ATE260928T1 - Ketolidantibiotika - Google Patents

Ketolidantibiotika

Info

Publication number
ATE260928T1
ATE260928T1 AT01301966T AT01301966T ATE260928T1 AT E260928 T1 ATE260928 T1 AT E260928T1 AT 01301966 T AT01301966 T AT 01301966T AT 01301966 T AT01301966 T AT 01301966T AT E260928 T1 ATE260928 T1 AT E260928T1
Authority
AT
Austria
Prior art keywords
compounds
formula
infections
relates
ketolide antibiotics
Prior art date
Application number
AT01301966T
Other languages
English (en)
Inventor
Takushi Kaneko
William Thomas Mcmillen
Wei-Guo Su
Hongjuan Zhao
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of ATE260928T1 publication Critical patent/ATE260928T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Public Health (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Fats And Perfumes (AREA)
AT01301966T 2000-03-06 2001-03-05 Ketolidantibiotika ATE260928T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US18697000P 2000-03-06 2000-03-06

Publications (1)

Publication Number Publication Date
ATE260928T1 true ATE260928T1 (de) 2004-03-15

Family

ID=22687057

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01301966T ATE260928T1 (de) 2000-03-06 2001-03-05 Ketolidantibiotika

Country Status (11)

Country Link
US (1) US6555524B2 (de)
EP (1) EP1132392B1 (de)
JP (1) JP2001261694A (de)
AT (1) ATE260928T1 (de)
BR (1) BR0100850A (de)
CA (1) CA2339051A1 (de)
DE (1) DE60102171T2 (de)
DK (1) DK1132392T3 (de)
ES (1) ES2214385T3 (de)
PT (1) PT1132392E (de)
TR (1) TR200400630T4 (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5413293A (en) * 1992-12-22 1995-05-09 Hughes Aircraft Company Magnetic torque attitude control systems
US6555581B1 (en) 2001-02-15 2003-04-29 Jones Pharma, Inc. Levothyroxine compositions and methods
US6995143B2 (en) * 2002-02-28 2006-02-07 Basilea Pharmaceutica Ag Macrolides with antibacterial activity
AR043050A1 (es) 2002-09-26 2005-07-13 Rib X Pharmaceuticals Inc Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos
WO2004080391A2 (en) 2003-03-10 2004-09-23 Optimer Pharmaceuticals, Inc. Novel antibacterial agents
JP5383037B2 (ja) 2004-02-27 2014-01-08 リブ−エックス ファーマシューティカルズ,インコーポレイテッド 大環状化合物およびそれらを製造し使用する方法
GEP20094834B (en) 2004-12-21 2009-11-25 Pfizer Prod Inc Macrolides, pharmaceutical compositions containing them and their use for treatment of bacterial infections
US7387972B2 (en) * 2006-03-01 2008-06-17 Promos Technologies Pte. Ltd. Reducing nitrogen concentration with in-situ steam generation
AU2008316830B2 (en) * 2007-10-25 2016-03-17 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
WO2010048600A1 (en) * 2008-10-24 2010-04-29 Cempra Pharmaceuticals, Inc. Methods for treating resistant diseases using triazole containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
ES2608285T3 (es) 2009-09-10 2017-04-07 Cempra Pharmaceuticals, Inc. Procedimientos para el tratamiento de paludismo, tuberculosis y enfermedades por MAC
RU2650883C2 (ru) 2010-03-22 2018-04-18 Семпра Фармасьютикалз, Инк. Кристаллические формы макролида и их применение
PL2571506T3 (pl) 2010-05-20 2017-10-31 Cempra Pharmaceuticals Inc Sposoby sporządzania makrolidów i ketolidów oraz ich produktów pośrednich
KR20180110181A (ko) 2010-09-10 2018-10-08 셈프라 파마슈티컬스, 인크. 질환을 치료하기 위한 수소결합 형성 플루오로 케토라이드
MX2014011537A (es) 2012-03-27 2015-02-10 Cempra Pharmaceuticals Inc Formulaciones parenterales para la administracion de antibioticos macrolidos.
EP2968801B1 (de) 2013-03-14 2018-09-26 Cempra Pharmaceuticals, Inc. Verfahren zur behandlung von atemwegserkrankungen und formulierungen dafür
AU2014233240B2 (en) 2013-03-15 2018-08-09 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of the history of erythromycin
FR2742757B1 (fr) 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
CO4990960A1 (es) 1997-10-29 2000-12-26 Abbott Lab Derivados de cetolidos 2-halo-6-o sustituidos
FR2777282B1 (fr) 1998-04-08 2001-04-20 Hoechst Marion Roussel Inc Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments

Also Published As

Publication number Publication date
DK1132392T3 (da) 2004-06-07
EP1132392B1 (de) 2004-03-03
DE60102171D1 (de) 2004-04-08
US6555524B2 (en) 2003-04-29
JP2001261694A (ja) 2001-09-26
BR0100850A (pt) 2001-11-27
US20020065235A1 (en) 2002-05-30
EP1132392A1 (de) 2001-09-12
DE60102171T2 (de) 2005-03-03
ES2214385T3 (es) 2004-09-16
TR200400630T4 (tr) 2004-05-21
PT1132392E (pt) 2004-06-30
CA2339051A1 (en) 2001-09-06

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