DK2746265T3 - Heterocyclisk derivat som mikrosomal prostaglandin-E-syntase-(mPGEs)-inhibitor - Google Patents
Heterocyclisk derivat som mikrosomal prostaglandin-E-syntase-(mPGEs)-inhibitor Download PDFInfo
- Publication number
- DK2746265T3 DK2746265T3 DK12823510.8T DK12823510T DK2746265T3 DK 2746265 T3 DK2746265 T3 DK 2746265T3 DK 12823510 T DK12823510 T DK 12823510T DK 2746265 T3 DK2746265 T3 DK 2746265T3
- Authority
- DK
- Denmark
- Prior art keywords
- mpges
- synthase
- inhibitor
- heterocyclic derivative
- microsomal prostaglandin
- Prior art date
Links
- 102000004226 Prostaglandin-E Synthases Human genes 0.000 title 1
- 108090000748 Prostaglandin-E Synthases Proteins 0.000 title 1
- 125000000623 heterocyclic group Chemical group 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 230000003228 microsomal effect Effects 0.000 title 1
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- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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AU2015342883B2 (en) | 2014-11-06 | 2020-07-02 | Bial - R&D Investments, S.A. | Substituted pyrrolo(1,2-a)pyrimidines and their use in the treatment of medical disorders |
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2014
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2015
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2016
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