ES2307751T3 - Nuevos esteres heterociclicos centi-inflamatorios 17 alfa de derivados 17 beta de carbotioato de androstano. - Google Patents

Nuevos esteres heterociclicos centi-inflamatorios 17 alfa de derivados 17 beta de carbotioato de androstano. Download PDF

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Publication number
ES2307751T3
ES2307751T3 ES02730498T ES02730498T ES2307751T3 ES 2307751 T3 ES2307751 T3 ES 2307751T3 ES 02730498 T ES02730498 T ES 02730498T ES 02730498 T ES02730498 T ES 02730498T ES 2307751 T3 ES2307751 T3 ES 2307751T3
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Spain
Prior art keywords
methyl
hydroxy
oxy
oxo
androsta
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Expired - Lifetime
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ES02730498T
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English (en)
Spanish (es)
Inventor
Keith GlaxoSmithKline BIGGADIKE
Paul GlaxoSmithKline JONES
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Glaxo Group Ltd
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Glaxo Group Ltd
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Priority claimed from GB0114338A external-priority patent/GB0114338D0/en
Priority claimed from GB0202636A external-priority patent/GB0202636D0/en
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Publication of ES2307751T3 publication Critical patent/ES2307751T3/es
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/44—Glucocorticosteroids; Drugs increasing or potentiating the activity of glucocorticosteroids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
ES02730498T 2001-06-12 2002-06-11 Nuevos esteres heterociclicos centi-inflamatorios 17 alfa de derivados 17 beta de carbotioato de androstano. Expired - Lifetime ES2307751T3 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0114338A GB0114338D0 (en) 2001-06-12 2001-06-12 Novel compounds
GB0114338 2001-06-12
GB0202636 2002-02-05
GB0202636A GB0202636D0 (en) 2002-02-05 2002-02-05 Novel compounds

Publications (1)

Publication Number Publication Date
ES2307751T3 true ES2307751T3 (es) 2008-12-01

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
ES02730498T Expired - Lifetime ES2307751T3 (es) 2001-06-12 2002-06-11 Nuevos esteres heterociclicos centi-inflamatorios 17 alfa de derivados 17 beta de carbotioato de androstano.

Country Status (8)

Country Link
US (1) US20040248867A1 (enExample)
EP (1) EP1395604B1 (enExample)
JP (1) JP2005500290A (enExample)
AR (1) AR034475A1 (enExample)
AT (1) ATE399174T1 (enExample)
DE (1) DE60227254D1 (enExample)
ES (1) ES2307751T3 (enExample)
WO (1) WO2002100879A1 (enExample)

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ATE399174T1 (de) 2008-07-15
EP1395604B1 (en) 2008-06-25
AR034475A1 (es) 2004-02-25
EP1395604A1 (en) 2004-03-10
DE60227254D1 (de) 2008-08-07
US20040248867A1 (en) 2004-12-09
JP2005500290A (ja) 2005-01-06

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