IL146406A0 - Polymorphs of crystalline azabicyclo (2,2,2) octan-3-amine citrate and their pharmaceutical compositions - Google Patents

Polymorphs of crystalline azabicyclo (2,2,2) octan-3-amine citrate and their pharmaceutical compositions

Info

Publication number
IL146406A0
IL146406A0 IL14640600A IL14640600A IL146406A0 IL 146406 A0 IL146406 A0 IL 146406A0 IL 14640600 A IL14640600 A IL 14640600A IL 14640600 A IL14640600 A IL 14640600A IL 146406 A0 IL146406 A0 IL 146406A0
Authority
IL
Israel
Prior art keywords
octan
polymorphs
pharmaceutical compositions
amine citrate
azabicyclo
Prior art date
Application number
IL14640600A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of IL146406A0 publication Critical patent/IL146406A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Otolaryngology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL14640600A 1999-06-01 2000-05-18 Polymorphs of crystalline azabicyclo (2,2,2) octan-3-amine citrate and their pharmaceutical compositions IL146406A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13699299P 1999-06-01 1999-06-01
PCT/IB2000/000665 WO2000073304A1 (en) 1999-06-01 2000-05-18 Polymorphs of a crystalline azabicyclo (2,2,2) octan-3-amine citrate and their pharmaceutical compositions

Publications (1)

Publication Number Publication Date
IL146406A0 true IL146406A0 (en) 2002-07-25

Family

ID=22475338

Family Applications (1)

Application Number Title Priority Date Filing Date
IL14640600A IL146406A0 (en) 1999-06-01 2000-05-18 Polymorphs of crystalline azabicyclo (2,2,2) octan-3-amine citrate and their pharmaceutical compositions

Country Status (49)

Country Link
US (1) US6255320B1 (xx)
EP (1) EP1181290B1 (xx)
JP (1) JP3830816B2 (xx)
KR (1) KR100476606B1 (xx)
CN (1) CN1146565C (xx)
AP (1) AP2001002349A0 (xx)
AR (1) AR033331A1 (xx)
AT (1) ATE244239T1 (xx)
AU (1) AU767334B2 (xx)
BG (1) BG65240B1 (xx)
BR (1) BR0011094A (xx)
CA (1) CA2372238C (xx)
CO (1) CO5170463A1 (xx)
CY (1) CY2007011I1 (xx)
CZ (1) CZ295819B6 (xx)
DE (1) DE60003679T2 (xx)
DK (1) DK1181290T3 (xx)
DZ (1) DZ3050A1 (xx)
EA (1) EA003731B1 (xx)
EC (1) ECSP003508A (xx)
EE (1) EE200100656A (xx)
ES (1) ES2199825T3 (xx)
GT (1) GT200000087A (xx)
HK (1) HK1046284A1 (xx)
HN (1) HN2000000077A (xx)
HR (1) HRP20010904A2 (xx)
HU (1) HUP0201301A3 (xx)
IL (1) IL146406A0 (xx)
MA (1) MA26742A1 (xx)
MX (1) MXPA01012325A (xx)
MY (1) MY133508A (xx)
NO (1) NO20015848L (xx)
NZ (1) NZ515349A (xx)
OA (1) OA11956A (xx)
PA (1) PA8496101A1 (xx)
PE (1) PE20010209A1 (xx)
PL (1) PL196046B1 (xx)
PT (1) PT1181290E (xx)
SI (1) SI1181290T1 (xx)
SK (1) SK285820B6 (xx)
SV (1) SV2001000093A (xx)
TN (1) TNSN00120A1 (xx)
TR (1) TR200103473T2 (xx)
TW (1) TWI285204B (xx)
UA (1) UA66925C2 (xx)
UY (1) UY26176A1 (xx)
WO (1) WO2000073304A1 (xx)
YU (1) YU81101A (xx)
ZA (1) ZA200109775B (xx)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070155782A1 (en) * 2004-01-30 2007-07-05 Hickman Mary A Nk-1 receptor antagonists anesthesia recovery
RU2332997C2 (ru) * 2004-01-30 2008-09-10 Пфайзер Продактс Инк. АНТИМИКРОБНЫЕ КОНСЕРВАНТЫ ДЛЯ ДОСТИЖЕНИЯ МУЛЬТИДОЗОВЫХ РЕЦЕПТУР С ИСПОЛЬЗОВАНИЕМ β-ЦИКЛОДЕКСТРИНОВ ДЛЯ ЖИДКИХ ЛЕКАРСТВЕННЫХ ФОРМ
EP1713506A1 (en) * 2004-01-30 2006-10-25 Pfizer Products Incorporated Pharmaceutical compositions of neurokinin receptor antagonists and cyclodextrin and methods for improved injection site toleration
RU2320659C9 (ru) * 2004-02-02 2008-07-20 Пфайзер Продактс Инк. Способы получения 1-(2s, 3s)-2-бензгидрил-n-(5-трет-бутил-2-метоксибензил)хинуклидин-3-амина в виде камфорсульфатной соли, цитратной соли и свободного основания и промежуточное соединение
CN105188679B (zh) * 2013-03-15 2018-10-16 珍珠治疗公司 用于微粒晶体材料的状态调节的方法和系统
CN110577522B (zh) * 2018-06-07 2022-12-27 东莞市东阳光动物保健药品有限公司 马罗匹坦柠檬酸盐新晶型及其制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0733386B2 (ja) * 1991-05-31 1995-04-12 フアイザー・インコーポレイテツド キヌクリジン誘導体
US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis
US5576317A (en) * 1994-12-09 1996-11-19 Pfizer Inc. NK-1 receptor antagonists and 5HT3 receptor antagonists for the treatment of emesis

Also Published As

Publication number Publication date
HN2000000077A (es) 2001-02-02
CN1353711A (zh) 2002-06-12
SI1181290T1 (en) 2003-12-31
ES2199825T3 (es) 2004-03-01
PL196046B1 (pl) 2007-11-30
CA2372238C (en) 2006-12-19
EA200101108A1 (ru) 2002-04-25
EA003731B1 (ru) 2003-08-28
MY133508A (en) 2007-11-30
YU81101A (sh) 2004-07-15
ATE244239T1 (de) 2003-07-15
CZ20014269A3 (cs) 2002-04-17
NO20015848D0 (no) 2001-11-30
HUP0201301A3 (en) 2002-10-28
UY26176A1 (es) 2000-12-29
AR033331A1 (es) 2003-12-17
DE60003679T2 (de) 2004-05-27
PA8496101A1 (es) 2002-07-30
WO2000073304A1 (en) 2000-12-07
OA11956A (en) 2006-04-13
UA66925C2 (uk) 2004-06-15
KR100476606B1 (ko) 2005-03-18
DK1181290T3 (da) 2003-09-29
BR0011094A (pt) 2002-03-19
CN1146565C (zh) 2004-04-21
HUP0201301A2 (en) 2002-08-28
GT200000087A (es) 2001-11-22
TR200103473T2 (tr) 2002-04-22
SK17332001A3 (sk) 2002-07-02
AU4424800A (en) 2000-12-18
CY2007011I2 (el) 2010-07-28
JP2003501354A (ja) 2003-01-14
HK1046284A1 (en) 2003-01-03
KR20020010688A (ko) 2002-02-04
AU767334B2 (en) 2003-11-06
BG106204A (en) 2002-07-31
CO5170463A1 (es) 2002-06-27
TNSN00120A1 (fr) 2005-11-10
EE200100656A (et) 2003-02-17
CA2372238A1 (en) 2000-12-07
MXPA01012325A (es) 2002-07-22
SK285820B6 (sk) 2007-09-06
EP1181290B1 (en) 2003-07-02
BG65240B1 (bg) 2007-09-28
ZA200109775B (en) 2002-11-28
PE20010209A1 (es) 2001-03-01
NO20015848L (no) 2001-12-18
US6255320B1 (en) 2001-07-03
TWI285204B (en) 2007-08-11
NZ515349A (en) 2004-03-26
EP1181290A1 (en) 2002-02-27
DE60003679D1 (de) 2003-08-07
JP3830816B2 (ja) 2006-10-11
DZ3050A1 (fr) 2004-03-27
AP2001002349A0 (en) 2001-12-31
MA26742A1 (fr) 2004-12-20
PL352716A1 (en) 2003-09-08
SV2001000093A (es) 2001-11-08
PT1181290E (pt) 2003-09-30
CY2007011I1 (el) 2010-07-28
HRP20010904A2 (en) 2003-02-28
CZ295819B6 (cs) 2005-11-16
ECSP003508A (es) 2002-02-25

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Legal Events

Date Code Title Description
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees