PA8486101A1 - Derivados de higromicina - Google Patents

Derivados de higromicina

Info

Publication number
PA8486101A1
PA8486101A1 PA19998486101A PA8486101A PA8486101A1 PA 8486101 A1 PA8486101 A1 PA 8486101A1 PA 19998486101 A PA19998486101 A PA 19998486101A PA 8486101 A PA8486101 A PA 8486101A PA 8486101 A1 PA8486101 A1 PA 8486101A1
Authority
PA
Panama
Prior art keywords
infections
compounds
hygromycin
derivatives
hygromycin derivatives
Prior art date
Application number
PA19998486101A
Other languages
English (en)
Inventor
Matthew Merrill Hayward
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of PA8486101A1 publication Critical patent/PA8486101A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/02Local antiseptics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

LA PRESENTE INVENCI¾N SE REFIERE A COMPUESTOS FORMULADOS Y ASALES Y SOLVATOS FARMACÚUTICAMENTE ACEPTABLE DE LOS MISMOS, DONDE R1,R2,R3, X1 Y X2 SON COMO SE DEFINEN EN ESTE DOCUMEN-TO. LOS COMPUESTOS DE F¾RMULA 1 SON AGENTES ANTIBACTERIANOS Y ANTIPROTOZOARIOS QUE PUEDEN USARSE PARA TRATAR DIVERSAS INFECCIONES BACTERIANAS Y PROTOZOARIAS Y TRASTORNOS RELACIONADOS CON TALES INFECCIONES.
PA19998486101A 1998-12-02 1999-11-30 Derivados de higromicina PA8486101A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11061898P 1998-12-02 1998-12-02

Publications (1)

Publication Number Publication Date
PA8486101A1 true PA8486101A1 (es) 2000-09-29

Family

ID=22334003

Family Applications (1)

Application Number Title Priority Date Filing Date
PA19998486101A PA8486101A1 (es) 1998-12-02 1999-11-30 Derivados de higromicina

Country Status (38)

Country Link
US (1) US6245745B1 (es)
EP (1) EP1135400A1 (es)
JP (1) JP3393189B2 (es)
KR (1) KR100418167B1 (es)
CN (1) CN1329617A (es)
AP (1) AP2001002154A0 (es)
AR (1) AR019784A1 (es)
AU (1) AU6362799A (es)
BG (1) BG105645A (es)
BR (1) BR9915813A (es)
CA (1) CA2352332C (es)
CO (1) CO5150171A1 (es)
CZ (1) CZ20011904A3 (es)
DZ (1) DZ2932A1 (es)
EA (1) EA004303B1 (es)
EE (1) EE200100301A (es)
GE (1) GEP20033144B (es)
GT (1) GT199900205A (es)
HN (1) HN1999000202A (es)
HR (1) HRP20010413A2 (es)
HU (1) HUP0104949A3 (es)
ID (1) ID28848A (es)
IL (1) IL142882A0 (es)
IS (1) IS5930A (es)
MA (1) MA26705A1 (es)
NO (1) NO20012687D0 (es)
NZ (1) NZ511424A (es)
OA (1) OA11721A (es)
PA (1) PA8486101A1 (es)
PE (1) PE20001429A1 (es)
PL (1) PL348063A1 (es)
SK (1) SK7302001A3 (es)
TN (1) TNSN99211A1 (es)
TR (1) TR200101540T2 (es)
UY (1) UY25827A1 (es)
WO (1) WO2000032616A1 (es)
YU (1) YU32601A (es)
ZA (1) ZA200104434B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2389019A1 (en) * 1999-10-29 2001-05-03 Pfizer Products Inc. Hygromycin a prodrugs
EP1224197A1 (en) * 1999-10-29 2002-07-24 Pfizer Products Inc. Hygromycin derivatives
EA200201167A1 (ru) 2000-06-02 2003-06-26 Пфайзер Продактс Инк. Производные гигромицина а для лечения бактериальных и протозойных инфекций
EP1643901A4 (en) * 2003-06-19 2008-10-29 Compumed Inc METHOD AND SYSTEM FOR ANALYZING BONE CONDITIONS USING A RADIOGRAPHIC IMAGE OF COMPATIBLE DICOM OS

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL344521A1 (en) * 1998-05-04 2001-11-05 Pfizer Prod Inc Hygromycin a derivatives
AU762302B2 (en) * 1998-05-04 2003-06-19 Pfizer Products Inc. 2"-deoxy hygromycin derivatives

Also Published As

Publication number Publication date
EP1135400A1 (en) 2001-09-26
NO20012687L (no) 2001-05-31
BR9915813A (pt) 2001-08-21
CN1329617A (zh) 2002-01-02
OA11721A (en) 2005-01-25
IL142882A0 (en) 2002-03-10
NZ511424A (en) 2003-08-29
US6245745B1 (en) 2001-06-12
PE20001429A1 (es) 2000-12-18
YU32601A (sh) 2004-05-12
BG105645A (bg) 2002-02-28
GEP20033144B (en) 2003-12-25
TNSN99211A1 (fr) 2005-11-10
TR200101540T2 (tr) 2001-10-22
UY25827A1 (es) 2001-08-27
HRP20010413A2 (en) 2002-06-30
KR20010093136A (ko) 2001-10-27
HUP0104949A2 (hu) 2002-04-29
AR019784A1 (es) 2002-03-13
AP2001002154A0 (en) 2001-05-09
EE200100301A (et) 2002-08-15
GT199900205A (es) 2001-05-24
ID28848A (id) 2001-07-05
CA2352332C (en) 2004-12-07
PL348063A1 (en) 2002-05-06
AU6362799A (en) 2000-06-19
HUP0104949A3 (en) 2003-12-29
EA200100444A1 (ru) 2001-10-22
EA004303B1 (ru) 2004-02-26
CZ20011904A3 (cs) 2001-10-17
IS5930A (is) 2001-04-27
ZA200104434B (en) 2002-05-30
NO20012687D0 (no) 2001-05-31
CO5150171A1 (es) 2002-04-29
KR100418167B1 (ko) 2004-02-11
DZ2932A1 (fr) 2004-03-15
HN1999000202A (es) 2000-06-13
MA26705A1 (fr) 2004-12-20
WO2000032616A1 (en) 2000-06-08
JP3393189B2 (ja) 2003-04-07
JP2002531463A (ja) 2002-09-24
CA2352332A1 (en) 2000-06-08
SK7302001A3 (en) 2001-12-03

Similar Documents

Publication Publication Date Title
PT618190E (pt) 9-¬glicil substituido)amido|-6-(substituido)-5-hidroxi-6-desoxitetraciclinas
ES2161220T3 (es) 9-((glicil sustituido)amido)-6-desmetil-6-desoxitetraciclinas como agentes antibioticos.
PA8486001A1 (es) Composiciones de celecoxib
MX9700557A (es) Dihidrobenzofuranos.
LV12358A (lv) 7-(Aizvietoti)-9-(aizvietoti glicil)-amido-6-demetil-6-deoksitetraciklini
DE69612003T2 (de) Substituierte benzolaktamverbindungen als substanz-p-antagonisten
YU40997A (sh) Novi oksadiazoli, postupci za njihovo pripremanje
ES2092113T3 (es) Derivados fluoroalcoxibencilamino de heterociclos que contienen nitrogeno.
ME00768B (me) Derivati supstituisanih benzol sulfonamida kao pro-lekovi cox-2 inhibitora
ES2127946T3 (es) Antagonistas de neurocinina diazabiciclica.
PT1140944E (pt) Derivados de epotilona e sua utilizacao como agentes antitumorais
ES2170102T3 (es) Aminociclohexilesteres y utilizacion de los mismos.
PL343495A1 (en) Heterocyclically substituted amides used as calpain inhibitors
IT1285770B1 (it) Composti corticoidei
BR0109512A (pt) Imidazopiridinas tricìclicas
AR020563A1 (es) Compuestos (poli)tia-alquinoicos y sus derivados, composiciones que los incluyen y su utilizacion
SE9801494D0 (sv) Novel use
HU9500559D0 (en) New mercapto-acetamide tricyclic derivatives as enkephalinase-inhibitors
PA8486101A1 (es) Derivados de higromicina
BG105008A (en) Hygromycin a derivatives
BG104292A (en) Methods and compositions for the treatment of rheumatoid arthritis
SV1999000159A (es) Antibioticos de carbamato y carbazato cetolida ref.pc10406abcz/bb
PA8471901A1 (es) Derivados de 2"-desoxi higromicina
UY26741A1 (es) Derivados de higromicina a
PT1144348E (pt) Inibidores de lta, hidrolase