YU66900A - Derivati higromicina a - Google Patents
Derivati higromicina aInfo
- Publication number
- YU66900A YU66900A YU66900A YU66900A YU66900A YU 66900 A YU66900 A YU 66900A YU 66900 A YU66900 A YU 66900A YU 66900 A YU66900 A YU 66900A YU 66900 A YU66900 A YU 66900A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- compounds
- formula
- infections
- relates
- hygromycin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
- C12P19/00—Preparation of compounds containing saccharide radicals
- C12P19/44—Preparation of O-glycosides, e.g. glucosides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biotechnology (AREA)
- Veterinary Medicine (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Engineering & Computer Science (AREA)
- Oncology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Microbiology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Abstract
Pronalazak se odnosi na jedinjenja formule 1 i na njihove farmaceutski prihvatljive soli, prekursore lekova i solvate, gde su R1 i R2 kao što je ovde definisano. Jedinjenja formule (1) pokazuju antibakterijska i antiprotozozolna dejstva. Pronalazak se odnosi na farmaceutske preparate koji sadrže jedinjenja formule (1) koji takodje imaju antibakterijske i antiprotozoalne osobine.[The invention relates to compounds of formula (1) and to pharmaceutically acceptable salts, prodrugs and solvates thereof, wherein R1 and R2 are as defined herein. The compounds of formula (1) are antibacterial and antiprotozoal agents that may be used to treat various bacterial and protozoal infections and disorders related to such infections. The invention also relates to pharmaceutical compositions containing the compounds of formula (1) and the methods of treating bacterial and protozoal infections by administering the compounds of formula (1).
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8404298P | 1998-05-04 | 1998-05-04 |
Publications (1)
Publication Number | Publication Date |
---|---|
YU66900A true YU66900A (sh) | 2003-12-31 |
Family
ID=22182520
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
YU66900A YU66900A (sh) | 1998-05-04 | 1999-05-03 | Derivati higromicina a |
Country Status (37)
Country | Link |
---|---|
US (1) | US6313100B1 (sh) |
EP (1) | EP1075483B1 (sh) |
JP (1) | JP2002513796A (sh) |
KR (1) | KR100402560B1 (sh) |
CN (1) | CN1299365A (sh) |
AP (3) | AP0102296A0 (sh) |
AR (1) | AR016251A1 (sh) |
AT (2) | ATE255588T1 (sh) |
AU (1) | AU755806B2 (sh) |
BG (1) | BG105008A (sh) |
BR (1) | BR9910206A (sh) |
CA (1) | CA2331297C (sh) |
DE (2) | DE69929723D1 (sh) |
DK (1) | DK1075483T3 (sh) |
DZ (1) | DZ2780A1 (sh) |
EA (2) | EA200200779A1 (sh) |
ES (1) | ES2209419T3 (sh) |
GT (1) | GT199900064A (sh) |
HR (1) | HRP20000747A2 (sh) |
HU (1) | HUP0102066A3 (sh) |
ID (1) | ID27030A (sh) |
IL (1) | IL139165A0 (sh) |
IS (1) | IS5681A (sh) |
MA (1) | MA24852A1 (sh) |
NO (1) | NO20005552L (sh) |
NZ (1) | NZ507452A (sh) |
OA (1) | OA11508A (sh) |
PA (1) | PA8471801A1 (sh) |
PE (1) | PE20000478A1 (sh) |
PL (1) | PL344521A1 (sh) |
PT (1) | PT1075483E (sh) |
SK (1) | SK16452000A3 (sh) |
TN (1) | TNSN99083A1 (sh) |
TR (1) | TR200003250T2 (sh) |
WO (1) | WO1999057125A2 (sh) |
YU (1) | YU66900A (sh) |
ZA (1) | ZA993064B (sh) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CZ20011904A3 (cs) * | 1998-12-02 | 2001-10-17 | Pfizer Products Inc. | Deriváty hygromycinu jako antibakteriální činidla |
GB9923078D0 (en) * | 1999-09-29 | 1999-12-01 | Phytopharm Plc | Sapogenin derivatives and their use |
US6771019B1 (en) * | 1999-05-14 | 2004-08-03 | Ifire Technology, Inc. | Electroluminescent laminate with patterned phosphor structure and thick film dielectric with improved dielectric properties |
EE200200671A (et) * | 2000-06-02 | 2004-08-16 | Pfizer Products Inc. | Hügromütsiin A derivaadid bakteriaalsete ja algloomadest põhjustatud infektsioonide ravimiseks |
CN102168034B (zh) * | 2010-11-29 | 2012-12-05 | 中国科学院南海海洋研究所 | 一种海洋链霉菌以及利用该菌制备替达霉素a和b的方法 |
JP2016069333A (ja) * | 2014-09-30 | 2016-05-09 | 公益財団法人微生物化学研究会 | 新規化合物、その製造方法、及びその用途、並びに、新規微生物 |
CN104480039B (zh) * | 2014-11-25 | 2017-09-12 | 辽宁大学 | 抗生素产生菌及其应用 |
WO2020041179A1 (en) * | 2018-08-20 | 2020-02-27 | Northeastern University | Hygromycin a compounds and methods of treating spirochete diseases |
TWI771766B (zh) | 2019-10-04 | 2022-07-21 | 美商輝瑞股份有限公司 | 二醯基甘油醯基轉移酶2 抑制劑 |
JP2022058085A (ja) | 2020-02-24 | 2022-04-11 | ファイザー・インク | ジアシルグリセロールアシルトランスフェラーゼ2阻害剤とアセチル-CoAカルボキシラーゼ阻害剤との組合せ |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0213692B1 (en) | 1985-06-27 | 1990-09-26 | Takeda Chemical Industries, Ltd. | Use of hygromycin and epihygromycin in the treatment of swine dysentery |
GB8605245D0 (en) | 1986-03-04 | 1986-04-09 | Fujisawa Pharmaceutical Co | Prophylactic & therapeutic agent |
-
1999
- 1999-05-03 EA EA200200779A patent/EA200200779A1/ru unknown
- 1999-05-03 EP EP99914722A patent/EP1075483B1/en not_active Expired - Lifetime
- 1999-05-03 DK DK99914722T patent/DK1075483T3/da active
- 1999-05-03 TR TR2000/03250T patent/TR200003250T2/xx unknown
- 1999-05-03 GT GT199900064A patent/GT199900064A/es unknown
- 1999-05-03 PT PT99914722T patent/PT1075483E/pt unknown
- 1999-05-03 DZ DZ990080A patent/DZ2780A1/xx active
- 1999-05-03 AP APAP/P/2001/002296A patent/AP0102296A0/en unknown
- 1999-05-03 SK SK1645-2000A patent/SK16452000A3/sk unknown
- 1999-05-03 AU AU33419/99A patent/AU755806B2/en not_active Ceased
- 1999-05-03 KR KR10-2000-7012266A patent/KR100402560B1/ko not_active IP Right Cessation
- 1999-05-03 ID IDW20002255A patent/ID27030A/id unknown
- 1999-05-03 ZA ZA9903064A patent/ZA993064B/xx unknown
- 1999-05-03 TN TNTNSN99083A patent/TNSN99083A1/fr unknown
- 1999-05-03 WO PCT/IB1999/000795 patent/WO1999057125A2/en active Search and Examination
- 1999-05-03 BR BR9910206-4A patent/BR9910206A/pt not_active IP Right Cessation
- 1999-05-03 DE DE69929723T patent/DE69929723D1/de not_active Expired - Lifetime
- 1999-05-03 CN CN99805807A patent/CN1299365A/zh active Pending
- 1999-05-03 DE DE69913333T patent/DE69913333T2/de not_active Expired - Fee Related
- 1999-05-03 US US09/462,592 patent/US6313100B1/en not_active Expired - Fee Related
- 1999-05-03 PE PE1999000362A patent/PE20000478A1/es not_active Application Discontinuation
- 1999-05-03 JP JP2000547094A patent/JP2002513796A/ja active Pending
- 1999-05-03 YU YU66900A patent/YU66900A/sh unknown
- 1999-05-03 AT AT99914722T patent/ATE255588T1/de not_active IP Right Cessation
- 1999-05-03 PL PL99344521A patent/PL344521A1/xx not_active Application Discontinuation
- 1999-05-03 MA MA25565A patent/MA24852A1/fr unknown
- 1999-05-03 CA CA002331297A patent/CA2331297C/en not_active Expired - Fee Related
- 1999-05-03 EA EA200001029A patent/EA003305B1/ru not_active IP Right Cessation
- 1999-05-03 NZ NZ507452A patent/NZ507452A/xx unknown
- 1999-05-03 IL IL13916599A patent/IL139165A0/xx unknown
- 1999-05-03 AR ARP990102059A patent/AR016251A1/es not_active Application Discontinuation
- 1999-05-03 HU HU0102066A patent/HUP0102066A3/hu unknown
- 1999-05-03 ES ES99914722T patent/ES2209419T3/es not_active Expired - Lifetime
- 1999-05-03 AT AT03020745T patent/ATE317448T1/de not_active IP Right Cessation
- 1999-05-04 AP AP2001002296A patent/AP2001002296A0/xx unknown
- 1999-05-04 PA PA19998471801A patent/PA8471801A1/es unknown
- 1999-05-04 AP APAP/P/1999/001527A patent/AP1266A/en active
-
2000
- 2000-10-24 IS IS5681A patent/IS5681A/is unknown
- 2000-10-27 OA OA1200000299A patent/OA11508A/en unknown
- 2000-11-03 HR HR20000747A patent/HRP20000747A2/hr not_active Application Discontinuation
- 2000-11-03 NO NO20005552A patent/NO20005552L/no not_active Application Discontinuation
- 2000-11-30 BG BG105008A patent/BG105008A/xx unknown
Also Published As
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