DK304488A - Borholdige peptider eller fysiologisk acceptable salte deraf og deres anvendelse samt mellemprodukter til dens fremstilling - Google Patents

Borholdige peptider eller fysiologisk acceptable salte deraf og deres anvendelse samt mellemprodukter til dens fremstilling

Info

Publication number
DK304488A
DK304488A DK304488A DK304488A DK304488A DK 304488 A DK304488 A DK 304488A DK 304488 A DK304488 A DK 304488A DK 304488 A DK304488 A DK 304488A DK 304488 A DK304488 A DK 304488A
Authority
DK
Denmark
Prior art keywords
sustainable
intermediates
peptides
manufacturing
acceptable salts
Prior art date
Application number
DK304488A
Other languages
Danish (da)
English (en)
Other versions
DK304488D0 (da
Inventor
Charles Adrian Kettner
Ashokkumar Bhikkappa Shenvi
Original Assignee
Du Pont
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont filed Critical Du Pont
Publication of DK304488D0 publication Critical patent/DK304488D0/da
Publication of DK304488A publication Critical patent/DK304488A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK304488A 1987-06-05 1988-06-03 Borholdige peptider eller fysiologisk acceptable salte deraf og deres anvendelse samt mellemprodukter til dens fremstilling DK304488A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5967087A 1987-06-05 1987-06-05
US07/178,368 US5187157A (en) 1987-06-05 1988-04-06 Peptide boronic acid inhibitors of trypsin-like proteases

Publications (2)

Publication Number Publication Date
DK304488D0 DK304488D0 (da) 1988-06-03
DK304488A true DK304488A (da) 1988-12-06

Family

ID=26739035

Family Applications (1)

Application Number Title Priority Date Filing Date
DK304488A DK304488A (da) 1987-06-05 1988-06-03 Borholdige peptider eller fysiologisk acceptable salte deraf og deres anvendelse samt mellemprodukter til dens fremstilling

Country Status (16)

Country Link
US (1) US5187157A (de)
EP (1) EP0293881B1 (de)
JP (1) JPH0730090B2 (de)
KR (1) KR910003619B1 (de)
AU (1) AU623592B2 (de)
CA (1) CA1328332C (de)
DE (1) DE3878991T2 (de)
DK (1) DK304488A (de)
ES (1) ES2046237T3 (de)
FI (1) FI97297C (de)
HU (1) HU205141B (de)
IE (1) IE64787B1 (de)
IL (1) IL86613A (de)
NO (1) NO882472L (de)
NZ (1) NZ224903A (de)
PT (1) PT87652B (de)

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* Cited by examiner, † Cited by third party
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KR890000514A (ko) 1989-03-15
FI882638A (fi) 1988-12-06
KR910003619B1 (ko) 1991-06-07
PT87652B (pt) 1992-09-30
NO882472D0 (no) 1988-06-03
IE881666L (en) 1988-12-05
US5187157A (en) 1993-02-16
FI97297C (fi) 1996-11-25
JPS6463583A (en) 1989-03-09
IE64787B1 (en) 1995-09-06
DE3878991D1 (de) 1993-04-15
JPH0730090B2 (ja) 1995-04-05
EP0293881A2 (de) 1988-12-07
HU205141B (en) 1992-03-30
FI97297B (fi) 1996-08-15
EP0293881A3 (en) 1990-05-30
DE3878991T2 (de) 1993-07-15
IL86613A (en) 1993-04-04
PT87652A (pt) 1988-07-01
HUT49629A (en) 1989-10-30
IL86613A0 (en) 1988-11-30
NO882472L (no) 1988-12-06
CA1328332C (en) 1994-04-05
DK304488D0 (da) 1988-06-03
AU1733288A (en) 1988-12-08
AU623592B2 (en) 1992-05-21
NZ224903A (en) 1990-02-26
FI882638A0 (fi) 1988-06-03
ES2046237T3 (es) 1994-02-01
EP0293881B1 (de) 1993-03-10

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