DK1181290T3 - Polymorfer af et krystallinsk azabicyclo[2,2,2]octan-3-amin-citrat samt deres farmaceutiske præparater - Google Patents

Polymorfer af et krystallinsk azabicyclo[2,2,2]octan-3-amin-citrat samt deres farmaceutiske præparater

Info

Publication number
DK1181290T3
DK1181290T3 DK00925528T DK00925528T DK1181290T3 DK 1181290 T3 DK1181290 T3 DK 1181290T3 DK 00925528 T DK00925528 T DK 00925528T DK 00925528 T DK00925528 T DK 00925528T DK 1181290 T3 DK1181290 T3 DK 1181290T3
Authority
DK
Denmark
Prior art keywords
polymorphs
octane
well
pharmaceutical preparations
amine citrate
Prior art date
Application number
DK00925528T
Other languages
Danish (da)
English (en)
Inventor
Michael James Castaldi
George Joseph Quallich
Lewin Theophilus Wint
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of DK1181290T3 publication Critical patent/DK1181290T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK00925528T 1999-06-01 2000-05-18 Polymorfer af et krystallinsk azabicyclo[2,2,2]octan-3-amin-citrat samt deres farmaceutiske præparater DK1181290T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13699299P 1999-06-01 1999-06-01
PCT/IB2000/000665 WO2000073304A1 (en) 1999-06-01 2000-05-18 Polymorphs of a crystalline azabicyclo (2,2,2) octan-3-amine citrate and their pharmaceutical compositions

Publications (1)

Publication Number Publication Date
DK1181290T3 true DK1181290T3 (da) 2003-09-29

Family

ID=22475338

Family Applications (1)

Application Number Title Priority Date Filing Date
DK00925528T DK1181290T3 (da) 1999-06-01 2000-05-18 Polymorfer af et krystallinsk azabicyclo[2,2,2]octan-3-amin-citrat samt deres farmaceutiske præparater

Country Status (48)

Country Link
US (1) US6255320B1 (cs)
EP (1) EP1181290B1 (cs)
JP (1) JP3830816B2 (cs)
KR (1) KR100476606B1 (cs)
CN (1) CN1146565C (cs)
AP (1) AP2001002349A0 (cs)
AR (1) AR033331A1 (cs)
AT (1) ATE244239T1 (cs)
AU (1) AU767334B2 (cs)
BG (1) BG65240B1 (cs)
BR (1) BR0011094A (cs)
CA (1) CA2372238C (cs)
CO (1) CO5170463A1 (cs)
CY (1) CY2007011I2 (cs)
CZ (1) CZ295819B6 (cs)
DE (1) DE60003679T2 (cs)
DK (1) DK1181290T3 (cs)
DZ (1) DZ3050A1 (cs)
EA (1) EA003731B1 (cs)
EC (1) ECSP003508A (cs)
EE (1) EE200100656A (cs)
ES (1) ES2199825T3 (cs)
GT (1) GT200000087A (cs)
HN (1) HN2000000077A (cs)
HR (1) HRP20010904A2 (cs)
HU (1) HUP0201301A3 (cs)
IL (1) IL146406A0 (cs)
MA (1) MA26742A1 (cs)
MX (1) MXPA01012325A (cs)
MY (1) MY133508A (cs)
NO (1) NO20015848L (cs)
NZ (1) NZ515349A (cs)
OA (1) OA11956A (cs)
PA (1) PA8496101A1 (cs)
PE (1) PE20010209A1 (cs)
PL (1) PL196046B1 (cs)
PT (1) PT1181290E (cs)
SI (1) SI1181290T1 (cs)
SK (1) SK285820B6 (cs)
SV (1) SV2001000093A (cs)
TN (1) TNSN00120A1 (cs)
TR (1) TR200103473T2 (cs)
TW (1) TWI285204B (cs)
UA (1) UA66925C2 (cs)
UY (1) UY26176A1 (cs)
WO (1) WO2000073304A1 (cs)
YU (1) YU81101A (cs)
ZA (1) ZA200109775B (cs)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2638113T3 (es) * 2004-01-30 2017-10-18 Zoetis Services Llc Conservantes antimicrobianos para lograr una formulación de dosis múltiples usando ciclodextrinas beta para formas de dosificación líquidas
US20070155782A1 (en) * 2004-01-30 2007-07-05 Hickman Mary A Nk-1 receptor antagonists anesthesia recovery
US20070129328A1 (en) * 2004-01-30 2007-06-07 BOETTNER Wayne Pharmaceutical compositions of neurokinin receptor antagonists and cyclodextrin and methods for improved injection site toleration
AU2005210259A1 (en) * 2004-02-02 2005-08-18 Pfizer Products Inc. Process for preparation of 1-(2S,3S)-2-benzhydr yl-N-(5-tert-butyl-2-methoxybenzyl)quinuclidin-3-amine
WO2014144894A1 (en) * 2013-03-15 2014-09-18 Pearl Therapeutics, Inc. Methods and systems for conditioning of particulate crystalline materials
CN110577522B (zh) * 2018-06-07 2022-12-27 东莞市东阳光动物保健药品有限公司 马罗匹坦柠檬酸盐新晶型及其制备方法
CN112979639B (zh) * 2019-12-16 2025-08-08 凯默斯医药科技(上海)有限公司 一种马罗皮坦新晶型及其制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2103269C1 (ru) * 1991-05-31 1998-01-27 Пфайзер Инк. Производные хинуклидина или их фармацевтически приемлемые соли и фармацевтическая композиция
US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis
US5576317A (en) * 1994-12-09 1996-11-19 Pfizer Inc. NK-1 receptor antagonists and 5HT3 receptor antagonists for the treatment of emesis

Also Published As

Publication number Publication date
HRP20010904A2 (en) 2003-02-28
ES2199825T3 (es) 2004-03-01
HUP0201301A3 (en) 2002-10-28
EA003731B1 (ru) 2003-08-28
BG65240B1 (bg) 2007-09-28
EE200100656A (et) 2003-02-17
MA26742A1 (fr) 2004-12-20
EP1181290A1 (en) 2002-02-27
CN1353711A (zh) 2002-06-12
NO20015848D0 (no) 2001-11-30
JP2003501354A (ja) 2003-01-14
TR200103473T2 (tr) 2002-04-22
HUP0201301A2 (en) 2002-08-28
SV2001000093A (es) 2001-11-08
CO5170463A1 (es) 2002-06-27
DE60003679T2 (de) 2004-05-27
YU81101A (sh) 2004-07-15
AU4424800A (en) 2000-12-18
PE20010209A1 (es) 2001-03-01
MY133508A (en) 2007-11-30
BG106204A (en) 2002-07-31
JP3830816B2 (ja) 2006-10-11
CA2372238C (en) 2006-12-19
AR033331A1 (es) 2003-12-17
CZ20014269A3 (cs) 2002-04-17
UA66925C2 (uk) 2004-06-15
WO2000073304A1 (en) 2000-12-07
HK1046284A1 (en) 2003-01-03
DZ3050A1 (fr) 2004-03-27
PL196046B1 (pl) 2007-11-30
TNSN00120A1 (fr) 2005-11-10
HN2000000077A (es) 2001-02-02
EA200101108A1 (ru) 2002-04-25
SK285820B6 (sk) 2007-09-06
IL146406A0 (en) 2002-07-25
SI1181290T1 (en) 2003-12-31
NZ515349A (en) 2004-03-26
DE60003679D1 (de) 2003-08-07
EP1181290B1 (en) 2003-07-02
KR20020010688A (ko) 2002-02-04
ECSP003508A (es) 2002-02-25
CZ295819B6 (cs) 2005-11-16
AP2001002349A0 (en) 2001-12-31
SK17332001A3 (sk) 2002-07-02
ZA200109775B (en) 2002-11-28
CY2007011I1 (el) 2010-07-28
BR0011094A (pt) 2002-03-19
AU767334B2 (en) 2003-11-06
PL352716A1 (en) 2003-09-08
GT200000087A (es) 2001-11-22
MXPA01012325A (es) 2002-07-22
CA2372238A1 (en) 2000-12-07
TWI285204B (en) 2007-08-11
ATE244239T1 (de) 2003-07-15
PA8496101A1 (es) 2002-07-30
OA11956A (en) 2006-04-13
CN1146565C (zh) 2004-04-21
UY26176A1 (es) 2000-12-29
KR100476606B1 (ko) 2005-03-18
NO20015848L (no) 2001-12-18
US6255320B1 (en) 2001-07-03
CY2007011I2 (el) 2010-07-28
PT1181290E (pt) 2003-09-30

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