CY2050B1 - 7-Piperazinyl-or 7-morpholino-4-oxo-quinoline-3-carboxylic acid derivatives their preparation and their use as antimicrobial agents - Google Patents

7-Piperazinyl-or 7-morpholino-4-oxo-quinoline-3-carboxylic acid derivatives their preparation and their use as antimicrobial agents

Info

Publication number
CY2050B1
CY2050B1 CY9802050A CY9802050A CY2050B1 CY 2050 B1 CY2050 B1 CY 2050B1 CY 9802050 A CY9802050 A CY 9802050A CY 9802050 A CY9802050 A CY 9802050A CY 2050 B1 CY2050 B1 CY 2050B1
Authority
CY
Cyprus
Prior art keywords
piperazinyl
morpholino
quinoline
oxo
preparation
Prior art date
Application number
CY9802050A
Other languages
English (en)
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of CY2050B1 publication Critical patent/CY2050B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CY9802050A 1987-04-16 1998-04-30 7-Piperazinyl-or 7-morpholino-4-oxo-quinoline-3-carboxylic acid derivatives their preparation and their use as antimicrobial agents CY2050B1 (en)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
JP9419887 1987-04-16
JP10235187 1987-04-24
JP10836187 1987-04-30
JP12659887 1987-05-22
JP14954487 1987-06-16
JP17612687 1987-07-14
JP28377687 1987-11-09
JP28710887 1987-11-12

Publications (1)

Publication Number Publication Date
CY2050B1 true CY2050B1 (en) 1998-04-30

Family

ID=27572879

Family Applications (1)

Application Number Title Priority Date Filing Date
CY9802050A CY2050B1 (en) 1987-04-16 1998-04-30 7-Piperazinyl-or 7-morpholino-4-oxo-quinoline-3-carboxylic acid derivatives their preparation and their use as antimicrobial agents

Country Status (13)

Country Link
US (5) US5563138A (fr)
EP (3) EP0287951B1 (fr)
JP (2) JPH0696557B2 (fr)
KR (2) KR940002113B1 (fr)
CN (1) CN1053666C (fr)
CY (1) CY2050B1 (fr)
DE (4) DE3855388T2 (fr)
DK (2) DK170640B1 (fr)
ES (3) ES2172734T3 (fr)
HK (1) HK128797A (fr)
NL (1) NL980011I2 (fr)
SA (1) SA97180461A (fr)
SG (3) SG101541A1 (fr)

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Also Published As

Publication number Publication date
KR940002113B1 (ko) 1994-03-17
US5811576A (en) 1998-09-22
US5591744A (en) 1997-01-07
EP0823413A2 (fr) 1998-02-11
DE3856434T2 (de) 2001-06-13
SG101541A1 (en) 2004-01-30
SA97180461A (ar) 2005-12-03
DE3856515T2 (de) 2002-08-14
DE3855388T2 (de) 1997-02-13
US5495020A (en) 1996-02-27
DK101492A (da) 1992-08-13
EP0287951A2 (fr) 1988-10-26
EP0287951B1 (fr) 1996-07-03
ES2091180T3 (es) 1996-11-01
EP0287951A3 (en) 1990-06-13
DE3855388D1 (de) 1996-08-08
DK207688A (da) 1988-10-17
EP0565132A2 (fr) 1993-10-13
DK171820B1 (da) 1997-06-23
CN1053666C (zh) 2000-06-21
HK128797A (en) 1997-09-19
ES2172734T3 (es) 2002-10-01
DE3856515D1 (de) 2002-03-21
JPH07138232A (ja) 1995-05-30
EP0565132A3 (en) 1994-05-18
JPH0696557B2 (ja) 1994-11-30
JP2654537B2 (ja) 1997-09-17
KR880012506A (ko) 1988-11-28
EP0565132B1 (fr) 2000-10-25
DE3856434D1 (de) 2000-11-30
EP0823413B1 (fr) 2002-02-13
DK170640B1 (da) 1995-11-20
CN1030237A (zh) 1989-01-11
KR960006145B1 (ko) 1996-05-09
US5563138A (en) 1996-10-08
DK101492D0 (da) 1992-08-13
ES2152936T3 (es) 2001-02-16
EP0823413A3 (fr) 1998-12-09
SG49836A1 (en) 1998-06-15
NL980011I2 (nl) 1998-10-01
DK207688D0 (da) 1988-04-15
NL980011I1 (nl) 1998-05-06
DE19775083I2 (de) 2001-06-13
US5723648A (en) 1998-03-03
JPH01230558A (ja) 1989-09-14
SG97777A1 (en) 2003-08-20

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