FI97297C - Menetelmä terapeuttisesti käyttökelpoisten booriaminohappojohdannaisten valmistamiseksi - Google Patents

Menetelmä terapeuttisesti käyttökelpoisten booriaminohappojohdannaisten valmistamiseksi

Info

Publication number
FI97297C
FI97297C FI882638A FI882638A FI97297C FI 97297 C FI97297 C FI 97297C FI 882638 A FI882638 A FI 882638A FI 882638 A FI882638 A FI 882638A FI 97297 C FI97297 C FI 97297C
Authority
FI
Finland
Prior art keywords
preparation
amino acid
acid derivatives
therapeutically useful
boronic amino
Prior art date
Application number
FI882638A
Other languages
English (en)
Swedish (sv)
Other versions
FI97297B (fi
FI882638A (fi
FI882638A0 (fi
Inventor
Charles Adrian Kettner
Ashokkumar Bhikkappa Shenvi
Original Assignee
Du Pont Merck Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont Merck Pharma filed Critical Du Pont Merck Pharma
Publication of FI882638A0 publication Critical patent/FI882638A0/fi
Publication of FI882638A publication Critical patent/FI882638A/fi
Application granted granted Critical
Publication of FI97297B publication Critical patent/FI97297B/fi
Publication of FI97297C publication Critical patent/FI97297C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
FI882638A 1987-06-05 1988-06-03 Menetelmä terapeuttisesti käyttökelpoisten booriaminohappojohdannaisten valmistamiseksi FI97297C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US5967087A 1987-06-05 1987-06-05
US5967087 1987-06-05
US17836888 1988-04-06
US07/178,368 US5187157A (en) 1987-06-05 1988-04-06 Peptide boronic acid inhibitors of trypsin-like proteases

Publications (4)

Publication Number Publication Date
FI882638A0 FI882638A0 (fi) 1988-06-03
FI882638A FI882638A (fi) 1988-12-06
FI97297B FI97297B (fi) 1996-08-15
FI97297C true FI97297C (fi) 1996-11-25

Family

ID=26739035

Family Applications (1)

Application Number Title Priority Date Filing Date
FI882638A FI97297C (fi) 1987-06-05 1988-06-03 Menetelmä terapeuttisesti käyttökelpoisten booriaminohappojohdannaisten valmistamiseksi

Country Status (16)

Country Link
US (1) US5187157A (fi)
EP (1) EP0293881B1 (fi)
JP (1) JPH0730090B2 (fi)
KR (1) KR910003619B1 (fi)
AU (1) AU623592B2 (fi)
CA (1) CA1328332C (fi)
DE (1) DE3878991T2 (fi)
DK (1) DK304488A (fi)
ES (1) ES2046237T3 (fi)
FI (1) FI97297C (fi)
HU (1) HU205141B (fi)
IE (1) IE64787B1 (fi)
IL (1) IL86613A (fi)
NO (1) NO882472L (fi)
NZ (1) NZ224903A (fi)
PT (1) PT87652B (fi)

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EP0293881B1 (en) 1993-03-10
CA1328332C (en) 1994-04-05
DK304488D0 (da) 1988-06-03
NZ224903A (en) 1990-02-26
AU1733288A (en) 1988-12-08
NO882472L (no) 1988-12-06
IE64787B1 (en) 1995-09-06
FI97297B (fi) 1996-08-15
PT87652B (pt) 1992-09-30
AU623592B2 (en) 1992-05-21
EP0293881A3 (en) 1990-05-30
DE3878991D1 (de) 1993-04-15
DE3878991T2 (de) 1993-07-15
PT87652A (pt) 1988-07-01
US5187157A (en) 1993-02-16
EP0293881A2 (en) 1988-12-07
HU205141B (en) 1992-03-30
KR890000514A (ko) 1989-03-15
IL86613A0 (en) 1988-11-30
FI882638A (fi) 1988-12-06
NO882472D0 (no) 1988-06-03
FI882638A0 (fi) 1988-06-03
HUT49629A (en) 1989-10-30
IL86613A (en) 1993-04-04
JPH0730090B2 (ja) 1995-04-05
ES2046237T3 (es) 1994-02-01
JPS6463583A (en) 1989-03-09
IE881666L (en) 1988-12-05
DK304488A (da) 1988-12-06
KR910003619B1 (ko) 1991-06-07

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