TR200003250T2 - Higromisin A türevleri - Google Patents

Higromisin A türevleri

Info

Publication number
TR200003250T2
TR200003250T2 TR2000/03250T TR200003250T TR200003250T2 TR 200003250 T2 TR200003250 T2 TR 200003250T2 TR 2000/03250 T TR2000/03250 T TR 2000/03250T TR 200003250 T TR200003250 T TR 200003250T TR 200003250 T2 TR200003250 T2 TR 200003250T2
Authority
TR
Turkey
Prior art keywords
compounds
formula
infections
hygromycin
derivatives
Prior art date
Application number
TR2000/03250T
Other languages
English (en)
Inventor
Elizabeth Brighty Katherine
Sam Guhan Subramanian
Raymond Jefson Martin
Gerald Ii Linde Robert
Lester Mccormick Ellen
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of TR200003250T2 publication Critical patent/TR200003250T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P19/00—Preparation of compounds containing saccharide radicals
    • C12P19/44—Preparation of O-glycosides, e.g. glucosides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biotechnology (AREA)
  • Veterinary Medicine (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Microbiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)

Abstract

Bulus, formül (1)'e ait bilesiklerle ve bunlarin farmasötik açidan kabul gören tuzlari, ön ilaçlari ve solvatlariyla ilgilidir; buradaki R1 ve R2, burada tanimlandigi gibidir. Formül (1)'e ait bilesikler, çesitli bakteriyel ve protozoal enfeksiyonlarin ve bu enfeksiyonlara bagli bozukluklarin tedavi edilmesi için kullanilabilen antibakteriyel ve antiprotozoal maddelerdir. Bulus, formül (1)'e ait bilesikleri ihtiva eden farmasötik kompozisyonlarla ve bakteriyel ve protozoal enfeksiyonlarin, formül (1)'e ait bilesiklerin uygulanmasi suretiyle tedavi edildigi metotlarla da ilgilidir.
TR2000/03250T 1998-05-04 1999-05-03 Higromisin A türevleri TR200003250T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8404298P 1998-05-04 1998-05-04

Publications (1)

Publication Number Publication Date
TR200003250T2 true TR200003250T2 (tr) 2001-01-22

Family

ID=22182520

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2000/03250T TR200003250T2 (tr) 1998-05-04 1999-05-03 Higromisin A türevleri

Country Status (37)

Country Link
US (1) US6313100B1 (tr)
EP (1) EP1075483B1 (tr)
JP (1) JP2002513796A (tr)
KR (1) KR100402560B1 (tr)
CN (1) CN1299365A (tr)
AP (3) AP0102296A0 (tr)
AR (1) AR016251A1 (tr)
AT (2) ATE255588T1 (tr)
AU (1) AU755806B2 (tr)
BG (1) BG105008A (tr)
BR (1) BR9910206A (tr)
CA (1) CA2331297C (tr)
DE (2) DE69929723D1 (tr)
DK (1) DK1075483T3 (tr)
DZ (1) DZ2780A1 (tr)
EA (2) EA200200779A1 (tr)
ES (1) ES2209419T3 (tr)
GT (1) GT199900064A (tr)
HR (1) HRP20000747A2 (tr)
HU (1) HUP0102066A3 (tr)
ID (1) ID27030A (tr)
IL (1) IL139165A0 (tr)
IS (1) IS5681A (tr)
MA (1) MA24852A1 (tr)
NO (1) NO20005552L (tr)
NZ (1) NZ507452A (tr)
OA (1) OA11508A (tr)
PA (1) PA8471801A1 (tr)
PE (1) PE20000478A1 (tr)
PL (1) PL344521A1 (tr)
PT (1) PT1075483E (tr)
SK (1) SK16452000A3 (tr)
TN (1) TNSN99083A1 (tr)
TR (1) TR200003250T2 (tr)
WO (1) WO1999057125A2 (tr)
YU (1) YU66900A (tr)
ZA (1) ZA993064B (tr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CZ20011904A3 (cs) * 1998-12-02 2001-10-17 Pfizer Products Inc. Deriváty hygromycinu jako antibakteriální činidla
GB9923078D0 (en) * 1999-09-29 1999-12-01 Phytopharm Plc Sapogenin derivatives and their use
US6771019B1 (en) * 1999-05-14 2004-08-03 Ifire Technology, Inc. Electroluminescent laminate with patterned phosphor structure and thick film dielectric with improved dielectric properties
EE200200671A (et) * 2000-06-02 2004-08-16 Pfizer Products Inc. Hügromütsiin A derivaadid bakteriaalsete ja algloomadest põhjustatud infektsioonide ravimiseks
CN102168034B (zh) * 2010-11-29 2012-12-05 中国科学院南海海洋研究所 一种海洋链霉菌以及利用该菌制备替达霉素a和b的方法
JP2016069333A (ja) * 2014-09-30 2016-05-09 公益財団法人微生物化学研究会 新規化合物、その製造方法、及びその用途、並びに、新規微生物
CN104480039B (zh) * 2014-11-25 2017-09-12 辽宁大学 抗生素产生菌及其应用
WO2020041179A1 (en) * 2018-08-20 2020-02-27 Northeastern University Hygromycin a compounds and methods of treating spirochete diseases
TWI771766B (zh) 2019-10-04 2022-07-21 美商輝瑞股份有限公司 二醯基甘油醯基轉移酶２ 抑制劑
JP2022058085A (ja) 2020-02-24 2022-04-11 ファイザー・インク ジアシルグリセロールアシルトランスフェラーゼ２阻害剤とアセチル－ＣｏＡカルボキシラーゼ阻害剤との組合せ

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0213692B1 (en) 1985-06-27 1990-09-26 Takeda Chemical Industries, Ltd. Use of hygromycin and epihygromycin in the treatment of swine dysentery
GB8605245D0 (en) 1986-03-04 1986-04-09 Fujisawa Pharmaceutical Co Prophylactic & therapeutic agent

Also Published As

Publication number Publication date
AP2001002296A0 (en) 2001-12-31
DE69929723D1 (de) 2006-04-20
IS5681A (is) 2000-10-24
KR20010043303A (ko) 2001-05-25
DZ2780A1 (fr) 2005-04-23
AR016251A1 (es) 2001-06-20
HRP20000747A2 (en) 2001-06-30
ATE255588T1 (de) 2003-12-15
ES2209419T3 (es) 2004-06-16
US6313100B1 (en) 2001-11-06
PA8471801A1 (es) 2000-09-29
NO20005552D0 (no) 2000-11-03
JP2002513796A (ja) 2002-05-14
NO20005552L (no) 2001-01-02
PE20000478A1 (es) 2000-05-31
DK1075483T3 (da) 2004-03-15
YU66900A (sh) 2003-12-31
AP0102296A0 (en) 2000-11-04
HUP0102066A3 (en) 2003-07-28
ID27030A (id) 2001-02-22
CA2331297A1 (en) 1999-11-11
AU755806B2 (en) 2002-12-19
CN1299365A (zh) 2001-06-13
AP9901527A0 (en) 1999-06-30
WO1999057125A2 (en) 1999-11-11
NZ507452A (en) 2003-04-29
EP1075483B1 (en) 2003-12-03
ATE317448T1 (de) 2006-02-15
WO1999057125A3 (en) 1999-12-29
TNSN99083A1 (fr) 2005-11-10
KR100402560B1 (ko) 2003-10-17
HUP0102066A2 (hu) 2001-11-28
OA11508A (en) 2004-02-09
BG105008A (en) 2001-09-28
EA200200779A1 (ru) 2002-12-26
MA24852A1 (fr) 1999-12-31
BR9910206A (pt) 2001-01-30
GT199900064A (es) 2000-10-24
EA003305B1 (ru) 2003-04-24
PL344521A1 (en) 2001-11-05
EP1075483A2 (en) 2001-02-14
SK16452000A3 (sk) 2001-09-11
PT1075483E (pt) 2004-03-31
IL139165A0 (en) 2001-11-25
ZA993064B (en) 2000-12-06
AP1266A (en) 2004-03-29
CA2331297C (en) 2004-12-28
EA200001029A1 (ru) 2001-04-23
DE69913333T2 (de) 2004-10-07
AU3341999A (en) 1999-11-23
DE69913333D1 (de) 2004-01-15

Similar Documents

Publication Publication Date Title
EA200100623A1 (ru) Кетолидные антибиотики
PA8486401A1 (es) Antibioticos cetolidos carbamato y carbazato
AP2001002131A0 (en) Novel macrolide antibiotics.
PT1132392E (pt) Antibioticos cetolidos
TR200003250T2 (tr) Higromisin A türevleri
TR200003249T2 (tr) 2''-Deoksi higromisin türevleri
PT1167376E (pt) Antibioticos macrolidos
AP2001002154A0 (en) Hygromycin a derivatives (changed by the ISA to read hygromycin a derivatives as antibacterial agents.
MXPA02011966A (es) Derivados de higromicina a para el el tratamiento de infecciones bacterianas y por protozoarios.
TR200201143T2 (tr) Higromisin a ön-ilaçları.
ECSP992931A (es) Derivados de 2'' desoxi higromicina
ECSP992943A (es) Derivados de higromicina a
ECSP993239A (es) Derivados de higromicina