DK1477472T3 - Substituerede phenylalkansyrederivater og anvendelse deraf - Google Patents

Substituerede phenylalkansyrederivater og anvendelse deraf

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Publication number
DK1477472T3
DK1477472T3 DK03706983T DK03706983T DK1477472T3 DK 1477472 T3 DK1477472 T3 DK 1477472T3 DK 03706983 T DK03706983 T DK 03706983T DK 03706983 T DK03706983 T DK 03706983T DK 1477472 T3 DK1477472 T3 DK 1477472T3
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group
carbon atoms
alkyl group
acid derivatives
integer
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DK03706983T
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Danish (da)
English (en)
Inventor
Motoshi Shoda
Hiroshi Kuriyama
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Asahi Kasei Pharma Corp
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Publication of DK1477472T3 publication Critical patent/DK1477472T3/da

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DK03706983T 2002-02-21 2003-02-20 Substituerede phenylalkansyrederivater og anvendelse deraf DK1477472T3 (da)

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PCT/JP2003/001849 WO2003070686A1 (fr) 2002-02-21 2003-02-20 Derive de l'acide phenylalcanoyle substitue et son utilisation

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AT (1) ATE420847T1 (es)
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CA2477208C (en) * 2002-02-21 2010-11-30 Asahi Kasei Pharma Corporation Substituted phenylalkanoic acid derivatives and use thereof
EP1559422B1 (en) * 2002-11-08 2014-04-30 Takeda Pharmaceutical Company Limited Receptor function controlling agent
JP4594611B2 (ja) * 2002-11-08 2010-12-08 武田薬品工業株式会社 受容体機能調節剤
US7615575B2 (en) * 2003-02-13 2009-11-10 Wellstat Therapeutics Corporation Compounds for the treatment of metabolic disorders
EP1660427A4 (en) 2003-08-14 2006-12-20 Asahi Kasei Pharma Corp SUBSTITUTED ARYLALKANIC DERIVATIVE AND ITS USE
JP4922615B2 (ja) * 2003-11-26 2012-04-25 武田薬品工業株式会社 受容体機能調節剤
JP2007526324A (ja) * 2004-03-02 2007-09-13 スミスクライン・ビーチャム・コーポレイション Akt活性のある阻害剤
GB0409921D0 (en) * 2004-05-04 2004-06-09 Novartis Ag Organic compounds
TW200716588A (en) * 2005-06-02 2007-05-01 Kyowa Hakko Kogyo Kk A process for preparing dibenzoxepin derivative
US7405302B2 (en) * 2005-10-11 2008-07-29 Amira Pharmaceuticals, Inc. 5-lipoxygenase-activating protein (FLAP) inhibitors
AU2007274477B2 (en) * 2006-07-20 2010-11-25 Asahi Kasei Pharma Corporation Novel crystal of substituted phenylalkanoic acid and production process
TW200845988A (en) * 2007-04-05 2008-12-01 Astrazeneca Ab New compounds and their uses 707
US20100274022A1 (en) * 2007-04-26 2010-10-28 Pharmafrontier Co., Ltd. G protein-coupled receptor inhibitor and pharmaceutical product
US7928140B2 (en) * 2007-08-02 2011-04-19 Amgen Inc. Benzothiazole PI3 kinase modulators for cancer treatment
CA2712170C (en) * 2008-01-18 2014-04-22 Asahi Kasei Pharma Corporation Stable pharmaceutical composition
KR101269393B1 (ko) * 2008-04-28 2013-05-29 아사히 가세이 파마 가부시키가이샤 페닐프로피온산 유도체 및 이의 용도
PT2292592E (pt) 2008-06-05 2012-11-12 Asahi Kasei Pharma Corp Composto de sulfonamida e sua aplicação
CN102391264A (zh) * 2011-09-21 2012-03-28 河北九派制药有限公司 6-溴咪唑并[1,2-a]吡啶的制备方法
JP5802518B2 (ja) 2011-10-31 2015-10-28 公益財団法人微生物化学研究会 新規化合物、その製造方法、及びその用途
US8889730B2 (en) 2012-04-10 2014-11-18 Pfizer Inc. Indole and indazole compounds that activate AMPK
US9394285B2 (en) 2013-03-15 2016-07-19 Pfizer Inc. Indole and indazole compounds that activate AMPK
CN105315167A (zh) * 2014-08-01 2016-02-10 华东师范大学 一种2,2,3-三芳基-3-芳基氨基丙酸甲酯衍生物及其合成方法和应用
AU2015367977B9 (en) * 2014-12-24 2020-02-06 Lg Chem, Ltd Biaryl derivative as GPR120 agonist
JP6635999B2 (ja) * 2017-10-13 2020-01-29 株式会社ダイセル カリウム塩の製造方法、及びカリウム塩
CN110092774B (zh) * 2018-01-29 2022-04-08 中国科学院上海药物研究所 芳香丙酸类衍生物、及其制备方法和用途
JP2024506909A (ja) * 2021-02-12 2024-02-15 ニンバス サターン, インコーポレイテッド Hpk1アンタゴニスト及びその使用
WO2022187856A1 (en) 2021-03-05 2022-09-09 Nimbus Saturn, Inc. Hpk1 antagonists and uses thereof

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JP3802581B2 (ja) * 1995-03-01 2006-07-26 富山化学工業株式会社 新規なビフェニル誘導体またはその塩およびそれらを含有する抗炎症剤
US6376546B1 (en) * 1997-10-14 2002-04-23 Asahi Kasei Kabushiki Kaisha Biphenyl-5-alkanoic acid derivatives and use thereof
CA2477208C (en) * 2002-02-21 2010-11-30 Asahi Kasei Pharma Corporation Substituted phenylalkanoic acid derivatives and use thereof

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JP5048017B2 (ja) 2012-10-17
HK1076445A1 (en) 2006-01-20
JP2009167216A (ja) 2009-07-30
CN100387576C (zh) 2008-05-14
JP5000683B2 (ja) 2012-08-15
JP4390563B2 (ja) 2009-12-24
AU2003211384B2 (en) 2008-12-11
CA2477208C (en) 2010-11-30
CA2477208A1 (en) 2003-08-28
ATE420847T1 (de) 2009-01-15
PT1477472E (pt) 2009-03-17
DE60325830D1 (de) 2009-03-05
AU2003211384A1 (en) 2003-09-09
ES2319753T3 (es) 2009-05-12
KR20040094712A (ko) 2004-11-10
JPWO2003070686A1 (ja) 2005-06-09
WO2003070686A1 (fr) 2003-08-28
CN1653032A (zh) 2005-08-10
EP1477472A4 (en) 2005-12-14
KR100938950B1 (ko) 2010-01-26
JP2009167217A (ja) 2009-07-30
EP1477472A1 (en) 2004-11-17
EP1477472B1 (en) 2009-01-14
MXPA04008176A (es) 2004-11-26

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