Patents
Formulaciones de liberación sostenida Download PDFInfo
- Publication number
- ES2400687T3 ES2400687T3 ES05742315T ES05742315T ES2400687T3 ES 2400687 T3 ES2400687 T3 ES 2400687T3 ES 05742315 T ES05742315 T ES 05742315T ES 05742315 T ES05742315 T ES 05742315T ES 2400687 T3 ES2400687 T3 ES 2400687T3
- Authority
- ES
- Spain
- Prior art keywords
- peptide
- complex
- gallic acid
- acid ester
- pgg
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
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- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
Landscapes
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- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Peptides Or Proteins (AREA)
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| US7252834B2 (en) * | 2005-04-25 | 2007-08-07 | Clemson University Research Foundation (Curf) | Elastin stabilization of connective tissue |
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| AU2007275638B2 (en) * | 2006-07-21 | 2014-01-16 | Amgen Inc. | Method of detecting and/ or measuring hepcidin in a sample |
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| EP2162540A2 (en) | 2007-05-22 | 2010-03-17 | Amgen Inc. | Compositions and methods for producing bioactive fusion proteins |
| CA2709354C (en) | 2007-12-21 | 2014-06-17 | Amgen Inc. | Anti-amyloid antibodies and uses thereof |
| US20090214654A1 (en) * | 2008-02-21 | 2009-08-27 | Isenburg Jason C | Treatment of aneurysm with application of connective tissue stabilization agent in combination with a delivery vehicle |
| US20100016833A1 (en) * | 2008-07-15 | 2010-01-21 | Ogle Matthew F | Devices for the Treatment of Vascular Aneurysm |
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| US8444624B2 (en) * | 2009-10-19 | 2013-05-21 | Vatrix Medical, Inc. | Vascular medical devices with sealing elements and procedures for the treatment of isolated vessel sections |
| US8911468B2 (en) | 2011-01-31 | 2014-12-16 | Vatrix Medical, Inc. | Devices, therapeutic compositions and corresponding percutaneous treatment methods for aortic dissection |
| SG10201601789TA (en) | 2011-03-16 | 2016-04-28 | Amgen Inc | Potent And Selective Inhibitors Of Nav1.3 And Nav1.7 |
| EP2709711B8 (en) | 2011-05-18 | 2017-03-22 | Vatrix Medical, Inc. | Coated balloons for blood vessel stabilization |
| JP6145112B2 (ja) | 2011-12-19 | 2017-06-07 | アムジエン・インコーポレーテツド | 単独でのまたは化学療法と組み合わされた変異アクチビン受容体ポリペプチド、およびその使用 |
| US20160067347A1 (en) | 2012-12-20 | 2016-03-10 | Amgen Inc. | Apj receptor agonists and uses thereof |
| CA2899889A1 (en) | 2013-02-01 | 2014-08-07 | Santa Maria Biotherapeutics, Inc. | Administration of an anti-activin-a compound to a subject |
| US10344060B2 (en) | 2013-03-12 | 2019-07-09 | Amgen Inc. | Potent and selective inhibitors of Nav1.7 |
| AU2015274574B2 (en) | 2014-06-10 | 2019-10-10 | Amgen Inc. | Apelin polypeptides |
| TW201618783A (zh) | 2014-08-07 | 2016-06-01 | 艾森塔製藥公司 | 以布魯頓(Bruton)氏酪胺酸激酶(BTK)佔據和BTK再合成速率為基礎之治療癌症、免疫和自體免疫疾病及發炎性疾病之方法 |
| US11318190B2 (en) | 2017-05-05 | 2022-05-03 | United States Government As Represented By The Department Of Veterans Affairs | Methods and compositions for treating liver disease |
| EP3634507B1 (en) * | 2017-06-07 | 2025-01-15 | EGY-Nano Pharma, LP | Oral prolonged drug delivery platforms |
| KR20210080349A (ko) | 2018-08-03 | 2021-06-30 | 넥테로 메디칼, 인크. | 정제된 펜타갈로일 글루코스 및 전달용 장치 |
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| CN119326891B (zh) * | 2024-10-31 | 2025-07-01 | 中国人民解放军空军军医大学 | Ei24激动剂以及在制备抑制食管鳞癌增殖的制剂的应用 |
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| US5151265A (en) * | 1987-11-03 | 1992-09-29 | Genentech, Inc. | Gamma interferon formulation |
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| WO1994008599A1 (en) | 1992-10-14 | 1994-04-28 | The Regents Of The University Of Colorado | Ion-pairing of drugs for improved efficacy and delivery |
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| AU4414497A (en) | 1996-09-13 | 1998-04-02 | University Technology Corporation | Biocompatible cationic detergents and uses therefor |
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| BR9811478A (pt) * | 1997-07-23 | 2000-08-15 | Perio Prod Ltd | Composições de polìmero-ácido tânico para a liberação controlada de agentes farmacêuticos particularmente na cavidade oral |
| US5962522A (en) | 1997-09-05 | 1999-10-05 | Avmax, Inc. | Propyl gallate to increase bioavailability of orally administered pharmaceutical compounds |
| US6180666B1 (en) | 1997-09-05 | 2001-01-30 | Anmax, Inc. | Use of gallic acid esters to increase bioavailability of orally administered pharmaceutical compounds |
| US6613358B2 (en) | 1998-03-18 | 2003-09-02 | Theodore W. Randolph | Sustained-release composition including amorphous polymer |
| DE69921636T2 (de) * | 1998-04-20 | 2005-11-03 | Genzyme Corp., Cambridge | Medikamentöse verabreichung von proteinen aus polymergemischen |
| JP2000080027A (ja) * | 1998-09-02 | 2000-03-21 | Taiyo Kagaku Co Ltd | 徐放性製剤 |
| US6428818B1 (en) | 1999-03-30 | 2002-08-06 | Purdue Research Foundation | Tea catechin formulations and processes for making same |
| AU1360901A (en) | 1999-11-01 | 2001-05-14 | University Technology Corporation | Compositions and methods for controlled-release delivery and increased potency of pharmaceuticals via hydrophobic ion-pairing |
| US6713506B2 (en) * | 2000-10-11 | 2004-03-30 | University Of South Florida | Tea polyphenol esters and analogs thereof for cancer prevention and treatment |
| WO2002067966A1 (en) | 2001-02-22 | 2002-09-06 | Purdue Research Foundation | Compositions based on vanilloid-catechin synergies for prevention and treatment of cancer |
| JP5013152B2 (ja) | 2001-02-28 | 2012-08-29 | 株式会社ビーエムジー | 蛋白質複合体形成剤 |
| US20040142048A1 (en) * | 2002-02-22 | 2004-07-22 | Morre Dorothy M. | Compositions based on proanthocyanadin-catechin synergies for prevention and treatment of cancer |
| US20050271603A1 (en) * | 2002-07-26 | 2005-12-08 | Stephanie Krammer | Compositions comprising lactoferrin |
| US8912174B2 (en) * | 2003-04-16 | 2014-12-16 | Mylan Pharmaceuticals Inc. | Formulations and methods for treating rhinosinusitis |
| US7605120B2 (en) * | 2003-10-22 | 2009-10-20 | Amgen Inc. | Antagonists of the brandykinin B1 receptor |
| US7323169B2 (en) * | 2004-04-23 | 2008-01-29 | Amgen Inc. | Sustained release formulations |
-
2005
- 2005-04-25 US US11/114,473 patent/US7323169B2/en not_active Expired - Fee Related
- 2005-04-25 WO PCT/US2005/014254 patent/WO2005105057A1/en not_active Ceased
- 2005-04-25 ES ES05742315T patent/ES2400687T3/es not_active Expired - Lifetime
- 2005-04-25 CA CA2563185A patent/CA2563185C/en not_active Expired - Fee Related
- 2005-04-25 JP JP2007509735A patent/JP5036533B2/ja not_active Expired - Fee Related
- 2005-04-25 CN CNA2005800124592A patent/CN1997356A/zh active Pending
- 2005-04-25 PT PT57423154T patent/PT1750683E/pt unknown
- 2005-04-25 EP EP05742315A patent/EP1750683B1/en not_active Expired - Lifetime
- 2005-04-25 PL PL05742315T patent/PL1750683T3/pl unknown
- 2005-04-25 DK DK05742315.4T patent/DK1750683T3/da active
- 2005-04-25 KR KR1020067021346A patent/KR101201638B1/ko not_active Expired - Fee Related
- 2005-04-25 SI SI200531678T patent/SI1750683T1/sl unknown
- 2005-04-25 CN CN201410023256.4A patent/CN103920162B/zh not_active Expired - Fee Related
- 2005-04-25 AU AU2005237542A patent/AU2005237542B2/en not_active Ceased
-
2006
- 2006-10-15 IL IL178596A patent/IL178596A/en not_active IP Right Cessation
- 2006-11-13 ZA ZA200609401A patent/ZA200609401B/en unknown
-
2007
- 2007-08-30 US US11/847,984 patent/US7732399B2/en not_active Expired - Fee Related
-
2011
- 2011-09-09 JP JP2011196884A patent/JP2012036194A/ja active Pending
- 2011-09-09 JP JP2011196883A patent/JP5829870B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP5829870B2 (ja) | 2015-12-09 |
| CN103920162A (zh) | 2014-07-16 |
| AU2005237542B2 (en) | 2009-12-17 |
| JP2007534698A (ja) | 2007-11-29 |
| CA2563185C (en) | 2010-04-20 |
| PT1750683E (pt) | 2013-01-25 |
| JP2012036194A (ja) | 2012-02-23 |
| JP5036533B2 (ja) | 2012-09-26 |
| WO2005105057A1 (en) | 2005-11-10 |
| EP1750683B1 (en) | 2013-01-09 |
| SI1750683T1 (sl) | 2013-04-30 |
| CA2563185A1 (en) | 2005-11-10 |
| EP1750683A1 (en) | 2007-02-14 |
| JP2012046520A (ja) | 2012-03-08 |
| CN103920162B (zh) | 2017-07-11 |
| ZA200609401B (en) | 2008-05-28 |
| IL178596A0 (en) | 2007-02-11 |
| PL1750683T3 (pl) | 2013-05-31 |
| US20050271722A1 (en) | 2005-12-08 |
| US7323169B2 (en) | 2008-01-29 |
| AU2005237542A1 (en) | 2005-11-10 |
| CN1997356A (zh) | 2007-07-11 |
| HK1103023A1 (en) | 2007-12-14 |
| US7732399B2 (en) | 2010-06-08 |
| DK1750683T3 (da) | 2013-04-15 |
| HK1200092A1 (en) | 2015-07-31 |
| KR20070026457A (ko) | 2007-03-08 |
| KR101201638B1 (ko) | 2012-11-15 |
| IL178596A (en) | 2012-06-28 |
| US20070292506A1 (en) | 2007-12-20 |
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