DK433787D0 - 1-phenylquinazolin-1h,3h-2,4-dioner og 1-phenylpyrido oe2,3-daapyrimidin-1h,3h-dioner, estere og syreadditionssalte deraf samt farmaceutiske midler indeholdende saadanne forbindelser - Google Patents

1-phenylquinazolin-1h,3h-2,4-dioner og 1-phenylpyrido oe2,3-daapyrimidin-1h,3h-dioner, estere og syreadditionssalte deraf samt farmaceutiske midler indeholdende saadanne forbindelser

Info

Publication number
DK433787D0
DK433787D0 DK433787A DK433787A DK433787D0 DK 433787 D0 DK433787 D0 DK 433787D0 DK 433787 A DK433787 A DK 433787A DK 433787 A DK433787 A DK 433787A DK 433787 D0 DK433787 D0 DK 433787D0
Authority
DK
Denmark
Prior art keywords
dione
daapyrimidine
phenylpyrido
phenylquinazoline
esters
Prior art date
Application number
DK433787A
Other languages
English (en)
Other versions
DK433787A (da
Inventor
Iii John Adams Lowe
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK433787D0 publication Critical patent/DK433787D0/da
Publication of DK433787A publication Critical patent/DK433787A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • C07D239/96Two oxygen atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines Containing Plant Substances (AREA)
DK433787A 1986-08-21 1987-08-20 1-phenylquinazolin-1h,3h-2,4-dioner og 1-phenylpyrido oe2,3-daapyrimidin-1h,3h-dioner, estere og syreadditionssalte deraf samt farmaceutiske midler indeholdende saadanne forbindelser DK433787A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US1986/001718 WO1988001270A1 (en) 1986-08-21 1986-08-21 Pyridopyrimidinediones

Publications (2)

Publication Number Publication Date
DK433787D0 true DK433787D0 (da) 1987-08-20
DK433787A DK433787A (da) 1988-02-22

Family

ID=22195608

Family Applications (1)

Application Number Title Priority Date Filing Date
DK433787A DK433787A (da) 1986-08-21 1987-08-20 1-phenylquinazolin-1h,3h-2,4-dioner og 1-phenylpyrido oe2,3-daapyrimidin-1h,3h-dioner, estere og syreadditionssalte deraf samt farmaceutiske midler indeholdende saadanne forbindelser

Country Status (25)

Country Link
US (1) US4797403A (da)
JP (1) JPH0625166B2 (da)
KR (1) KR900003497B1 (da)
CN (1) CN1014992B (da)
AR (1) AR243513A1 (da)
AT (1) AT388378B (da)
AU (1) AU579047B2 (da)
CA (1) CA1294618C (da)
CS (1) CS268189B2 (da)
DD (1) DD261598A5 (da)
DK (1) DK433787A (da)
EG (1) EG18270A (da)
FI (1) FI84720C (da)
HU (1) HU196798B (da)
IE (1) IE59937B1 (da)
IL (1) IL83569A (da)
MX (1) MX7829A (da)
MY (1) MY101821A (da)
NO (1) NO165493C (da)
NZ (1) NZ221502A (da)
PH (1) PH23853A (da)
PT (1) PT85555B (da)
RU (1) RU1769758C (da)
WO (1) WO1988001270A1 (da)
ZA (1) ZA876172B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0260817B1 (en) * 1986-08-21 1991-05-15 Pfizer Inc. Quinazolinediones and pyridopyrimidinediones
US5290780A (en) * 1991-01-30 1994-03-01 American Cyanamid Co. Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
NZ322197A (en) * 1995-11-21 1999-02-25 Yamanouchi Pharma Co Ltd Pyrido[2,3-d] pyrimidine derivatives and pharmaceutical compositions thereof
GB0507298D0 (en) * 2005-04-11 2005-05-18 Novartis Ag Organic compounds
SA08280783B1 (ar) * 2007-01-11 2011-04-24 استرازينيكا ايه بي مشتقات بيريدوبيريميدين كمثبطات pde4
FR2943673B1 (fr) * 2009-03-27 2013-03-29 Sanofi Aventis Applications therapeutiques de derives de quinazolinedione
EP2686305B1 (en) * 2011-03-14 2020-09-16 Impact Therapeutics, Inc. Quinazolinediones and their use
TWI527800B (zh) 2011-04-01 2016-04-01 南京英派藥業有限公司 作為聚(二磷酸腺苷酸-核醣)聚合酶(parp)之抑制劑之1-(芳基甲基)喹唑啉-2,4(1h,3h)-二酮及其應用

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH490801A (de) * 1968-02-27 1970-05-31 Ciba Geigy Schädlingsbekämpfungsmittel und dessen Verwendung
US3794643A (en) * 1971-04-20 1974-02-26 Hisamitsu Pharmaceutical Co Quinazolinedione derivatives
GB1401549A (en) * 1972-07-07 1975-07-16 Hisamitsu Pharmaceutical Co Pyrido-2,3-d-pyrimidine-2,4-1h,3h- diones and methods of preparing them
US3922275A (en) * 1972-11-09 1975-11-25 Hisamitsu Pharmaceutical Co Pyrido{8 2,3-D{9 {0 pyrimidine-2,4(1H,3H)-diones
JPS5069096A (da) * 1973-10-25 1975-06-09
JPS5649917B2 (da) * 1973-12-18 1981-11-25
JPS5849559B2 (ja) * 1974-02-19 1983-11-05 ヒサミツセイヤク カブシキガイシヤ シンキナ ピリドピリミジンジオンユウドウタイノ セイゾウホウ
JPS50116493A (da) * 1974-02-20 1975-09-11
JPS50157393A (da) * 1974-05-24 1975-12-19
JPS5813551B2 (ja) * 1975-03-15 1983-03-14 ヒサミツセイヤク カブシキガイシヤ シンキナピリド ( 4,3−d ) ピリミジンジオンユウドウタイノセイゾウホウ
US4266056A (en) * 1978-04-07 1981-05-05 Zoecon Corporation Phenyl uracils
DK167280B1 (da) * 1985-03-20 1993-10-04 Ciba Geigy Ag 3-aryluracilderivater, fremgangsmaade til fremstilling deraf, ukrudtsbekaempelsesmidler indeholdende disse derivater samt anvendelsen af derivaterne til ukrudtsbekaempelse
GB8524663D0 (en) * 1985-10-07 1985-11-13 Fujisawa Pharmaceutical Co Quinazoline derivatives

Also Published As

Publication number Publication date
IL83569A0 (en) 1988-01-31
HU196798B (en) 1989-01-30
EG18270A (en) 1992-12-30
NZ221502A (en) 1989-11-28
FI84720C (fi) 1992-01-10
NO165493C (no) 1991-02-20
JPS6360974A (ja) 1988-03-17
CN87105791A (zh) 1988-03-09
RU1769758C (en) 1992-10-15
FI873608A0 (fi) 1987-08-20
FI873608A (fi) 1988-02-22
US4797403A (en) 1989-01-10
AU579047B2 (en) 1988-11-10
AT388378B (de) 1989-06-12
PT85555B (pt) 1990-05-31
IL83569A (en) 1991-12-15
ATA263087A (de) 1988-11-15
DD261598A5 (de) 1988-11-02
AU7724787A (en) 1988-03-10
MY101821A (en) 1992-01-31
NO873514L (no) 1988-02-22
CN1014992B (zh) 1991-12-04
NO165493B (no) 1990-11-12
HUT44786A (en) 1988-04-28
KR900003497B1 (ko) 1990-05-21
AR243513A1 (es) 1993-08-31
KR880002868A (ko) 1988-05-12
WO1988001270A1 (en) 1988-02-25
CA1294618C (en) 1992-01-21
IE872239L (en) 1989-01-20
CS268189B2 (en) 1990-03-14
ZA876172B (en) 1989-03-29
DK433787A (da) 1988-02-22
CS597487A2 (en) 1989-05-12
IE59937B1 (en) 1994-05-04
NO873514D0 (no) 1987-08-20
PH23853A (en) 1989-11-23
PT85555A (en) 1987-09-01
FI84720B (fi) 1991-09-30
MX7829A (es) 1993-08-01
JPH0625166B2 (ja) 1994-04-06

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