CR10060A - 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas - Google Patents

3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas

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Publication number
CR10060A
CR10060A CR10060A CR10060A CR10060A CR 10060 A CR10060 A CR 10060A CR 10060 A CR10060 A CR 10060A CR 10060 A CR10060 A CR 10060A CR 10060 A CR10060 A CR 10060A
Authority
CR
Costa Rica
Prior art keywords
chemiokin
aminociclopentanocarboxamids
receptors modulators
receptors
compounds
Prior art date
Application number
CR10060A
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English (en)
Inventor
Xue Chu-Biao
Original Assignee
Incyte Corp
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38126410&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR10060(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Incyte Corp filed Critical Incyte Corp
Publication of CR10060A publication Critical patent/CR10060A/es

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D498/04—Ortho-condensed systems

Abstract

La presente invención se refiere a compuestos de Fórmula I: que son moduladores de receptores de quimioquinas. Los compuestos de la invención, y las composiciones de los mismos, son útiles en el tratamiento de enfermedades relacionadas con la expresión y/o actividad de receptores de quimioquinas.
CR10060A 2005-12-21 2008-06-10 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas CR10060A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75232005P 2005-12-21 2005-12-21
US75247705P 2005-12-21 2005-12-21

Publications (1)

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CR10060A true CR10060A (es) 2008-07-17

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CR10060A CR10060A (es) 2005-12-21 2008-06-10 3-aminociclopentanocarboxamidas como moduladores de receptores de quimioquinas

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US (2) US7700624B2 (es)
EP (1) EP1971576A2 (es)
JP (1) JP2009520809A (es)
KR (1) KR20080070868A (es)
AP (1) AP2008004487A0 (es)
AR (1) AR058402A1 (es)
AU (1) AU2006327823A1 (es)
BR (1) BRPI0620073A2 (es)
CA (1) CA2634636A1 (es)
CR (1) CR10060A (es)
EA (1) EA200801220A1 (es)
EC (1) ECSP088527A (es)
IL (1) IL191602A0 (es)
MA (1) MA30077B1 (es)
ME (1) MEP1008A (es)
NL (1) NL2000380C2 (es)
NO (1) NO20082285L (es)
RS (1) RS20080246A (es)
TW (1) TW200734323A (es)
UY (1) UY30052A1 (es)
WO (1) WO2007072201A2 (es)

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MEP1008A (xx) * 2005-12-21 2010-02-10 Incyte Corp 3-aminociklopentankarboksamidi kao modulatori receptora hemokina
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WO2016020295A1 (en) 2014-08-04 2016-02-11 Nuevolution A/S Optionally fused heterocyclyl-substituted derivatives of pyrimidine useful for the treatment of inflammatory, metabolic, oncologic and autoimmune diseases
AU2020405446A1 (en) 2019-12-20 2022-05-26 Nuevolution A/S Compounds active towards nuclear receptors
EP4126874A1 (en) 2020-03-31 2023-02-08 Nuevolution A/S Compounds active towards nuclear receptors
WO2021198956A1 (en) 2020-03-31 2021-10-07 Nuevolution A/S Compounds active towards nuclear receptors

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UY30052A1 (es) 2007-07-31
AR058402A1 (es) 2008-01-30
AU2006327823A1 (en) 2007-06-28
TW200734323A (en) 2007-09-16
BRPI0620073A2 (pt) 2011-11-01
MEP1008A (xx) 2010-02-10
EP1971576A2 (en) 2008-09-24
KR20080070868A (ko) 2008-07-31
US20070149532A1 (en) 2007-06-28
EA200801220A1 (ru) 2008-12-30
NO20082285L (no) 2008-06-18
WO2007072201A2 (en) 2007-06-28
CA2634636A1 (en) 2007-06-28
NL2000380C2 (nl) 2007-11-28
US7700624B2 (en) 2010-04-20
RS20080246A (en) 2009-07-15
MA30077B1 (fr) 2008-12-01
WO2007072201A3 (en) 2007-10-04
US20100203039A1 (en) 2010-08-12
AP2008004487A0 (en) 2008-06-30
NL2000380A1 (nl) 2007-06-25
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JP2009520809A (ja) 2009-05-28
IL191602A0 (en) 2009-02-11

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