DK2035432T3 - 2-(substitueret amino)-benzothiazolsulfonamid-HIV-proteaseinhibitorer - Google Patents

2-(substitueret amino)-benzothiazolsulfonamid-HIV-proteaseinhibitorer

Info

Publication number
DK2035432T3
DK2035432T3 DK07765554.6T DK07765554T DK2035432T3 DK 2035432 T3 DK2035432 T3 DK 2035432T3 DK 07765554 T DK07765554 T DK 07765554T DK 2035432 T3 DK2035432 T3 DK 2035432T3
Authority
DK
Denmark
Prior art keywords
substituted amino
protease inhibitors
hiv protease
benzothiazole sulfonamide
sulfonamide hiv
Prior art date
Application number
DK07765554.6T
Other languages
Danish (da)
English (en)
Inventor
Kock Herman De
Tim Hugo Maria Jonckers
Paul Jozef Gabriel Maria Boonants
Stefaan Julien Last
Inge Dierynck
Judith Eva Baumeister
T Klooster Gerben Albert Eleutherius Van
Original Assignee
Tibotec Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd
Application granted granted Critical
Publication of DK2035432T3 publication Critical patent/DK2035432T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Virology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK07765554.6T 2006-06-23 2007-06-22 2-(substitueret amino)-benzothiazolsulfonamid-HIV-proteaseinhibitorer DK2035432T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06116003 2006-06-23
PCT/EP2007/056235 WO2007147884A1 (en) 2006-06-23 2007-06-22 2-(substituted-amino)-benzothiazole sulfonamide hiv protease inhibitors

Publications (1)

Publication Number Publication Date
DK2035432T3 true DK2035432T3 (da) 2012-05-14

Family

ID=37596252

Family Applications (1)

Application Number Title Priority Date Filing Date
DK07765554.6T DK2035432T3 (da) 2006-06-23 2007-06-22 2-(substitueret amino)-benzothiazolsulfonamid-HIV-proteaseinhibitorer

Country Status (30)

Country Link
US (1) US8202887B2 (https=)
EP (1) EP2035432B1 (https=)
JP (1) JP5232776B2 (https=)
KR (1) KR101419320B1 (https=)
CN (1) CN101479275B (https=)
AP (1) AP2069A (https=)
AR (1) AR061619A1 (https=)
AT (1) ATE544769T1 (https=)
AU (1) AU2007262943B2 (https=)
BR (1) BRPI0713487B1 (https=)
CA (1) CA2653233C (https=)
CL (1) CL2007001826A1 (https=)
CY (1) CY1112971T1 (https=)
DK (1) DK2035432T3 (https=)
EA (1) EA016387B1 (https=)
ES (1) ES2381129T3 (https=)
IL (1) IL195381A (https=)
JO (1) JO2841B1 (https=)
MX (1) MX2009000160A (https=)
MY (1) MY146805A (https=)
NZ (1) NZ573286A (https=)
PE (1) PE20080342A1 (https=)
PL (1) PL2035432T3 (https=)
PT (1) PT2035432E (https=)
SI (1) SI2035432T1 (https=)
TW (1) TWI415851B (https=)
UA (1) UA96445C2 (https=)
UY (1) UY30416A1 (https=)
WO (1) WO2007147884A1 (https=)
ZA (1) ZA200810350B (https=)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3090B1 (ar) * 2009-12-11 2017-03-15 Janssen Sciences Ireland Uc 5- امينو-4- هيدروكسي-بنتويل اميدات
AP2013006706A0 (en) 2010-07-02 2013-02-28 Gilead Sciences Inc Napht-2-ylacetic acid derivatives to treat AIDS
KR20130124291A (ko) 2010-07-02 2013-11-13 길리애드 사이언시즈, 인코포레이티드 Hiv 항바이러스 화합물로서의 2-퀴놀리닐-아세트산 유도체
US9024038B2 (en) * 2010-12-27 2015-05-05 Purdue Research Foundation Compunds and methods for treating HIV
BR112013027096A2 (pt) * 2011-04-21 2016-12-27 Gilead Sciences Inc compostos de benzotiazol e seu uso farmacêutico
US9284323B2 (en) 2012-01-04 2016-03-15 Gilead Sciences, Inc. Naphthalene acetic acid derivatives against HIV infection
WO2013103724A1 (en) 2012-01-04 2013-07-11 Gilead Sciences, Inc. 2- (tert - butoxy) -2- (7 -methylquinolin- 6 - yl) acetic acid derivatives for treating aids
ES2571479T3 (es) 2012-04-20 2016-05-25 Gilead Sciences Inc Derivados del ácido benzotiazol-6-il acético y su uso para tratar una infección por VIH
US20230218644A1 (en) 2020-04-16 2023-07-13 Som Innovation Biotech, S.A. Compounds for use in the treatment of viral infections by respiratory syndrome-related coronavirus
US12083099B2 (en) 2020-10-28 2024-09-10 Accencio LLC Methods of treating symptoms of coronavirus infection with viral protease inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2275866T3 (es) * 2001-02-14 2007-06-16 Tibotec Pharmaceuticals Ltd. 2-(aminosustituido)-benzotiazol-sulfonamidas de amplio esprecto inhibidoras de la proteasa de vih.
TWI286476B (en) * 2001-12-12 2007-09-11 Tibotec Pharm Ltd Combination of cytochrome P450 dependent protease inhibitors
PL374948A1 (en) * 2002-08-02 2005-11-14 Tibotec Pharmaceuticals Ltd. Broadspectrum 2-amino-benzothiazole sulfonamide hiv protease inhibitors
US20080234288A1 (en) * 2003-09-30 2008-09-25 Kenneth Alan Simmen Hcv Inhibiting Sulfonamides

Also Published As

Publication number Publication date
UY30416A1 (es) 2008-01-31
CN101479275A (zh) 2009-07-08
CY1112971T1 (el) 2016-04-13
JP2009541272A (ja) 2009-11-26
NZ573286A (en) 2011-09-30
EA200970052A1 (ru) 2009-04-28
PT2035432E (pt) 2012-04-24
JP5232776B2 (ja) 2013-07-10
TWI415851B (zh) 2013-11-21
IL195381A (en) 2013-01-31
SI2035432T1 (sl) 2012-06-29
ATE544769T1 (de) 2012-02-15
EA016387B1 (ru) 2012-04-30
KR20090024257A (ko) 2009-03-06
WO2007147884A1 (en) 2007-12-27
ES2381129T3 (es) 2012-05-23
AP2069A (en) 2009-12-08
MY146805A (en) 2012-09-28
AU2007262943A1 (en) 2007-12-27
KR101419320B1 (ko) 2014-07-14
JO2841B1 (en) 2014-09-15
TW200817416A (en) 2008-04-16
HK1125633A1 (en) 2009-08-14
UA96445C2 (ru) 2011-11-10
US20090209583A1 (en) 2009-08-20
PL2035432T3 (pl) 2012-07-31
BRPI0713487B1 (pt) 2022-07-26
CL2007001826A1 (es) 2008-01-18
ZA200810350B (en) 2010-05-26
IL195381A0 (en) 2009-08-03
BRPI0713487A8 (pt) 2018-01-02
EP2035432B1 (en) 2012-02-08
AP2008004679A0 (en) 2008-12-31
MX2009000160A (es) 2009-01-23
CA2653233A1 (en) 2007-12-27
AU2007262943B2 (en) 2012-04-12
CA2653233C (en) 2015-09-29
BRPI0713487A2 (https=) 2012-11-13
PE20080342A1 (es) 2008-04-25
CN101479275B (zh) 2012-03-07
US8202887B2 (en) 2012-06-19
EP2035432A1 (en) 2009-03-18
AR061619A1 (es) 2008-09-10

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