TR200400630T4 - Ketolit antibiyotikleri - Google Patents

Ketolit antibiyotikleri

Info

Publication number
TR200400630T4
TR200400630T4 TR2004/00630T TR200400630T TR200400630T4 TR 200400630 T4 TR200400630 T4 TR 200400630T4 TR 2004/00630 T TR2004/00630 T TR 2004/00630T TR 200400630 T TR200400630 T TR 200400630T TR 200400630 T4 TR200400630 T4 TR 200400630T4
Authority
TR
Turkey
Prior art keywords
compounds
formula
ketolite
antibiotics
infections
Prior art date
Application number
TR2004/00630T
Other languages
English (en)
Inventor
Kaneko Takushi
Thomas Mcmillen William
Su Wei-Guo
Zhao Hongjuan
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of TR200400630T4 publication Critical patent/TR200400630T4/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Fats And Perfumes (AREA)
  • Cephalosporin Compounds (AREA)

Abstract

Bu bulus, formül 1 bilesikleri Formül (I) ve bunlarin farmasötik açidan kabul gören tuzlari, ön ilaçlari ve solvatlari ile ilgilidir; buradaki X1,R1,R2,R8,R9 ve R10, burada tanimlandigi gibidir. Formül 1 bilesikleri, çesitli bakteriyel ve protozoal enfeksiyonlarin ve bu enfeksiyonlar ile baglantili bozukluklarin tedavisinde kullanilabilen antibakteriyel ve antiprotozoal maddelerdir. Bulus, formül 1 bilesikleri içeren farmasötik kompozisyonlarla ve formül 1 bilesiklerinin uygulanmasi suretiyle bakteriyel ve protozoal enfeksiyonlarin tedavi edildigi metotlarla da ilgilidir.
TR2004/00630T 2000-03-06 2001-03-05 Ketolit antibiyotikleri TR200400630T4 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US18697000P 2000-03-06 2000-03-06

Publications (1)

Publication Number Publication Date
TR200400630T4 true TR200400630T4 (tr) 2004-05-21

Family

ID=22687057

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2004/00630T TR200400630T4 (tr) 2000-03-06 2001-03-05 Ketolit antibiyotikleri

Country Status (11)

Country Link
US (1) US6555524B2 (tr)
EP (1) EP1132392B1 (tr)
JP (1) JP2001261694A (tr)
AT (1) ATE260928T1 (tr)
BR (1) BR0100850A (tr)
CA (1) CA2339051A1 (tr)
DE (1) DE60102171T2 (tr)
DK (1) DK1132392T3 (tr)
ES (1) ES2214385T3 (tr)
PT (1) PT1132392E (tr)
TR (1) TR200400630T4 (tr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5413293A (en) * 1992-12-22 1995-05-09 Hughes Aircraft Company Magnetic torque attitude control systems
US6555581B1 (en) 2001-02-15 2003-04-29 Jones Pharma, Inc. Levothyroxine compositions and methods
US6995143B2 (en) * 2002-02-28 2006-02-07 Basilea Pharmaceutica Ag Macrolides with antibacterial activity
US7091196B2 (en) 2002-09-26 2006-08-15 Rib-X Pharmaceuticals, Inc. Bifunctional heterocyclic compounds and methods of making and using same
EP1638549A4 (en) 2003-03-10 2011-06-15 Optimer Pharmaceuticals Inc NEW ANTIBACTERIAL AGENTS
EP1723159B1 (en) 2004-02-27 2019-06-12 Melinta Therapeutics, Inc. Macrocyclic compounds and methods of making and using the same
AU2005317735B2 (en) 2004-12-21 2009-06-04 Pfizer Products Inc. Macrolides
US7387972B2 (en) * 2006-03-01 2008-06-17 Promos Technologies Pte. Ltd. Reducing nitrogen concentration with in-situ steam generation
EP2214484A4 (en) * 2007-10-25 2013-01-02 Cempra Pharmaceuticals Inc PROCESS FOR PREPARING ANTIBACTERIAL MAKROLIDE AGENTS
US8796232B2 (en) * 2008-10-24 2014-08-05 Cempra Pharmaceuticals, Inc. Methods for treating resistant diseases using triazole containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
AU2010292010B2 (en) * 2009-09-10 2016-01-07 Cempra Pharmaceuticals, Inc. Methods for treating malaria, tuberculosis and MAC diseases
CN103080122A (zh) 2010-03-22 2013-05-01 森普拉制药公司 大环内脂的结晶形式及其用途
US9051346B2 (en) 2010-05-20 2015-06-09 Cempra Pharmaceuticals, Inc. Process for preparing triazole-containing ketolide antibiotics
JP6042334B2 (ja) 2010-09-10 2016-12-14 センプラ ファーマシューティカルズ，インコーポレイテッド 疾患治療のための水素結合形成フルオロケトライド
CN104470527B (zh) 2012-03-27 2019-05-28 森普拉制药公司 用于施用大环内酯抗生素的肠胃外制剂
WO2014152326A1 (en) 2013-03-14 2014-09-25 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
US9751908B2 (en) 2013-03-15 2017-09-05 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of the history of erythromycin
FR2742757B1 (fr) * 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
CO4990960A1 (es) 1997-10-29 2000-12-26 Abbott Lab Derivados de cetolidos 2-halo-6-o sustituidos
FR2777282B1 (fr) 1998-04-08 2001-04-20 Hoechst Marion Roussel Inc Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments

Also Published As

Publication number Publication date
US20020065235A1 (en) 2002-05-30
ES2214385T3 (es) 2004-09-16
DE60102171D1 (de) 2004-04-08
BR0100850A (pt) 2001-11-27
EP1132392B1 (en) 2004-03-03
DK1132392T3 (da) 2004-06-07
ATE260928T1 (de) 2004-03-15
CA2339051A1 (en) 2001-09-06
EP1132392A1 (en) 2001-09-12
JP2001261694A (ja) 2001-09-26
DE60102171T2 (de) 2005-03-03
US6555524B2 (en) 2003-04-29
PT1132392E (pt) 2004-06-30

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