ECSP067025A - DERIVADOS DE TETRAAZABENZO [e] AZULENO Y SUS ANÁLOGOS - Google Patents
DERIVADOS DE TETRAAZABENZO [e] AZULENO Y SUS ANÁLOGOSInfo
- Publication number
- ECSP067025A ECSP067025A EC2006007025A ECSP067025A ECSP067025A EC SP067025 A ECSP067025 A EC SP067025A EC 2006007025 A EC2006007025 A EC 2006007025A EC SP067025 A ECSP067025 A EC SP067025A EC SP067025 A ECSP067025 A EC SP067025A
- Authority
- EC
- Ecuador
- Prior art keywords
- azuleno
- tetraazabenzo
- analogs
- derivatives
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/24—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Esta invención se refiere a agonistas CCK-A de fórmula en que R1-R4, A, B, X, D, E y G son como se definen en la memoria descriptiva, así como, entre otras cosas, las composiciones farmacéuticas que contienen los compuestos y los métodos para usar los compuestos y composiciones. Los compuestos son útiles para tratar la obesidad.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US57403304P | 2004-05-25 | 2004-05-25 |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP067025A true ECSP067025A (es) | 2006-12-29 |
Family
ID=34967684
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EC2006007025A ECSP067025A (es) | 2004-05-25 | 2006-11-24 | DERIVADOS DE TETRAAZABENZO [e] AZULENO Y SUS ANÁLOGOS |
Country Status (26)
Country | Link |
---|---|
US (2) | US7265104B2 (es) |
EP (1) | EP1753766A1 (es) |
JP (1) | JP4069159B2 (es) |
CN (1) | CN1950374A (es) |
AP (1) | AP2006003768A0 (es) |
AR (1) | AR049187A1 (es) |
AU (1) | AU2005247693A1 (es) |
BR (1) | BRPI0510273A (es) |
CA (1) | CA2568056A1 (es) |
CR (1) | CR8753A (es) |
EA (1) | EA010888B1 (es) |
EC (1) | ECSP067025A (es) |
GE (1) | GEP20094723B (es) |
GT (1) | GT200500119A (es) |
IL (1) | IL178220A0 (es) |
MA (1) | MA28605B1 (es) |
NL (1) | NL1029105C2 (es) |
NO (1) | NO20064288L (es) |
PA (1) | PA8634101A1 (es) |
PE (1) | PE20060363A1 (es) |
SV (1) | SV2006002127A (es) |
TN (1) | TNSN06386A1 (es) |
TW (1) | TWI297688B (es) |
UA (1) | UA84208C2 (es) |
UY (1) | UY28915A1 (es) |
WO (1) | WO2005116034A1 (es) |
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-
2005
- 2005-05-13 GE GEAP20059708A patent/GEP20094723B/en unknown
- 2005-05-13 UA UAA200612379A patent/UA84208C2/ru unknown
- 2005-05-13 JP JP2007514174A patent/JP4069159B2/ja not_active Expired - Fee Related
- 2005-05-13 AU AU2005247693A patent/AU2005247693A1/en not_active Abandoned
- 2005-05-13 CN CNA2005800147946A patent/CN1950374A/zh active Pending
- 2005-05-13 CA CA002568056A patent/CA2568056A1/en not_active Abandoned
- 2005-05-13 AP AP2006003768A patent/AP2006003768A0/xx unknown
- 2005-05-13 BR BRPI0510273-1A patent/BRPI0510273A/pt not_active IP Right Cessation
- 2005-05-13 EA EA200601773A patent/EA010888B1/ru not_active IP Right Cessation
- 2005-05-13 EP EP05739440A patent/EP1753766A1/en not_active Withdrawn
- 2005-05-13 WO PCT/IB2005/001469 patent/WO2005116034A1/en active Application Filing
- 2005-05-19 US US11/134,790 patent/US7265104B2/en not_active Expired - Fee Related
- 2005-05-20 GT GT200500119A patent/GT200500119A/es unknown
- 2005-05-23 PE PE2005000568A patent/PE20060363A1/es not_active Application Discontinuation
- 2005-05-23 AR ARP050102117A patent/AR049187A1/es not_active Application Discontinuation
- 2005-05-23 UY UY28915A patent/UY28915A1/es not_active Application Discontinuation
- 2005-05-24 PA PA20058634101A patent/PA8634101A1/es unknown
- 2005-05-24 NL NL1029105A patent/NL1029105C2/nl not_active IP Right Cessation
- 2005-05-24 TW TW094116913A patent/TWI297688B/zh active
- 2005-05-25 SV SV2005002127A patent/SV2006002127A/es not_active Application Discontinuation
-
2006
- 2006-09-20 IL IL178220A patent/IL178220A0/en unknown
- 2006-09-21 NO NO20064288A patent/NO20064288L/no not_active Application Discontinuation
- 2006-11-16 CR CR8753A patent/CR8753A/es not_active Application Discontinuation
- 2006-11-24 MA MA29486A patent/MA28605B1/fr unknown
- 2006-11-24 TN TNP2006000386A patent/TNSN06386A1/fr unknown
- 2006-11-24 EC EC2006007025A patent/ECSP067025A/es unknown
-
2007
- 2007-07-20 US US11/780,988 patent/US7358242B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
NL1029105A1 (nl) | 2005-11-30 |
EA010888B1 (ru) | 2008-12-30 |
MA28605B1 (fr) | 2007-05-02 |
CA2568056A1 (en) | 2005-12-08 |
TNSN06386A1 (fr) | 2008-02-22 |
NL1029105C2 (nl) | 2006-06-13 |
AP2006003768A0 (en) | 2006-10-31 |
PE20060363A1 (es) | 2006-05-08 |
WO2005116034A1 (en) | 2005-12-08 |
GEP20094723B (en) | 2009-07-10 |
SV2006002127A (es) | 2006-02-15 |
JP4069159B2 (ja) | 2008-04-02 |
TW200609235A (en) | 2006-03-16 |
US20070265193A1 (en) | 2007-11-15 |
TWI297688B (en) | 2008-06-11 |
CR8753A (es) | 2006-12-13 |
AU2005247693A1 (en) | 2005-12-08 |
UA84208C2 (en) | 2008-09-25 |
JP2008500326A (ja) | 2008-01-10 |
US7265104B2 (en) | 2007-09-04 |
IL178220A0 (en) | 2006-12-31 |
UY28915A1 (es) | 2005-12-30 |
EP1753766A1 (en) | 2007-02-21 |
BRPI0510273A (pt) | 2007-10-30 |
CN1950374A (zh) | 2007-04-18 |
EA200601773A1 (ru) | 2007-06-29 |
GT200500119A (es) | 2006-01-12 |
US20050267100A1 (en) | 2005-12-01 |
PA8634101A1 (es) | 2006-06-02 |
AR049187A1 (es) | 2006-07-05 |
NO20064288L (no) | 2006-10-23 |
US7358242B2 (en) | 2008-04-15 |
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