DE60227254D1 - Neue anti inflammatorische 17.alpha.-heterozyklische ester von 17.beta.-carbothioat androstan derivativen - Google Patents
Neue anti inflammatorische 17.alpha.-heterozyklische ester von 17.beta.-carbothioat androstan derivativenInfo
- Publication number
- DE60227254D1 DE60227254D1 DE60227254T DE60227254T DE60227254D1 DE 60227254 D1 DE60227254 D1 DE 60227254D1 DE 60227254 T DE60227254 T DE 60227254T DE 60227254 T DE60227254 T DE 60227254T DE 60227254 D1 DE60227254 D1 DE 60227254D1
- Authority
- DE
- Germany
- Prior art keywords
- carbothioat
- beta
- alpha
- new anti
- anti inflammatory
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
- A61P5/44—Glucocorticosteroids; Drugs increasing or potentiating the activity of glucocorticosteroids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0114338A GB0114338D0 (en) | 2001-06-12 | 2001-06-12 | Novel compounds |
GB0202636A GB0202636D0 (en) | 2002-02-05 | 2002-02-05 | Novel compounds |
PCT/GB2002/002686 WO2002100879A1 (en) | 2001-06-12 | 2002-06-11 | Novel anti-inflammatory 17.alpha.-heterocyclic-esters of 17.beta.carbothioate androstane derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
DE60227254D1 true DE60227254D1 (de) | 2008-08-07 |
Family
ID=26246181
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60227254T Expired - Fee Related DE60227254D1 (de) | 2001-06-12 | 2002-06-11 | Neue anti inflammatorische 17.alpha.-heterozyklische ester von 17.beta.-carbothioat androstan derivativen |
Country Status (8)
Country | Link |
---|---|
US (1) | US20040248867A1 (de) |
EP (1) | EP1395604B1 (de) |
JP (1) | JP2005500290A (de) |
AR (1) | AR034475A1 (de) |
AT (1) | ATE399174T1 (de) |
DE (1) | DE60227254D1 (de) |
ES (1) | ES2307751T3 (de) |
WO (1) | WO2002100879A1 (de) |
Families Citing this family (107)
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CN101939054B (zh) | 2007-12-10 | 2014-10-29 | 诺华股份有限公司 | 有机化合物 |
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-
2002
- 2002-06-11 AT AT02730498T patent/ATE399174T1/de not_active IP Right Cessation
- 2002-06-11 JP JP2003503645A patent/JP2005500290A/ja active Pending
- 2002-06-11 DE DE60227254T patent/DE60227254D1/de not_active Expired - Fee Related
- 2002-06-11 WO PCT/GB2002/002686 patent/WO2002100879A1/en active IP Right Grant
- 2002-06-11 US US10/480,071 patent/US20040248867A1/en not_active Abandoned
- 2002-06-11 ES ES02730498T patent/ES2307751T3/es not_active Expired - Lifetime
- 2002-06-11 EP EP02730498A patent/EP1395604B1/de not_active Expired - Lifetime
- 2002-06-12 AR ARP020102212A patent/AR034475A1/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
JP2005500290A (ja) | 2005-01-06 |
EP1395604B1 (de) | 2008-06-25 |
AR034475A1 (es) | 2004-02-25 |
EP1395604A1 (de) | 2004-03-10 |
ATE399174T1 (de) | 2008-07-15 |
US20040248867A1 (en) | 2004-12-09 |
WO2002100879A1 (en) | 2002-12-19 |
ES2307751T3 (es) | 2008-12-01 |
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