ES2071334T3 - Analogos de anillos fusionados de nitrogeno conteniendo heterociclos no aromaticos. - Google Patents

Analogos de anillos fusionados de nitrogeno conteniendo heterociclos no aromaticos.

Info

Publication number
ES2071334T3
ES2071334T3 ES91918058T ES91918058T ES2071334T3 ES 2071334 T3 ES2071334 T3 ES 2071334T3 ES 91918058 T ES91918058 T ES 91918058T ES 91918058 T ES91918058 T ES 91918058T ES 2071334 T3 ES2071334 T3 ES 2071334T3
Authority
ES
Spain
Prior art keywords
analogs
containing non
rings containing
aromatic hetero
fused nitrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES91918058T
Other languages
English (en)
Spanish (es)
Inventor
Manoj C Desai
Harry R Howard
Terry J Rosen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Pfizer Corp SRL
Original Assignee
Pfizer Corp Belgium
Pfizer Corp SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium, Pfizer Corp SRL filed Critical Pfizer Corp Belgium
Application granted granted Critical
Publication of ES2071334T3 publication Critical patent/ES2071334T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Polyoxymethylene Polymers And Polymers With Carbon-To-Carbon Bonds (AREA)
  • Electroluminescent Light Sources (AREA)
  • Eye Examination Apparatus (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
ES91918058T 1990-09-28 1991-08-20 Analogos de anillos fusionados de nitrogeno conteniendo heterociclos no aromaticos. Expired - Lifetime ES2071334T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US59042390A 1990-09-28 1990-09-28

Publications (1)

Publication Number Publication Date
ES2071334T3 true ES2071334T3 (es) 1995-06-16

Family

ID=24362216

Family Applications (1)

Application Number Title Priority Date Filing Date
ES91918058T Expired - Lifetime ES2071334T3 (es) 1990-09-28 1991-08-20 Analogos de anillos fusionados de nitrogeno conteniendo heterociclos no aromaticos.

Country Status (22)

Country Link
EP (1) EP0550635B1 (enExample)
JP (1) JPH0772175B2 (enExample)
CN (1) CN1060285A (enExample)
AT (1) ATE121389T1 (enExample)
AU (1) AU651145B2 (enExample)
BR (1) BR9106905A (enExample)
CA (1) CA2089736A1 (enExample)
CZ (1) CZ387492A3 (enExample)
DE (1) DE69109125T2 (enExample)
DK (1) DK0550635T3 (enExample)
ES (1) ES2071334T3 (enExample)
FI (1) FI931370A7 (enExample)
HU (1) HUT68667A (enExample)
IE (1) IE66042B1 (enExample)
IL (1) IL99525A0 (enExample)
MX (1) MX9101274A (enExample)
NO (1) NO931151L (enExample)
PT (1) PT99064A (enExample)
TW (1) TW199144B (enExample)
WO (1) WO1992006079A1 (enExample)
YU (1) YU159291A (enExample)
ZA (1) ZA917744B (enExample)

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US6048859A (en) * 1992-06-29 2000-04-11 Merck & Co., Inc. Morpholine and thiomorpholine tachykinin receptor antagonists
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Also Published As

Publication number Publication date
NO931151D0 (no) 1993-03-26
HUT68667A (en) 1995-07-28
EP0550635A1 (en) 1993-07-14
WO1992006079A1 (en) 1992-04-16
IE913396A1 (en) 1992-04-08
PT99064A (pt) 1992-08-31
YU159291A (sh) 1994-01-20
ATE121389T1 (de) 1995-05-15
IE66042B1 (en) 1995-12-13
JPH06501267A (ja) 1994-02-10
MX9101274A (es) 1992-05-04
CA2089736A1 (en) 1992-03-29
BR9106905A (pt) 1993-08-17
FI931370A0 (fi) 1993-03-26
EP0550635B1 (en) 1995-04-19
IL99525A0 (en) 1992-08-18
CZ387492A3 (en) 1994-02-16
DE69109125T2 (de) 1995-09-28
JPH0772175B2 (ja) 1995-08-02
AU651145B2 (en) 1994-07-14
FI931370L (fi) 1993-03-26
DK0550635T3 (da) 1995-09-04
CN1060285A (zh) 1992-04-15
ZA917744B (en) 1993-03-29
HU9300898D0 (en) 1993-06-28
NO931151L (no) 1993-03-26
DE69109125D1 (de) 1995-05-24
TW199144B (enExample) 1993-02-01
AU8746391A (en) 1992-04-28
FI931370A7 (fi) 1993-03-26

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