PA8634101A1 - DERIVADOS DE TETRAAZABENZO[e] AZULENO Y SUS ANALOGOS - Google Patents

DERIVADOS DE TETRAAZABENZO[e] AZULENO Y SUS ANALOGOS

Info

Publication number
PA8634101A1
PA8634101A1 PA20058634101A PA8634101A PA8634101A1 PA 8634101 A1 PA8634101 A1 PA 8634101A1 PA 20058634101 A PA20058634101 A PA 20058634101A PA 8634101 A PA8634101 A PA 8634101A PA 8634101 A1 PA8634101 A1 PA 8634101A1
Authority
PA
Panama
Prior art keywords
azuleno
tetraazabenzo
analogs
derivatives
compounds
Prior art date
Application number
PA20058634101A
Other languages
English (en)
Inventor
Marlys Hammond
Cameron Kimberly Okeefe
Richard Louis Elliott
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of PA8634101A1 publication Critical patent/PA8634101A1/es

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

ESTA INVENCION SE REFIERE A AGONISTAS CCK-A DE FORMULA EN QUE R1-R4, A, B, X, D, E Y G SON COMO SE DEFINEN EN LA MEMORIA DESCRIPTIVA, ASI COMO, ENTRE OTRAS COSAS, LAS COMPOSICIONES FARMACEUTICAS QUE CONTIENEN LOS COMPUESTOS Y LOS METODOS PARA USAR LOS COMPUESTOS Y COMPOSICIONES. LOS COMPUESTOS SON UTILES PARA TRATAR LA OBESIDAD.
PA20058634101A 2004-05-25 2005-05-24 DERIVADOS DE TETRAAZABENZO[e] AZULENO Y SUS ANALOGOS PA8634101A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US57403304P 2004-05-25 2004-05-25

Publications (1)

Publication Number Publication Date
PA8634101A1 true PA8634101A1 (es) 2006-06-02

Family

ID=34967684

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20058634101A PA8634101A1 (es) 2004-05-25 2005-05-24 DERIVADOS DE TETRAAZABENZO[e] AZULENO Y SUS ANALOGOS

Country Status (26)

Country Link
US (2) US7265104B2 (es)
EP (1) EP1753766A1 (es)
JP (1) JP4069159B2 (es)
CN (1) CN1950374A (es)
AP (1) AP2006003768A0 (es)
AR (1) AR049187A1 (es)
AU (1) AU2005247693A1 (es)
BR (1) BRPI0510273A (es)
CA (1) CA2568056A1 (es)
CR (1) CR8753A (es)
EA (1) EA010888B1 (es)
EC (1) ECSP067025A (es)
GE (1) GEP20094723B (es)
GT (1) GT200500119A (es)
IL (1) IL178220A0 (es)
MA (1) MA28605B1 (es)
NL (1) NL1029105C2 (es)
NO (1) NO20064288L (es)
PA (1) PA8634101A1 (es)
PE (1) PE20060363A1 (es)
SV (1) SV2006002127A (es)
TN (1) TNSN06386A1 (es)
TW (1) TWI297688B (es)
UA (1) UA84208C2 (es)
UY (1) UY28915A1 (es)
WO (1) WO2005116034A1 (es)

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UY28915A1 (es) 2005-12-30
AR049187A1 (es) 2006-07-05
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SV2006002127A (es) 2006-02-15
UA84208C2 (en) 2008-09-25
AP2006003768A0 (en) 2006-10-31
CN1950374A (zh) 2007-04-18
NO20064288L (no) 2006-10-23
EA010888B1 (ru) 2008-12-30
BRPI0510273A (pt) 2007-10-30
TWI297688B (en) 2008-06-11
US20070265193A1 (en) 2007-11-15
EP1753766A1 (en) 2007-02-21
JP2008500326A (ja) 2008-01-10
AU2005247693A1 (en) 2005-12-08
MA28605B1 (fr) 2007-05-02
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US7265104B2 (en) 2007-09-04
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PE20060363A1 (es) 2006-05-08
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US7358242B2 (en) 2008-04-15
IL178220A0 (en) 2006-12-31
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