EA200100444A1 - Производные гигромицина а в качестве антибактериальных агентов - Google Patents
Производные гигромицина а в качестве антибактериальных агентовInfo
- Publication number
- EA200100444A1 EA200100444A1 EA200100444A EA200100444A EA200100444A1 EA 200100444 A1 EA200100444 A1 EA 200100444A1 EA 200100444 A EA200100444 A EA 200100444A EA 200100444 A EA200100444 A EA 200100444A EA 200100444 A1 EA200100444 A1 EA 200100444A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- formula
- compounds
- hygromycin
- derivatives
- antibacterial agents
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/02—Local antiseptics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
Abstract
Данное изобретение относится к соединениям формулы (1) и их фармацевтически приемлемым солям и сольватам, где R, R, R, Xи Xтакие, как определено в материалах заявки. Соединения формулы (1) представляют собой антибактериальные и антипротозойные агенты, которые можно применять для лечения различных бактериальных и протозойных инфекций и расстройств, связанных с такими инфекциями. Данное изобретение также относится к фармацевтическим композициям, содержащим соединения формулы (1), способам лечения бактериальных и протозойных инфекций путем введения соединений формулы (1) и способам получения некоторых соединений формулы (1).Международная заявка была опубликована вместе с отчетом о международном поиске.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US11061898P | 1998-12-02 | 1998-12-02 | |
| PCT/IB1999/001798 WO2000032616A1 (en) | 1998-12-02 | 1999-11-09 | Hygromycin a derivatives as antibacterial agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EA200100444A1 true EA200100444A1 (ru) | 2001-10-22 |
| EA004303B1 EA004303B1 (ru) | 2004-02-26 |
Family
ID=22334003
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA200100444A EA004303B1 (ru) | 1998-12-02 | 1999-11-09 | Производные гигромицина а в качестве антибактериальных агентов |
Country Status (38)
| Country | Link |
|---|---|
| US (1) | US6245745B1 (ru) |
| EP (1) | EP1135400A1 (ru) |
| JP (1) | JP3393189B2 (ru) |
| KR (1) | KR100418167B1 (ru) |
| CN (1) | CN1329617A (ru) |
| AP (1) | AP2001002154A0 (ru) |
| AR (1) | AR019784A1 (ru) |
| AU (1) | AU6362799A (ru) |
| BG (1) | BG105645A (ru) |
| BR (1) | BR9915813A (ru) |
| CA (1) | CA2352332C (ru) |
| CO (1) | CO5150171A1 (ru) |
| CZ (1) | CZ20011904A3 (ru) |
| DZ (1) | DZ2932A1 (ru) |
| EA (1) | EA004303B1 (ru) |
| EE (1) | EE200100301A (ru) |
| GE (1) | GEP20033144B (ru) |
| GT (1) | GT199900205A (ru) |
| HN (1) | HN1999000202A (ru) |
| HR (1) | HRP20010413A2 (ru) |
| HU (1) | HUP0104949A3 (ru) |
| ID (1) | ID28848A (ru) |
| IL (1) | IL142882A0 (ru) |
| IS (1) | IS5930A (ru) |
| MA (1) | MA26705A1 (ru) |
| NO (1) | NO20012687L (ru) |
| NZ (1) | NZ511424A (ru) |
| OA (1) | OA11721A (ru) |
| PA (1) | PA8486101A1 (ru) |
| PE (1) | PE20001429A1 (ru) |
| PL (1) | PL348063A1 (ru) |
| SK (1) | SK7302001A3 (ru) |
| TN (1) | TNSN99211A1 (ru) |
| TR (1) | TR200101540T2 (ru) |
| UY (1) | UY25827A1 (ru) |
| WO (1) | WO2000032616A1 (ru) |
| YU (1) | YU32601A (ru) |
| ZA (1) | ZA200104434B (ru) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20020043255A (ko) * | 1999-10-29 | 2002-06-08 | 실버스타인 아써 에이. | 하이그로마이신 ａ 전구물질 |
| KR20020063885A (ko) * | 1999-10-29 | 2002-08-05 | 화이자 프로덕츠 인코포레이티드 | 하이그로마이신 유도체 |
| AU2001260528A1 (en) * | 2000-06-02 | 2001-12-11 | Pfizer Products Inc. | Hygromycin a derivatives for the treatment of bacterial and protozoal infections |
| WO2004112580A2 (en) * | 2003-06-19 | 2004-12-29 | Compumed, Inc. | Method and system for analyzing bone conditions using dicom compliant bone radiographic image |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| YU66900A (sh) * | 1998-05-04 | 2003-12-31 | Pfizer Products Inc. | Derivati higromicina a |
| ATE243218T1 (de) * | 1998-05-04 | 2003-07-15 | Pfizer Prod Inc | 2''-deoxyhygromycinderivate |
-
1999
- 1999-11-09 YU YU32601A patent/YU32601A/sh unknown
- 1999-11-09 TR TR2001/01540T patent/TR200101540T2/xx unknown
- 1999-11-09 EE EEP200100301A patent/EE200100301A/xx unknown
- 1999-11-09 OA OA1200100135A patent/OA11721A/en unknown
- 1999-11-09 GE GEAP19995922A patent/GEP20033144B/en unknown
- 1999-11-09 CN CN99813939A patent/CN1329617A/zh active Pending
- 1999-11-09 NZ NZ511424A patent/NZ511424A/en unknown
- 1999-11-09 IL IL14288299A patent/IL142882A0/xx unknown
- 1999-11-09 PL PL99348063A patent/PL348063A1/xx not_active Application Discontinuation
- 1999-11-09 AP APAP/P/2001/002154A patent/AP2001002154A0/en unknown
- 1999-11-09 EA EA200100444A patent/EA004303B1/ru not_active IP Right Cessation
- 1999-11-09 HU HU0104949A patent/HUP0104949A3/hu unknown
- 1999-11-09 BR BR9915813-2A patent/BR9915813A/pt not_active IP Right Cessation
- 1999-11-09 SK SK730-2001A patent/SK7302001A3/sk unknown
- 1999-11-09 JP JP2000585257A patent/JP3393189B2/ja not_active Expired - Fee Related
- 1999-11-09 EP EP99951055A patent/EP1135400A1/en not_active Withdrawn
- 1999-11-09 KR KR10-2001-7006849A patent/KR100418167B1/ko not_active IP Right Cessation
- 1999-11-09 WO PCT/IB1999/001798 patent/WO2000032616A1/en not_active Application Discontinuation
- 1999-11-09 AU AU63627/99A patent/AU6362799A/en not_active Abandoned
- 1999-11-09 ID IDW00200101182A patent/ID28848A/id unknown
- 1999-11-09 CA CA002352332A patent/CA2352332C/en not_active Expired - Fee Related
- 1999-11-09 CZ CZ20011904A patent/CZ20011904A3/cs unknown
- 1999-11-10 DZ DZ990232A patent/DZ2932A1/xx active
- 1999-11-10 TN TNTNSN99211A patent/TNSN99211A1/fr unknown
- 1999-11-10 MA MA25843A patent/MA26705A1/fr unknown
- 1999-11-15 AR ARP990105799A patent/AR019784A1/es not_active Application Discontinuation
- 1999-11-18 HN HN1999000202A patent/HN1999000202A/es unknown
- 1999-11-25 CO CO99074411A patent/CO5150171A1/es unknown
- 1999-11-29 PE PE1999001195A patent/PE20001429A1/es not_active Application Discontinuation
- 1999-11-30 UY UY25827A patent/UY25827A1/es unknown
- 1999-11-30 PA PA19998486101A patent/PA8486101A1/es unknown
- 1999-12-01 GT GT199900205A patent/GT199900205A/es unknown
- 1999-12-02 US US09/453,429 patent/US6245745B1/en not_active Expired - Fee Related
-
2001
- 2001-04-27 IS IS5930A patent/IS5930A/is unknown
- 2001-05-29 HR HR20010413A patent/HRP20010413A2/hr not_active Application Discontinuation
- 2001-05-30 ZA ZA200104434A patent/ZA200104434B/en unknown
- 2001-05-31 NO NO20012687A patent/NO20012687L/no not_active Application Discontinuation
- 2001-06-25 BG BG105645A patent/BG105645A/bg unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |