ECSP11010930A - Nuevos compuestos químicos - Google Patents

Nuevos compuestos químicos

Info

Publication number
ECSP11010930A
ECSP11010930A EC2011010930A ECSP11010930A ECSP11010930A EC SP11010930 A ECSP11010930 A EC SP11010930A EC 2011010930 A EC2011010930 A EC 2011010930A EC SP11010930 A ECSP11010930 A EC SP11010930A EC SP11010930 A ECSP11010930 A EC SP11010930A
Authority
EC
Ecuador
Prior art keywords
chemical compounds
new chemical
treatment
radicals
excessive
Prior art date
Application number
EC2011010930A
Other languages
English (en)
Inventor
Peter Ettmayer
Andreas Mantoulidis
Steffen Steurer
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40019293&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP11010930(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of ECSP11010930A publication Critical patent/ECSP11010930A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Abstract

La presente invención comprende compuestos de la fórmula general (1),en donde los radicales R1 a R3, X1, X2, X3 y L1 se definen como en la reivindicación 1, los cuales son adecuados para el tratamiento de enfermedades que se caracterizan por una proliferación celular excesiva o anormal, así como su utilización en el caso de un tratamiento de este tipo.
EC2011010930A 2008-09-29 2011-03-29 Nuevos compuestos químicos ECSP11010930A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP08165437 2008-09-29

Publications (1)

Publication Number Publication Date
ECSP11010930A true ECSP11010930A (es) 2011-04-29

Family

ID=40019293

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2011010930A ECSP11010930A (es) 2008-09-29 2011-03-29 Nuevos compuestos químicos

Country Status (20)

Country Link
US (1) US8778929B2 (es)
EP (1) EP2350052B1 (es)
JP (1) JP5603869B2 (es)
KR (1) KR20110063574A (es)
CN (1) CN102227421A (es)
AR (1) AR073700A1 (es)
AU (1) AU2009295855A1 (es)
BR (1) BRPI0920608A2 (es)
CA (1) CA2738448A1 (es)
CL (1) CL2011000691A1 (es)
CO (1) CO6351739A2 (es)
EA (1) EA201100564A1 (es)
EC (1) ECSP11010930A (es)
IL (1) IL211744A0 (es)
MA (1) MA32656B1 (es)
MX (1) MX2011003292A (es)
PE (1) PE20110294A1 (es)
TW (1) TW201018670A (es)
UY (1) UY32146A (es)
WO (1) WO2010034838A2 (es)

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PT2861579T (pt) 2012-05-15 2018-04-27 Novartis Ag Derivados de benzamida para inibir a atividade de abl1, abl2 e bcr-abl
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JP6078640B2 (ja) 2012-05-15 2017-02-08 ノバルティス アーゲー Abl1、abl2およびbcr−abl1の活性を阻害するためのベンズアミド誘導体
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Also Published As

Publication number Publication date
WO2010034838A3 (en) 2010-11-18
CO6351739A2 (es) 2011-12-20
EP2350052B1 (en) 2014-08-13
BRPI0920608A2 (pt) 2019-09-24
EA201100564A1 (ru) 2011-12-30
KR20110063574A (ko) 2011-06-10
AR073700A1 (es) 2010-11-24
CL2011000691A1 (es) 2011-07-29
MX2011003292A (es) 2011-04-21
JP2012504114A (ja) 2012-02-16
TW201018670A (en) 2010-05-16
US8778929B2 (en) 2014-07-15
JP5603869B2 (ja) 2014-10-08
US20110312939A1 (en) 2011-12-22
EP2350052A2 (en) 2011-08-03
CA2738448A1 (en) 2010-04-01
CN102227421A (zh) 2011-10-26
WO2010034838A2 (en) 2010-04-01
UY32146A (es) 2010-04-30
MA32656B1 (fr) 2011-09-01
PE20110294A1 (es) 2011-05-26
AU2009295855A1 (en) 2010-04-01
IL211744A0 (en) 2011-06-30

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