PT1181300E - Derivados 6-o-carbamato de cetolido - Google Patents

Derivados 6-o-carbamato de cetolido

Info

Publication number
PT1181300E
PT1181300E PT00936424T PT00936424T PT1181300E PT 1181300 E PT1181300 E PT 1181300E PT 00936424 T PT00936424 T PT 00936424T PT 00936424 T PT00936424 T PT 00936424T PT 1181300 E PT1181300 E PT 1181300E
Authority
PT
Portugal
Prior art keywords
carbamate
cetolid
derivatives
compound
prodrug
Prior art date
Application number
PT00936424T
Other languages
English (en)
Portuguese (pt)
Inventor
Ly T Phan
Yat Sun Or
Zhenkun Ma
Yan Chen
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of PT1181300E publication Critical patent/PT1181300E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
PT00936424T 1999-06-07 2000-05-31 Derivados 6-o-carbamato de cetolido PT1181300E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US32778499A 1999-06-07 1999-06-07

Publications (1)

Publication Number Publication Date
PT1181300E true PT1181300E (pt) 2004-02-27

Family

ID=23278051

Family Applications (1)

Application Number Title Priority Date Filing Date
PT00936424T PT1181300E (pt) 1999-06-07 2000-05-31 Derivados 6-o-carbamato de cetolido

Country Status (10)

Country Link
EP (1) EP1181300B1 (enExample)
JP (1) JP2003501439A (enExample)
AT (1) ATE250076T1 (enExample)
CA (1) CA2378671C (enExample)
DE (1) DE60005334T2 (enExample)
DK (1) DK1181300T3 (enExample)
ES (1) ES2208334T3 (enExample)
MX (1) MXPA01012661A (enExample)
PT (1) PT1181300E (enExample)
WO (1) WO2000075156A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
IL145976A0 (en) 1999-04-16 2002-07-25 Ortho Mcneil Pharm Inc Ketolide antibacterials
EP1146051A3 (en) * 2000-04-10 2001-10-31 Pfizer Products Inc. Erythromycin A derivatives
US6472372B1 (en) 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
CN1589277A (zh) * 2001-09-17 2005-03-02 奥索-麦克尼尔药品公司 6-o-氨基甲酸酯-11,12-内酯-酮内酯抗菌剂
AU2002346475A1 (en) 2001-12-05 2003-06-23 Ortho-Mcneil Pharmaceutical, Inc. 6-o-acyl ketolide derivatives of erythromycine useful as antibacterials
WO2003102010A1 (en) 2002-05-31 2003-12-11 Janssen Pharmaceutica N.V. 3-descladinosyl-6-o-carbamoyl and 6-o-carbonoyl macrolide antibacterial agents

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8521402D0 (en) * 1985-08-28 1985-10-02 Beecham Group Plc Chemical compounds
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
US5750510A (en) * 1997-04-04 1998-05-12 Abbott Laboratories 3-descladinose-2,3-anhydroerythromycin derivatives
SK285534B6 (sk) * 1996-09-04 2007-03-01 Abbott Laboratories 6-O-substituované ketolidy s antibakteriálnou aktivitou, farmaceutická kompozícia s ich obsahom, ich použitie a spôsob ich prípravy
AU4472797A (en) * 1996-10-31 1998-05-22 Taisho Pharmaceutical Co., Ltd. Erythromycin a derivatives
CA2290421C (en) * 1997-05-29 2007-05-08 Abbott Laboratories Multicyclic erythromycin derivatives
CN1259135A (zh) * 1997-06-11 2000-07-05 辉瑞产品公司 9-肟红霉素衍生物

Also Published As

Publication number Publication date
ATE250076T1 (de) 2003-10-15
JP2003501439A (ja) 2003-01-14
DK1181300T3 (da) 2004-01-26
WO2000075156A1 (en) 2000-12-14
EP1181300A1 (en) 2002-02-27
ES2208334T3 (es) 2004-06-16
MXPA01012661A (es) 2002-07-22
DE60005334T2 (de) 2004-06-24
CA2378671A1 (en) 2000-12-14
DE60005334D1 (de) 2003-10-23
CA2378671C (en) 2007-04-24
EP1181300B1 (en) 2003-09-17

Similar Documents

Publication Publication Date Title
MY133996A (en) Compounds for the treatment of ischemia
AP9801378A0 (en) 9-amino-3- keto erythromycin derivatives.
IL165715A0 (en) 2-ureido-6-heteroaryl-3h-benzoimidazole-4-carboxylic acid derivatives, pharmaceutical compositions containing the same and methods for the preparation thereof
BG103945A (bg) Производни на 4"-заместен-9-деоксо-9а-аза-9а- хомоеритромицин а
AP9801253A0 (en) 9-Oxime erythromycin derivatives.
PT915898E (pt) Forma i cristalina de claritromicina
TR200200579T2 (tr) Amino-tirazolpiridin türevleri.
WO2001092288A3 (en) Cobalamin compounds useful as antibiotic agents and as imaging agents
TR200103395T2 (tr) 13-metil eritromisin türevleri.
NZ515339A (en) Use of macrolide compounds for the treatment of dry eye
AR034343A1 (es) Combinaciones farmaceuticas
EP0992509A3 (en) Novel macrolide derivatives
DK1181300T3 (da) 6-O-carbamatketolidderivater
AP9801377A0 (en) Tricyclic erythromycin derivatives.
EE05241B1 (et) Distamtsiini a-halogenoakrlolderivaadi kasutamine
BG102661A (en) Benzo/o/quinolysine derivatives, their preparation and application as 5a-reductase inhibitors
AU2001252711A1 (en) Aqueous-prodrug compound comprising moiety of paclitxel or derivatives thereof, method of preparing same and pharmaceutical composition comprising same
HUP0202988A3 (en) Substituted 3-phenyl-5-alkoxi-1,3,4-oxdiazol-2-one derivatives and their use as lipase inhibitors, process for their preparation and pharmaceutical compositions containing them
BR0208655A (pt) Composição farmacêuticas
AP9801235A0 (en) Erythromycin derivatives.
ATE397615T1 (de) 6-o-alkyl-2-nor-2-substituierte ketolidderivate
AP9901559A0 (en) Tricyclic 3-keto derivatives of 6-0-methylerythromycin.
PT952157E (pt) Derivados 9a, 11b-desidro de 9-oxima-3-ceto-6-o-metileritromicina
HU9800835D0 (en) Pharmaceutical composition for treatment diseases causing by ascophaera apis
UA34056A (uk) Склад для профілактики алергодерматозів