EA201190224A1 - Ингибиторы гепатита c, содержащие конденсированные кольца - Google Patents
Ингибиторы гепатита c, содержащие конденсированные кольцаInfo
- Publication number
- EA201190224A1 EA201190224A1 EA201190224A EA201190224A EA201190224A1 EA 201190224 A1 EA201190224 A1 EA 201190224A1 EA 201190224 A EA201190224 A EA 201190224A EA 201190224 A EA201190224 A EA 201190224A EA 201190224 A1 EA201190224 A1 EA 201190224A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- hepatitis
- condensed rings
- containing condensed
- inhibitors containing
- inhibitors
- Prior art date
Links
- 208000006454 hepatitis Diseases 0.000 title 1
- 231100000283 hepatitis Toxicity 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 208000005176 Hepatitis C Diseases 0.000 abstract 1
- 238000002648 combination therapy Methods 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Gastroenterology & Hepatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US16434209P | 2009-03-27 | 2009-03-27 | |
| US21488309P | 2009-04-28 | 2009-04-28 | |
| PCT/US2010/028730 WO2010111534A1 (en) | 2009-03-27 | 2010-03-25 | Fused ring inhibitors of hepatitis c |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| EA201190224A1 true EA201190224A1 (ru) | 2012-03-30 |
Family
ID=42781523
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA201190224A EA201190224A1 (ru) | 2009-03-27 | 2010-03-25 | Ингибиторы гепатита c, содержащие конденсированные кольца |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US9150554B2 (enExample) |
| EP (1) | EP2410843A4 (enExample) |
| JP (1) | JP5735482B2 (enExample) |
| KR (1) | KR20110131312A (enExample) |
| CN (1) | CN102427726B (enExample) |
| AR (1) | AR076164A1 (enExample) |
| AU (1) | AU2010229795A1 (enExample) |
| BR (1) | BRPI1012282A2 (enExample) |
| CA (1) | CA2755658A1 (enExample) |
| CL (1) | CL2011002377A1 (enExample) |
| CO (1) | CO6450600A2 (enExample) |
| EA (1) | EA201190224A1 (enExample) |
| IL (1) | IL215202A0 (enExample) |
| MX (1) | MX2011010132A (enExample) |
| PE (1) | PE20120773A1 (enExample) |
| SG (1) | SG174883A1 (enExample) |
| TW (1) | TW201038560A (enExample) |
| WO (1) | WO2010111534A1 (enExample) |
| ZA (1) | ZA201107753B (enExample) |
Families Citing this family (102)
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| US8242156B2 (en) | 2009-02-17 | 2012-08-14 | Enanta Pharmaceuticals, Inc. | Linked dibenzimidazole derivatives |
| US8188132B2 (en) | 2009-02-17 | 2012-05-29 | Enanta Pharmaceuticals, Inc. | Linked dibenzimidazole derivatives |
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| US8673954B2 (en) | 2009-02-27 | 2014-03-18 | Enanta Pharmaceuticals, Inc. | Benzimidazole derivatives |
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| US9765087B2 (en) | 2009-02-27 | 2017-09-19 | Enanta Pharmaceuticals, Inc. | Benzimidazole derivatives |
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| KR101387274B1 (ko) | 2009-03-27 | 2014-04-25 | 머크 샤프 앤드 돔 코포레이션 | Ｃ형 간염 바이러스 복제의 억제제 |
| US8796466B2 (en) | 2009-03-30 | 2014-08-05 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| TW201038559A (en) | 2009-04-09 | 2010-11-01 | Bristol Myers Squibb Co | Hepatitis C virus inhibitors |
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| JP5734956B2 (ja) | 2009-04-15 | 2015-06-17 | アッヴィ・インコーポレイテッド | 抗ウィルス化合物 |
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| AR077060A1 (es) | 2009-06-11 | 2011-07-27 | Abbott Lab | Compuestos antivirales |
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-
2010
- 2010-03-25 EP EP10756872A patent/EP2410843A4/en not_active Withdrawn
- 2010-03-25 CN CN201080021446.2A patent/CN102427726B/zh not_active Expired - Fee Related
- 2010-03-25 SG SG2011067683A patent/SG174883A1/en unknown
- 2010-03-25 AU AU2010229795A patent/AU2010229795A1/en not_active Abandoned
- 2010-03-25 WO PCT/US2010/028730 patent/WO2010111534A1/en not_active Ceased
- 2010-03-25 KR KR1020117025221A patent/KR20110131312A/ko not_active Withdrawn
- 2010-03-25 MX MX2011010132A patent/MX2011010132A/es active IP Right Grant
- 2010-03-25 JP JP2012502264A patent/JP5735482B2/ja not_active Expired - Fee Related
- 2010-03-25 PE PE2011001719A patent/PE20120773A1/es not_active Application Discontinuation
- 2010-03-25 BR BRPI1012282A patent/BRPI1012282A2/pt not_active IP Right Cessation
- 2010-03-25 US US13/260,378 patent/US9150554B2/en not_active Expired - Fee Related
- 2010-03-25 CA CA2755658A patent/CA2755658A1/en not_active Abandoned
- 2010-03-25 EA EA201190224A patent/EA201190224A1/ru unknown
- 2010-03-26 TW TW099109325A patent/TW201038560A/zh unknown
- 2010-03-29 AR ARP100101000A patent/AR076164A1/es unknown
-
2011
- 2011-09-18 IL IL215202A patent/IL215202A0/en unknown
- 2011-09-26 CL CL2011002377A patent/CL2011002377A1/es unknown
- 2011-10-24 ZA ZA2011/07753A patent/ZA201107753B/en unknown
- 2011-10-27 CO CO11145231A patent/CO6450600A2/es active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| EP2410843A1 (en) | 2012-02-01 |
| HK1166446A1 (en) | 2012-11-02 |
| CN102427726A (zh) | 2012-04-25 |
| AR076164A1 (es) | 2011-05-26 |
| CO6450600A2 (es) | 2012-05-31 |
| CN102427726B (zh) | 2014-10-08 |
| EP2410843A4 (en) | 2012-08-08 |
| SG174883A1 (en) | 2011-11-28 |
| KR20110131312A (ko) | 2011-12-06 |
| AU2010229795A1 (en) | 2011-10-13 |
| WO2010111534A1 (en) | 2010-09-30 |
| TW201038560A (en) | 2010-11-01 |
| CA2755658A1 (en) | 2010-09-30 |
| BRPI1012282A2 (pt) | 2015-09-22 |
| ZA201107753B (en) | 2012-07-25 |
| US20120040962A1 (en) | 2012-02-16 |
| MX2011010132A (es) | 2011-10-14 |
| US9150554B2 (en) | 2015-10-06 |
| IL215202A0 (en) | 2011-12-29 |
| JP2012522003A (ja) | 2012-09-20 |
| JP5735482B2 (ja) | 2015-06-17 |
| CL2011002377A1 (es) | 2012-01-20 |
| PE20120773A1 (es) | 2012-07-19 |
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