DK158357C - 9-deoxo-9a-(ethyl eller n-propyl)-9a-aza-9a-homoerythromycin a og farmaceutisk acceptable syreadditionssalte deraf samt farmaceutiske praeparater indeholdende disse forbindelser - Google Patents
9-deoxo-9a-(ethyl eller n-propyl)-9a-aza-9a-homoerythromycin a og farmaceutisk acceptable syreadditionssalte deraf samt farmaceutiske praeparater indeholdende disse forbindelserInfo
- Publication number
- DK158357C DK158357C DK319884A DK319884A DK158357C DK 158357 C DK158357 C DK 158357C DK 319884 A DK319884 A DK 319884A DK 319884 A DK319884 A DK 319884A DK 158357 C DK158357 C DK 158357C
- Authority
- DK
- Denmark
- Prior art keywords
- homoerythromycin
- deoxo
- aza
- propyl
- ethyl
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- QUPDWYMUPZLYJZ-UHFFFAOYSA-N ethyl Chemical class C[CH2] QUPDWYMUPZLYJZ-UHFFFAOYSA-N 0.000 title 1
- 239000000825 pharmaceutical preparation Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/509,538 US4464527A (en) | 1983-06-30 | 1983-06-30 | Antibacterial 9-deoxo-9a-alkyl-9a-aza-9a-homoerythromycin A derivatives and intermediates therefore |
US50953883 | 1983-06-30 |
Publications (4)
Publication Number | Publication Date |
---|---|
DK319884D0 DK319884D0 (da) | 1984-06-29 |
DK319884A DK319884A (da) | 1984-12-31 |
DK158357B DK158357B (da) | 1990-05-07 |
DK158357C true DK158357C (da) | 1990-10-08 |
Family
ID=24027046
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK319884A DK158357C (da) | 1983-06-30 | 1984-06-29 | 9-deoxo-9a-(ethyl eller n-propyl)-9a-aza-9a-homoerythromycin a og farmaceutisk acceptable syreadditionssalte deraf samt farmaceutiske praeparater indeholdende disse forbindelser |
Country Status (7)
Country | Link |
---|---|
US (1) | US4464527A (da) |
EP (1) | EP0132944B1 (da) |
JP (1) | JPS6025998A (da) |
DE (1) | DE3461805D1 (da) |
DK (1) | DK158357C (da) |
GR (1) | GR79536B (da) |
IE (1) | IE57564B1 (da) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MX13723A (es) * | 1987-11-10 | 1993-05-01 | Pfizer | Procedimiento para preparar derivados de 9-desoxo-9a-alil- y propargil-9a-aza-9a-homoeritromicina a |
US5912331A (en) * | 1991-03-15 | 1999-06-15 | Merck & Co., Inc. | Process for the preparation of 9-deoxo-9(Z)-hydroxyiminoerythromycin A |
US5985844A (en) * | 1992-03-26 | 1999-11-16 | Merck & Co., Inc. | Homoerythromycin A derivatives modified at the 4"-and 8A-positions |
US5215980A (en) * | 1992-01-17 | 1993-06-01 | Merck & Co., Inc. | 10-AZA-9-deoxo-11-deoxy-erythromycin A and derivatives thereof |
US5210235A (en) * | 1992-08-26 | 1993-05-11 | Merck & Co., Inc. | Methods of elaborating erythromycin fragments into amine-containing fragments of azalide antibiotics |
AU6082594A (en) * | 1993-01-11 | 1994-08-15 | Merck & Co., Inc. | 8a-aza and 9a-aza macrolide antibiotics, and a process for producing same and methods of use |
US5332807A (en) * | 1993-04-14 | 1994-07-26 | Merck & Co., Inc. | Process of producing 8A- and 9A-azalide antibiotics |
ATE154806T1 (de) * | 1993-05-19 | 1997-07-15 | Pfizer | Zwischenprodukt für azithromycin |
HRP931480B1 (en) * | 1993-12-08 | 1997-08-31 | Sour Pliva | 9a-N-(N'-CARBAMONYL) and 9a-N-(N'-THIOCARBAMONYL) DERIVATES OF 9-DEOXO-9a-HOMOERYTHROMYCIN A |
US6043227A (en) * | 1998-08-19 | 2000-03-28 | Pfizer Inc. | C11 carbamates of macrolide antibacterials |
EP1437360A3 (en) * | 1998-08-19 | 2005-04-06 | Pfizer Products Inc. | C11 Carbamates of macrolide antibacterials |
ATE306491T1 (de) | 2000-08-23 | 2005-10-15 | Wockhardt Ltd | Verfahren zur herstellung von wasserfreiem azithromycin |
ITMI20022292A1 (it) * | 2002-10-29 | 2004-04-30 | Zambon Spa | 9a-azalidi ad attivita' antiinfiammatoria. |
HRP20020885B1 (en) | 2002-11-11 | 2007-05-31 | GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. | SUBSTITUTED 9a-N-{N'-[4-(SULFONYL)PHENYLCARBAMOYL]}DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHROMYCIN A AND 5-O-DESOZAMINYL-9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHRONOLIDE A |
HRP20020991A2 (en) | 2002-12-12 | 2005-02-28 | Pliva-Istra�iva�ki institut d.o.o. | N"-Substituted 9a-N-(N'-carbamoyl-Gamma-aminopropyl), 9a-N-(N'? -thiocarbamoyl-Gamma-aminopropyl), 9a-N-(N'-((Beta-cyanoethyl)-N'-carbamoyl-Gamma? -aminopropyl) and 9a-N-(N'-(Beta-cyanoethyl)-N'-thiocarbamoyl-Gamma? -aminopropyl) derivatives of 9-de |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SI7910768A8 (en) * | 1979-04-02 | 1996-06-30 | Pliva Pharm & Chem Works | Process for pripering 11-aza-4-0-cladinosyl-6-0-desosaminyl-15-ethyl- 7,13,14-trihydroxy-3,5,7,9,12,14-hexamethyl- oxacyclopentadecane-2-one and their derivatives |
SI8110592A8 (en) * | 1981-03-06 | 1996-06-30 | Pliva Pharm & Chem Works | Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof |
US4474768A (en) * | 1982-07-19 | 1984-10-02 | Pfizer Inc. | N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor |
-
1983
- 1983-06-30 US US06/509,538 patent/US4464527A/en not_active Expired - Lifetime
-
1984
- 1984-06-21 DE DE8484304185T patent/DE3461805D1/de not_active Expired
- 1984-06-21 EP EP84304185A patent/EP0132944B1/en not_active Expired
- 1984-06-27 GR GR75138A patent/GR79536B/el unknown
- 1984-06-29 JP JP59133396A patent/JPS6025998A/ja active Pending
- 1984-06-29 IE IE1665/84A patent/IE57564B1/en not_active IP Right Cessation
- 1984-06-29 DK DK319884A patent/DK158357C/da not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
IE57564B1 (en) | 1992-12-16 |
DE3461805D1 (en) | 1987-02-05 |
GR79536B (da) | 1984-10-30 |
IE841665L (en) | 1984-12-30 |
EP0132944A1 (en) | 1985-02-13 |
JPS6025998A (ja) | 1985-02-08 |
EP0132944B1 (en) | 1986-12-30 |
DK158357B (da) | 1990-05-07 |
DK319884A (da) | 1984-12-31 |
US4464527A (en) | 1984-08-07 |
DK319884D0 (da) | 1984-06-29 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PUP | Patent expired |