DK1100796T3 - Fremgangsmåde til fremstilling af en ikke-krystallinsk anhydratform af paroxetinhydrochlorid - Google Patents
Fremgangsmåde til fremstilling af en ikke-krystallinsk anhydratform af paroxetinhydrochloridInfo
- Publication number
- DK1100796T3 DK1100796T3 DK99940290T DK99940290T DK1100796T3 DK 1100796 T3 DK1100796 T3 DK 1100796T3 DK 99940290 T DK99940290 T DK 99940290T DK 99940290 T DK99940290 T DK 99940290T DK 1100796 T3 DK1100796 T3 DK 1100796T3
- Authority
- DK
- Denmark
- Prior art keywords
- preparing
- paroxetine hydrochloride
- anhydrate form
- crystalline anhydrate
- crystalline
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4525—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9817196.0A GB9817196D0 (en) | 1998-08-07 | 1998-08-07 | Novel process |
| GBGB9828777.4A GB9828777D0 (en) | 1998-12-29 | 1998-12-29 | Novel compounds |
| PCT/GB1999/002592 WO2000008017A1 (en) | 1998-08-07 | 1999-08-06 | Process for the preparation of a non-crystalline anhydrate form of paroxetine hydrochloride |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1100796T3 true DK1100796T3 (da) | 2003-08-25 |
Family
ID=26314179
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK99940290T DK1100796T3 (da) | 1998-08-07 | 1999-08-06 | Fremgangsmåde til fremstilling af en ikke-krystallinsk anhydratform af paroxetinhydrochlorid |
Country Status (24)
| Country | Link |
|---|---|
| EP (2) | EP1100796B1 (bg) |
| JP (1) | JP2002522434A (bg) |
| KR (1) | KR20010072323A (bg) |
| CN (1) | CN1321155A (bg) |
| AP (2) | AP0102072A0 (bg) |
| AT (1) | ATE239016T1 (bg) |
| AU (1) | AU5428999A (bg) |
| BG (1) | BG105310A (bg) |
| BR (1) | BR9912858A (bg) |
| CA (1) | CA2339857A1 (bg) |
| DE (1) | DE69907467T2 (bg) |
| DK (1) | DK1100796T3 (bg) |
| EA (1) | EA200100221A1 (bg) |
| ES (1) | ES2198940T3 (bg) |
| HK (1) | HK1038230A1 (bg) |
| HU (1) | HUP0105466A3 (bg) |
| ID (1) | ID27914A (bg) |
| IL (1) | IL141286A0 (bg) |
| NO (1) | NO20010629L (bg) |
| PL (1) | PL345885A1 (bg) |
| PT (1) | PT1100796E (bg) |
| SK (1) | SK1972001A3 (bg) |
| TR (1) | TR200100444T2 (bg) |
| WO (1) | WO2000008017A1 (bg) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE69739561D1 (de) | 1996-06-13 | 2009-10-15 | Sumitomo Chemical Co | Piperidin Derivative als Zwischenprodukte zur Herstellung von Paroxetine und Verfahren zu ihrer Herstellung |
| JP3796351B2 (ja) | 1998-04-13 | 2006-07-12 | 住友化学株式会社 | パロキセチン塩酸塩無水和物の乾燥方法 |
| GB9923446D0 (en) * | 1999-10-04 | 1999-12-08 | Smithkline Beecham Plc | Novel process |
| AU2002224322A1 (en) * | 2000-11-17 | 2002-05-27 | Eli Lilly And Company | Lactam dipeptide and its use in inhibiting beta-amyloid peptiderelease |
| US8697094B2 (en) | 2002-10-16 | 2014-04-15 | Takeda Pharmaceutical Company Limited | Stable solid preparations |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1422263A (en) * | 1973-01-30 | 1976-01-21 | Ferrosan As | 4-phenyl-piperidine compounds |
| ES2058061T3 (es) * | 1985-10-25 | 1994-11-01 | Beecham Group Plc | Derivado de piperidina, su preparacion y su uso como medicamento. |
| AR001982A1 (es) * | 1995-02-06 | 1998-01-07 | Smithkline Beecham Plc | Clorhidrato de paroxetina anhidratado, y procedimiento para su preparacion |
| NZ336587A (en) * | 1997-01-15 | 2001-01-26 | Smithkline Beecham P | Spray dried paroxetine compositions using organic solvent selected from pyridine, acetic acid, acetonitrile, acetone, ethanol, propan-1-ol or tetrahydrofuran |
| JP3796351B2 (ja) * | 1998-04-13 | 2006-07-12 | 住友化学株式会社 | パロキセチン塩酸塩無水和物の乾燥方法 |
-
1999
- 1999-08-06 IL IL14128699A patent/IL141286A0/xx unknown
- 1999-08-06 JP JP2000563650A patent/JP2002522434A/ja active Pending
- 1999-08-06 PL PL99345885A patent/PL345885A1/xx not_active Application Discontinuation
- 1999-08-06 BR BR9912858-6A patent/BR9912858A/pt not_active Application Discontinuation
- 1999-08-06 EA EA200100221A patent/EA200100221A1/ru unknown
- 1999-08-06 AU AU54289/99A patent/AU5428999A/en not_active Abandoned
- 1999-08-06 DK DK99940290T patent/DK1100796T3/da active
- 1999-08-06 EP EP99940290A patent/EP1100796B1/en not_active Expired - Lifetime
- 1999-08-06 TR TR2001/00444T patent/TR200100444T2/xx unknown
- 1999-08-06 ID IDW20010296A patent/ID27914A/id unknown
- 1999-08-06 DE DE69907467T patent/DE69907467T2/de not_active Expired - Fee Related
- 1999-08-06 CA CA002339857A patent/CA2339857A1/en not_active Abandoned
- 1999-08-06 PT PT99940290T patent/PT1100796E/pt unknown
- 1999-08-06 EP EP02080022A patent/EP1321465A3/en not_active Withdrawn
- 1999-08-06 AT AT99940290T patent/ATE239016T1/de not_active IP Right Cessation
- 1999-08-06 ES ES99940290T patent/ES2198940T3/es not_active Expired - Lifetime
- 1999-08-06 AP APAP/P/2001/002072A patent/AP0102072A0/en unknown
- 1999-08-06 SK SK197-2001A patent/SK1972001A3/sk unknown
- 1999-08-06 CN CN99811643A patent/CN1321155A/zh active Pending
- 1999-08-06 WO PCT/GB1999/002592 patent/WO2000008017A1/en not_active Application Discontinuation
- 1999-08-06 AP AP2001002072A patent/AP2001002072A0/xx unknown
- 1999-08-06 KR KR1020017001635A patent/KR20010072323A/ko not_active Application Discontinuation
- 1999-08-06 HU HU0105466A patent/HUP0105466A3/hu unknown
-
2001
- 2001-02-06 NO NO20010629A patent/NO20010629L/no not_active Application Discontinuation
- 2001-03-06 BG BG105310A patent/BG105310A/bg unknown
- 2001-11-08 HK HK01107862A patent/HK1038230A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| AP2001002072A0 (en) | 2001-03-31 |
| PT1100796E (pt) | 2003-09-30 |
| BG105310A (bg) | 2001-12-29 |
| JP2002522434A (ja) | 2002-07-23 |
| DE69907467T2 (de) | 2004-03-11 |
| BR9912858A (pt) | 2001-11-20 |
| ATE239016T1 (de) | 2003-05-15 |
| AP0102072A0 (en) | 2001-02-06 |
| EP1100796A1 (en) | 2001-05-23 |
| NO20010629L (no) | 2001-03-20 |
| HK1038230A1 (en) | 2002-03-08 |
| KR20010072323A (ko) | 2001-07-31 |
| WO2000008017A1 (en) | 2000-02-17 |
| HUP0105466A3 (en) | 2002-11-28 |
| CA2339857A1 (en) | 2000-02-17 |
| HUP0105466A2 (hu) | 2002-05-29 |
| EA200100221A1 (ru) | 2001-08-27 |
| EP1321465A2 (en) | 2003-06-25 |
| SK1972001A3 (en) | 2001-08-06 |
| AU5428999A (en) | 2000-02-28 |
| TR200100444T2 (tr) | 2001-07-23 |
| NO20010629D0 (no) | 2001-02-06 |
| PL345885A1 (en) | 2002-01-14 |
| ID27914A (id) | 2001-05-03 |
| ES2198940T3 (es) | 2004-02-01 |
| IL141286A0 (en) | 2002-03-10 |
| EP1321465A3 (en) | 2003-09-03 |
| EP1100796B1 (en) | 2003-05-02 |
| CN1321155A (zh) | 2001-11-07 |
| DE69907467D1 (de) | 2003-06-05 |
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