ES2208334T3 - Derivados cetolida de 6-0 carbamato. - Google Patents

Derivados cetolida de 6-0 carbamato.

Info

Publication number
ES2208334T3
ES2208334T3 ES00936424T ES00936424T ES2208334T3 ES 2208334 T3 ES2208334 T3 ES 2208334T3 ES 00936424 T ES00936424 T ES 00936424T ES 00936424 T ES00936424 T ES 00936424T ES 2208334 T3 ES2208334 T3 ES 2208334T3
Authority
ES
Spain
Prior art keywords
group
compound
aryl
formula
heteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES00936424T
Other languages
English (en)
Spanish (es)
Inventor
Ly T. Phan
Yat Sun Or
Zhenkun Ma
Yan Chen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Laboratories
Original Assignee
Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Application granted granted Critical
Publication of ES2208334T3 publication Critical patent/ES2208334T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biotechnology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
ES00936424T 1999-06-07 2000-05-31 Derivados cetolida de 6-0 carbamato. Expired - Lifetime ES2208334T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32778499A 1999-06-07 1999-06-07
US327784 1999-06-07

Publications (1)

Publication Number Publication Date
ES2208334T3 true ES2208334T3 (es) 2004-06-16

Family

ID=23278051

Family Applications (1)

Application Number Title Priority Date Filing Date
ES00936424T Expired - Lifetime ES2208334T3 (es) 1999-06-07 2000-05-31 Derivados cetolida de 6-0 carbamato.

Country Status (10)

Country Link
EP (1) EP1181300B1 (enExample)
JP (1) JP2003501439A (enExample)
AT (1) ATE250076T1 (enExample)
CA (1) CA2378671C (enExample)
DE (1) DE60005334T2 (enExample)
DK (1) DK1181300T3 (enExample)
ES (1) ES2208334T3 (enExample)
MX (1) MXPA01012661A (enExample)
PT (1) PT1181300E (enExample)
WO (1) WO2000075156A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
CA2370743A1 (en) 1999-04-16 2000-10-26 Dennis Hlasta Ketolide antibacterials
EP1146051A3 (en) * 2000-04-10 2001-10-31 Pfizer Products Inc. Erythromycin A derivatives
US6472372B1 (en) 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
CA2460947A1 (en) 2001-09-17 2003-03-27 Ortho-Mcneil Pharmaceutical, Inc. 6-o-carbamate-11,12-lacto-ketolide antimicrobials
RU2004117082A (ru) 2001-12-05 2005-04-10 Орто-Макнейл Фармасьютикал, Инк. (Us) Кетолидные 6-0-ацил-производные эритромицина в качестве антибактериальных средств
CA2487918A1 (en) * 2002-05-31 2003-12-11 Janssen Pharmaceutica N.V. 3-descladinosyl-6-o-carbamoyl and 6-o-carbonoyl macrolide antibacterial agents

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8521402D0 (en) * 1985-08-28 1985-10-02 Beecham Group Plc Chemical compounds
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of erythromycin derivatives
US5750510A (en) * 1997-04-04 1998-05-12 Abbott Laboratories 3-descladinose-2,3-anhydroerythromycin derivatives
ES2242983T3 (es) * 1996-09-04 2005-11-16 Abbott Laboratories Cetolidos 6-0-sustituidos que tienen una actividad antibacteriana.
AU4472797A (en) * 1996-10-31 1998-05-22 Taisho Pharmaceutical Co., Ltd. Erythromycin a derivatives
KR20010013041A (ko) * 1997-05-29 2001-02-26 스티븐 에프. 웨인스톡 다환식 에리트로마이신 유도체
CN1259135A (zh) * 1997-06-11 2000-07-05 辉瑞产品公司 9-肟红霉素衍生物

Also Published As

Publication number Publication date
ATE250076T1 (de) 2003-10-15
DK1181300T3 (da) 2004-01-26
PT1181300E (pt) 2004-02-27
EP1181300A1 (en) 2002-02-27
EP1181300B1 (en) 2003-09-17
DE60005334D1 (de) 2003-10-23
WO2000075156A1 (en) 2000-12-14
MXPA01012661A (es) 2002-07-22
JP2003501439A (ja) 2003-01-14
CA2378671A1 (en) 2000-12-14
CA2378671C (en) 2007-04-24
DE60005334T2 (de) 2004-06-24

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