ATE260928T1 - Ketolidantibiotika - Google Patents
KetolidantibiotikaInfo
- Publication number
- ATE260928T1 ATE260928T1 AT01301966T AT01301966T ATE260928T1 AT E260928 T1 ATE260928 T1 AT E260928T1 AT 01301966 T AT01301966 T AT 01301966T AT 01301966 T AT01301966 T AT 01301966T AT E260928 T1 ATE260928 T1 AT E260928T1
- Authority
- AT
- Austria
- Prior art keywords
- compounds
- formula
- infections
- relates
- ketolide antibiotics
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Public Health (AREA)
- Biochemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Fats And Perfumes (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US18697000P | 2000-03-06 | 2000-03-06 |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE260928T1 true ATE260928T1 (de) | 2004-03-15 |
Family
ID=22687057
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT01301966T ATE260928T1 (de) | 2000-03-06 | 2001-03-05 | Ketolidantibiotika |
Country Status (11)
Country | Link |
---|---|
US (1) | US6555524B2 (de) |
EP (1) | EP1132392B1 (de) |
JP (1) | JP2001261694A (de) |
AT (1) | ATE260928T1 (de) |
BR (1) | BR0100850A (de) |
CA (1) | CA2339051A1 (de) |
DE (1) | DE60102171T2 (de) |
DK (1) | DK1132392T3 (de) |
ES (1) | ES2214385T3 (de) |
PT (1) | PT1132392E (de) |
TR (1) | TR200400630T4 (de) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5413293A (en) * | 1992-12-22 | 1995-05-09 | Hughes Aircraft Company | Magnetic torque attitude control systems |
US6555581B1 (en) | 2001-02-15 | 2003-04-29 | Jones Pharma, Inc. | Levothyroxine compositions and methods |
US6995143B2 (en) * | 2002-02-28 | 2006-02-07 | Basilea Pharmaceutica Ag | Macrolides with antibacterial activity |
AR043050A1 (es) | 2002-09-26 | 2005-07-13 | Rib X Pharmaceuticals Inc | Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos |
WO2004080391A2 (en) | 2003-03-10 | 2004-09-23 | Optimer Pharmaceuticals, Inc. | Novel antibacterial agents |
JP5383037B2 (ja) | 2004-02-27 | 2014-01-08 | リブ−エックス ファーマシューティカルズ,インコーポレイテッド | 大環状化合物およびそれらを製造し使用する方法 |
GEP20094834B (en) | 2004-12-21 | 2009-11-25 | Pfizer Prod Inc | Macrolides, pharmaceutical compositions containing them and their use for treatment of bacterial infections |
US7387972B2 (en) * | 2006-03-01 | 2008-06-17 | Promos Technologies Pte. Ltd. | Reducing nitrogen concentration with in-situ steam generation |
AU2008316830B2 (en) * | 2007-10-25 | 2016-03-17 | Cempra Pharmaceuticals, Inc. | Process for the preparation of macrolide antibacterial agents |
WO2010048600A1 (en) * | 2008-10-24 | 2010-04-29 | Cempra Pharmaceuticals, Inc. | Methods for treating resistant diseases using triazole containing macrolides |
US9937194B1 (en) | 2009-06-12 | 2018-04-10 | Cempra Pharmaceuticals, Inc. | Compounds and methods for treating inflammatory diseases |
ES2608285T3 (es) | 2009-09-10 | 2017-04-07 | Cempra Pharmaceuticals, Inc. | Procedimientos para el tratamiento de paludismo, tuberculosis y enfermedades por MAC |
RU2650883C2 (ru) | 2010-03-22 | 2018-04-18 | Семпра Фармасьютикалз, Инк. | Кристаллические формы макролида и их применение |
PL2571506T3 (pl) | 2010-05-20 | 2017-10-31 | Cempra Pharmaceuticals Inc | Sposoby sporządzania makrolidów i ketolidów oraz ich produktów pośrednich |
KR20180110181A (ko) | 2010-09-10 | 2018-10-08 | 셈프라 파마슈티컬스, 인크. | 질환을 치료하기 위한 수소결합 형성 플루오로 케토라이드 |
MX2014011537A (es) | 2012-03-27 | 2015-02-10 | Cempra Pharmaceuticals Inc | Formulaciones parenterales para la administracion de antibioticos macrolidos. |
EP2968801B1 (de) | 2013-03-14 | 2018-09-26 | Cempra Pharmaceuticals, Inc. | Verfahren zur behandlung von atemwegserkrankungen und formulierungen dafür |
AU2014233240B2 (en) | 2013-03-15 | 2018-08-09 | Cempra Pharmaceuticals, Inc. | Convergent processes for preparing macrolide antibacterial agents |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL114589A (en) * | 1990-11-21 | 1999-12-22 | Roussel Uclaf | Intermediates for the preparation of the history of erythromycin |
FR2742757B1 (fr) | 1995-12-22 | 1998-01-30 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
CO4990960A1 (es) | 1997-10-29 | 2000-12-26 | Abbott Lab | Derivados de cetolidos 2-halo-6-o sustituidos |
FR2777282B1 (fr) | 1998-04-08 | 2001-04-20 | Hoechst Marion Roussel Inc | Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments |
-
2001
- 2001-02-22 JP JP2001046374A patent/JP2001261694A/ja active Pending
- 2001-02-26 US US09/792,937 patent/US6555524B2/en not_active Expired - Fee Related
- 2001-03-02 CA CA002339051A patent/CA2339051A1/en not_active Abandoned
- 2001-03-05 PT PT01301966T patent/PT1132392E/pt unknown
- 2001-03-05 EP EP01301966A patent/EP1132392B1/de not_active Expired - Lifetime
- 2001-03-05 ES ES01301966T patent/ES2214385T3/es not_active Expired - Lifetime
- 2001-03-05 TR TR2004/00630T patent/TR200400630T4/xx unknown
- 2001-03-05 DE DE60102171T patent/DE60102171T2/de not_active Expired - Fee Related
- 2001-03-05 AT AT01301966T patent/ATE260928T1/de not_active IP Right Cessation
- 2001-03-05 DK DK01301966T patent/DK1132392T3/da active
- 2001-03-06 BR BR0100850-1A patent/BR0100850A/pt not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
DK1132392T3 (da) | 2004-06-07 |
EP1132392B1 (de) | 2004-03-03 |
DE60102171D1 (de) | 2004-04-08 |
US6555524B2 (en) | 2003-04-29 |
JP2001261694A (ja) | 2001-09-26 |
BR0100850A (pt) | 2001-11-27 |
US20020065235A1 (en) | 2002-05-30 |
EP1132392A1 (de) | 2001-09-12 |
DE60102171T2 (de) | 2005-03-03 |
ES2214385T3 (es) | 2004-09-16 |
TR200400630T4 (tr) | 2004-05-21 |
PT1132392E (pt) | 2004-06-30 |
CA2339051A1 (en) | 2001-09-06 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
UEP | Publication of translation of european patent specification |
Ref document number: 1132392 Country of ref document: EP |
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REN | Ceased due to non-payment of the annual fee |