HUP0201301A3 - Polymorphs of a crystalline azabicyclo(2,2,2)octan-3-amine citrate and their pharmaceutical compositions and process for preparation of the compounds - Google Patents

Polymorphs of a crystalline azabicyclo(2,2,2)octan-3-amine citrate and their pharmaceutical compositions and process for preparation of the compounds

Info

Publication number
HUP0201301A3
HUP0201301A3 HU0201301A HUP0201301A HUP0201301A3 HU P0201301 A3 HUP0201301 A3 HU P0201301A3 HU 0201301 A HU0201301 A HU 0201301A HU P0201301 A HUP0201301 A HU P0201301A HU P0201301 A3 HUP0201301 A3 HU P0201301A3
Authority
HU
Hungary
Prior art keywords
octan
polymorphs
compounds
preparation
pharmaceutical compositions
Prior art date
Application number
HU0201301A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of HUP0201301A2 publication Critical patent/HUP0201301A2/hu
Publication of HUP0201301A3 publication Critical patent/HUP0201301A3/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HU0201301A 1999-06-01 2000-05-18 Polymorphs of a crystalline azabicyclo(2,2,2)octan-3-amine citrate and their pharmaceutical compositions and process for preparation of the compounds HUP0201301A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13699299P 1999-06-01 1999-06-01

Publications (2)

Publication Number Publication Date
HUP0201301A2 HUP0201301A2 (en) 2002-08-28
HUP0201301A3 true HUP0201301A3 (en) 2002-10-28

Family

ID=22475338

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0201301A HUP0201301A3 (en) 1999-06-01 2000-05-18 Polymorphs of a crystalline azabicyclo(2,2,2)octan-3-amine citrate and their pharmaceutical compositions and process for preparation of the compounds

Country Status (49)

Country Link
US (1) US6255320B1 (hu)
EP (1) EP1181290B1 (hu)
JP (1) JP3830816B2 (hu)
KR (1) KR100476606B1 (hu)
CN (1) CN1146565C (hu)
AP (1) AP2001002349A0 (hu)
AR (1) AR033331A1 (hu)
AT (1) ATE244239T1 (hu)
AU (1) AU767334B2 (hu)
BG (1) BG65240B1 (hu)
BR (1) BR0011094A (hu)
CA (1) CA2372238C (hu)
CO (1) CO5170463A1 (hu)
CY (1) CY2007011I2 (hu)
CZ (1) CZ295819B6 (hu)
DE (1) DE60003679T2 (hu)
DK (1) DK1181290T3 (hu)
DZ (1) DZ3050A1 (hu)
EA (1) EA003731B1 (hu)
EC (1) ECSP003508A (hu)
EE (1) EE200100656A (hu)
ES (1) ES2199825T3 (hu)
GT (1) GT200000087A (hu)
HK (1) HK1046284A1 (hu)
HN (1) HN2000000077A (hu)
HR (1) HRP20010904A2 (hu)
HU (1) HUP0201301A3 (hu)
IL (1) IL146406A0 (hu)
MA (1) MA26742A1 (hu)
MX (1) MXPA01012325A (hu)
MY (1) MY133508A (hu)
NO (1) NO20015848L (hu)
NZ (1) NZ515349A (hu)
OA (1) OA11956A (hu)
PA (1) PA8496101A1 (hu)
PE (1) PE20010209A1 (hu)
PL (1) PL196046B1 (hu)
PT (1) PT1181290E (hu)
SI (1) SI1181290T1 (hu)
SK (1) SK285820B6 (hu)
SV (1) SV2001000093A (hu)
TN (1) TNSN00120A1 (hu)
TR (1) TR200103473T2 (hu)
TW (1) TWI285204B (hu)
UA (1) UA66925C2 (hu)
UY (1) UY26176A1 (hu)
WO (1) WO2000073304A1 (hu)
YU (1) YU81101A (hu)
ZA (1) ZA200109775B (hu)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA06008648A (es) * 2004-01-30 2006-09-04 Pfizer Prod Inc Composiciones farmaceuticas de antagonistas del receptor de neuroquinina y ciclodextrina y metodos para una tolerancia mejorada en el sitio de inyeccion.
WO2005082416A2 (en) * 2004-01-30 2005-09-09 Pfizer Products Inc. Antimicrobial preservatives to achieve multi-dose formulation using beta-cyclodextrins for liquid dosage forms
JP2007519701A (ja) * 2004-01-30 2007-07-19 ファイザー・プロダクツ・インク 麻酔回復を改善するためのnk−1受容体拮抗剤
JP2007519710A (ja) * 2004-02-02 2007-07-19 ファイザー・プロダクツ・インク 1−(2S,3S)−2−ベンズヒドリル−N−(5−tert−ブチル−2−メトキシベンジル)キヌクリジン−3−アミンの製造方法
KR102391332B1 (ko) * 2013-03-15 2022-04-26 펄 테라퓨틱스 인코포레이티드 미립자 결정질 재료를 컨디셔닝하는 방법 및 시스템
CN110577522B (zh) * 2018-06-07 2022-12-27 东莞市东阳光动物保健药品有限公司 马罗匹坦柠檬酸盐新晶型及其制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69208877T2 (de) * 1991-05-31 1996-07-25 Pfizer Chinuclidinderivate
US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis
US5576317A (en) * 1994-12-09 1996-11-19 Pfizer Inc. NK-1 receptor antagonists and 5HT3 receptor antagonists for the treatment of emesis

Also Published As

Publication number Publication date
CY2007011I1 (el) 2010-07-28
HRP20010904A2 (en) 2003-02-28
TR200103473T2 (tr) 2002-04-22
SK285820B6 (sk) 2007-09-06
EE200100656A (et) 2003-02-17
YU81101A (sh) 2004-07-15
ECSP003508A (es) 2002-02-25
IL146406A0 (en) 2002-07-25
CN1353711A (zh) 2002-06-12
CZ295819B6 (cs) 2005-11-16
BG106204A (en) 2002-07-31
PE20010209A1 (es) 2001-03-01
HK1046284A1 (en) 2003-01-03
MXPA01012325A (es) 2002-07-22
CZ20014269A3 (cs) 2002-04-17
NO20015848L (no) 2001-12-18
US6255320B1 (en) 2001-07-03
EP1181290B1 (en) 2003-07-02
PT1181290E (pt) 2003-09-30
UA66925C2 (uk) 2004-06-15
NZ515349A (en) 2004-03-26
EA003731B1 (ru) 2003-08-28
KR20020010688A (ko) 2002-02-04
UY26176A1 (es) 2000-12-29
CA2372238C (en) 2006-12-19
OA11956A (en) 2006-04-13
NO20015848D0 (no) 2001-11-30
KR100476606B1 (ko) 2005-03-18
SI1181290T1 (en) 2003-12-31
AR033331A1 (es) 2003-12-17
TNSN00120A1 (fr) 2005-11-10
DE60003679D1 (de) 2003-08-07
DK1181290T3 (da) 2003-09-29
MA26742A1 (fr) 2004-12-20
PL352716A1 (en) 2003-09-08
CN1146565C (zh) 2004-04-21
JP3830816B2 (ja) 2006-10-11
MY133508A (en) 2007-11-30
AU767334B2 (en) 2003-11-06
CO5170463A1 (es) 2002-06-27
ZA200109775B (en) 2002-11-28
EP1181290A1 (en) 2002-02-27
ES2199825T3 (es) 2004-03-01
SK17332001A3 (sk) 2002-07-02
BG65240B1 (bg) 2007-09-28
GT200000087A (es) 2001-11-22
TWI285204B (en) 2007-08-11
BR0011094A (pt) 2002-03-19
EA200101108A1 (ru) 2002-04-25
AU4424800A (en) 2000-12-18
CY2007011I2 (el) 2010-07-28
JP2003501354A (ja) 2003-01-14
PL196046B1 (pl) 2007-11-30
SV2001000093A (es) 2001-11-08
HUP0201301A2 (en) 2002-08-28
PA8496101A1 (es) 2002-07-30
DE60003679T2 (de) 2004-05-27
WO2000073304A1 (en) 2000-12-07
HN2000000077A (es) 2001-02-02
DZ3050A1 (fr) 2004-03-27
ATE244239T1 (de) 2003-07-15
CA2372238A1 (en) 2000-12-07
AP2001002349A0 (en) 2001-12-31

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Legal Events

Date Code Title Description
FD9A Lapse of provisional protection due to non-payment of fees