DK170640B1 - Quinolinderivater - Google Patents

Quinolinderivater Download PDF

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Publication number
DK170640B1
DK170640B1 DK207688A DK207688A DK170640B1 DK 170640 B1 DK170640 B1 DK 170640B1 DK 207688 A DK207688 A DK 207688A DK 207688 A DK207688 A DK 207688A DK 170640 B1 DK170640 B1 DK 170640B1
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DK
Denmark
Prior art keywords
alkyl
group
formula
compound
methyl
Prior art date
Application number
DK207688A
Other languages
Danish (da)
English (en)
Other versions
DK207688D0 (da
DK207688A (da
Inventor
Hiraki Ueda
Hisashi Miyamoto
Hiroshi Yamashita
Hitoshi Tone
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of DK207688D0 publication Critical patent/DK207688D0/da
Publication of DK207688A publication Critical patent/DK207688A/da
Application granted granted Critical
Publication of DK170640B1 publication Critical patent/DK170640B1/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/06Peri-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK207688A 1987-04-16 1988-04-15 Quinolinderivater DK170640B1 (da)

Applications Claiming Priority (16)

Application Number Priority Date Filing Date Title
JP9419887 1987-04-16
JP9419887 1987-04-16
JP10235187 1987-04-24
JP10235187 1987-04-24
JP10836187 1987-04-30
JP10836187 1987-04-30
JP12659887 1987-05-22
JP12659887 1987-05-22
JP14954487 1987-06-16
JP14954487 1987-06-16
JP17612687 1987-07-14
JP17612687 1987-07-14
JP28377687 1987-11-09
JP28377687 1987-11-09
JP28710887 1987-11-12
JP28710887 1987-11-12

Publications (3)

Publication Number Publication Date
DK207688D0 DK207688D0 (da) 1988-04-15
DK207688A DK207688A (da) 1988-10-17
DK170640B1 true DK170640B1 (da) 1995-11-20

Family

ID=27572879

Family Applications (2)

Application Number Title Priority Date Filing Date
DK207688A DK170640B1 (da) 1987-04-16 1988-04-15 Quinolinderivater
DK101492A DK171820B1 (da) 1987-04-16 1992-08-13 Quinolinderivater

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK101492A DK171820B1 (da) 1987-04-16 1992-08-13 Quinolinderivater

Country Status (13)

Country Link
US (5) US5591744A (fr)
EP (3) EP0287951B1 (fr)
JP (2) JPH0696557B2 (fr)
KR (2) KR940002113B1 (fr)
CN (1) CN1053666C (fr)
CY (1) CY2050B1 (fr)
DE (4) DE19775083I2 (fr)
DK (2) DK170640B1 (fr)
ES (3) ES2091180T3 (fr)
HK (1) HK128797A (fr)
NL (1) NL980011I2 (fr)
SA (1) SA97180461A (fr)
SG (3) SG97777A1 (fr)

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DE4408212A1 (de) * 1994-03-11 1995-09-14 Bayer Ag 5-Vinyl- und 5-Ethinyl-chinolon- und -naphthyridon-carbonsäuren
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US6509327B1 (en) 1998-09-30 2003-01-21 Alcon Manufacturing, Ltd. Compositions and methods for treating otic, ophthalmic and nasal infections
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DE19850788A1 (de) * 1998-11-04 2000-05-11 Clariant Gmbh Verfahren zur Herstellung von Trifluorbenzoesäuren
EP2275141A1 (fr) 1999-03-17 2011-01-19 Daiichi Pharmaceutical Co., Ltd. Compositions pharmaceutiques au gout camoufle
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JP2005521712A (ja) * 2002-03-26 2005-07-21 アリゾナ ボード オブ リージェンツ オン ビハーフ オブ ザ ユニバーシティー オブ アリゾナ 弱塩基の可溶化
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WO2005023805A1 (fr) 2003-09-04 2005-03-17 Wockhardt Limited Arginine tetrahydrate d'acide benzoquinolizine-2-carboxylique
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CN101437801B (zh) 2006-03-06 2013-02-06 日本烟草产业株式会社 制备4-氧代喹啉化合物的方法
KR101438036B1 (ko) 2006-09-29 2014-09-04 씨아이피엘에이 엘티디. 테모졸로미드 및 유사체의 개선된 제조방법
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CN106913569B (zh) * 2016-01-04 2022-04-22 广东工业大学 苯酞类化合物在制备抗耐药菌药物中的应用
CN112266326A (zh) * 2020-11-10 2021-01-26 杭州臻挚生物科技有限公司 二氯甲苯硝化物中间体的制备方法

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Also Published As

Publication number Publication date
NL980011I2 (nl) 1998-10-01
US5811576A (en) 1998-09-22
DK171820B1 (da) 1997-06-23
EP0823413B1 (fr) 2002-02-13
DE3856434T2 (de) 2001-06-13
EP0287951B1 (fr) 1996-07-03
US5723648A (en) 1998-03-03
DE3856515D1 (de) 2002-03-21
CN1053666C (zh) 2000-06-21
JPH07138232A (ja) 1995-05-30
DE3855388D1 (de) 1996-08-08
ES2172734T3 (es) 2002-10-01
HK128797A (en) 1997-09-19
ES2091180T3 (es) 1996-11-01
DK207688D0 (da) 1988-04-15
EP0823413A2 (fr) 1998-02-11
EP0565132A3 (en) 1994-05-18
DE3856515T2 (de) 2002-08-14
SG101541A1 (en) 2004-01-30
CN1030237A (zh) 1989-01-11
KR960006145B1 (ko) 1996-05-09
DK207688A (da) 1988-10-17
SA97180461A (ar) 2005-12-03
SG49836A1 (en) 1998-06-15
US5495020A (en) 1996-02-27
DE19775083I2 (de) 2001-06-13
KR940002113B1 (ko) 1994-03-17
ES2152936T3 (es) 2001-02-16
DK101492A (da) 1992-08-13
CY2050B1 (en) 1998-04-30
EP0565132A2 (fr) 1993-10-13
NL980011I1 (nl) 1998-05-06
JPH01230558A (ja) 1989-09-14
SG97777A1 (en) 2003-08-20
EP0287951A3 (en) 1990-06-13
DK101492D0 (da) 1992-08-13
US5591744A (en) 1997-01-07
DE3856434D1 (de) 2000-11-30
US5563138A (en) 1996-10-08
KR880012506A (ko) 1988-11-28
EP0565132B1 (fr) 2000-10-25
JP2654537B2 (ja) 1997-09-17
EP0287951A2 (fr) 1988-10-26
EP0823413A3 (fr) 1998-12-09
JPH0696557B2 (ja) 1994-11-30
DE3855388T2 (de) 1997-02-13

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