DK0934319T3 - 1H-pyrido[3,4-b]indol-4-carboxamidderivater, fremstilling heraf og terapeutiske anvendelser heraf - Google Patents

1H-pyrido[3,4-b]indol-4-carboxamidderivater, fremstilling heraf og terapeutiske anvendelser heraf

Info

Publication number
DK0934319T3
DK0934319T3 DK97943932T DK97943932T DK0934319T3 DK 0934319 T3 DK0934319 T3 DK 0934319T3 DK 97943932 T DK97943932 T DK 97943932T DK 97943932 T DK97943932 T DK 97943932T DK 0934319 T3 DK0934319 T3 DK 0934319T3
Authority
DK
Denmark
Prior art keywords
pyrido
indole
preparation
therapeutic uses
carboxamide derivatives
Prior art date
Application number
DK97943932T
Other languages
Danish (da)
English (en)
Inventor
Christian Maloizel
Pascal George
Yannick Evanno
Mireille Sevrin
Odette Legalloudec
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Application granted granted Critical
Publication of DK0934319T3 publication Critical patent/DK0934319T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Anesthesiology (AREA)
  • Psychology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
DK97943932T 1996-10-08 1997-10-03 1H-pyrido[3,4-b]indol-4-carboxamidderivater, fremstilling heraf og terapeutiske anvendelser heraf DK0934319T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9612229A FR2754262B1 (fr) 1996-10-08 1996-10-08 Derives de 1h-pyrido[3,4-b]indole-4-carboxamide, leur preparation et leur application en therapeutique
PCT/FR1997/001750 WO1998015552A1 (fr) 1996-10-08 1997-10-03 DERIVES DE 1H-PYRIDO[3,4-b]INDOLE-4-CARBOXAMIDE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE

Publications (1)

Publication Number Publication Date
DK0934319T3 true DK0934319T3 (da) 2002-09-30

Family

ID=9496449

Family Applications (1)

Application Number Title Priority Date Filing Date
DK97943932T DK0934319T3 (da) 1996-10-08 1997-10-03 1H-pyrido[3,4-b]indol-4-carboxamidderivater, fremstilling heraf og terapeutiske anvendelser heraf

Country Status (33)

Country Link
US (1) US6075021A (ru)
EP (1) EP0934319B1 (ru)
JP (1) JP4227197B2 (ru)
KR (1) KR100488095B1 (ru)
CN (1) CN1089765C (ru)
AR (1) AR009112A1 (ru)
AT (1) ATE218567T1 (ru)
AU (1) AU721102B2 (ru)
BG (1) BG63751B1 (ru)
BR (1) BR9711879A (ru)
CA (1) CA2266376A1 (ru)
CO (1) CO4910141A1 (ru)
CY (1) CY2291B1 (ru)
CZ (1) CZ298906B6 (ru)
DE (1) DE69713124T2 (ru)
DK (1) DK0934319T3 (ru)
EE (1) EE03830B1 (ru)
ES (1) ES2178008T3 (ru)
FR (1) FR2754262B1 (ru)
HK (1) HK1023338A1 (ru)
HU (1) HUP9904623A3 (ru)
IL (1) IL129018A0 (ru)
NO (1) NO311938B1 (ru)
NZ (1) NZ334708A (ru)
PL (1) PL188244B1 (ru)
PT (1) PT934319E (ru)
RU (1) RU2180904C2 (ru)
SK (1) SK282970B6 (ru)
TR (1) TR199900712T2 (ru)
TW (1) TW461889B (ru)
UA (1) UA57037C2 (ru)
WO (1) WO1998015552A1 (ru)
ZA (1) ZA978970B (ru)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2766823B1 (fr) 1997-07-30 1999-10-08 Synthelabo Derives de 4-oxo-3,5-dihydro-4h-pyridazino[4,5-b] indole-1-acetamide, leur preparation et leur application en therapeutique
FR2788776B1 (fr) * 1999-01-26 2001-02-23 Synthelabo Derives de 4-oxo-3, 5-dihydro-4h-pyridazino [4,5-b] indole-1 -carboxamide, leur preparation et leur application en therapeutique
FR2788696B1 (fr) * 1999-01-26 2004-03-05 Synthelabo Utilisation de derives de pyridazino [4,5-b] indole-1-acetamide pour la preparation de medicaments destines aux maladies du systeme nerveux central
FR2811990A1 (fr) * 2000-07-24 2002-01-25 Sanofi Synthelabo DERIVES DE 1-(4-OXO-3,5-DIHYDRO-4H-PYRIDAZINO[4,5-b]INDOLE-1 -CARBONYL)PIPERAZINE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
FR2811897A1 (fr) * 2000-07-24 2002-01-25 Sanofi Synthelabo UTILISATION DE DERIVES DE PYRIDAZINO[4,5-b]INDOLE-1- ACETAMIDE POUR LA PREPARATION DE MEDICAMENTS DESTINES AU TRAITEMENT DES DYSFONCTIONNEMENTS DES RECEPTEURS DE TYPE PERIPHERIQUE AUX BENZODIAZEPINES
FR2833953B1 (fr) * 2001-12-21 2004-12-03 Sanofi Synthelabo DERIVES DE 3-HETEROARYL-3,5-DIHYDRO-4-OXO-4H-PYRIDAZINO [4,5-b]INDOLE-1-CARBOXAMIDE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
FR2838124B1 (fr) * 2002-04-03 2004-05-28 Sanofi Synthelabo Derives de 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino [4,5-b]indole-1-acetamide, leur preparation et leur application en therapeutique
PA8586801A1 (es) * 2002-10-31 2005-02-04 Pfizer Inhibidores de hiv-integrasa, composiciones farmaceuticas y metodos para su uso
CA2513141A1 (en) * 2003-01-27 2004-08-12 Pfizer Inc. Hiv-integrase inhibitors, pharmaceutical compositions, and methods for their use
WO2005103051A1 (en) * 2004-04-26 2005-11-03 Pfizer Inc. Inhibitors of the hiv integrase enzyme
EP1756103A2 (en) * 2004-04-26 2007-02-28 Pfizer, Inc. Pyrrolopyridine derivatives and their use as hiv-integrase inhibitors
KR20140002810A (ko) * 2005-05-05 2014-01-08 사노피-아벤티스 유.에스. 엘엘씨 안정한 나노입자 제형
CA2623506A1 (en) * 2005-10-07 2007-04-19 Pfizer Products Inc. Inhibitors of the hiv integrase enzyme
UA95788C2 (en) 2005-12-15 2011-09-12 Ф. Хоффманн-Ля Рош Аг Fused pyrrole derivatives
PE20080714A1 (es) * 2006-06-05 2008-07-31 Novartis Ag DERIVADOS HETEROCICLICOS COMO MODULADORES DE LA ACTIVIDAD DE LA ESTEARIL-CoA-DESATURASA
CN1946120B (zh) * 2006-10-20 2010-05-12 华为技术有限公司 实现话单关联的方法及系统
KR100688448B1 (ko) * 2006-12-06 2007-03-02 (주)경진건축사사무소 건축물 내부 조적구조

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2724384B1 (fr) * 1994-09-14 1999-04-16 Cemaf Nouveaux derives de la 3,4-dihydro beta-carboline agonistes de la melatonine, leur procede de preparation et leur utilisation a titre de medicament

Also Published As

Publication number Publication date
JP2001508403A (ja) 2001-06-26
CA2266376A1 (en) 1998-04-16
EE03830B1 (et) 2002-08-15
BG103301A (en) 2000-05-31
IL129018A0 (en) 2000-02-17
TR199900712T2 (xx) 1999-06-21
WO1998015552A1 (fr) 1998-04-16
HK1023338A1 (en) 2000-09-08
FR2754262A1 (fr) 1998-04-10
CO4910141A1 (es) 2000-04-24
ES2178008T3 (es) 2002-12-16
US6075021A (en) 2000-06-13
KR100488095B1 (ko) 2005-05-09
NZ334708A (en) 2000-10-27
NO311938B1 (no) 2002-02-18
RU2180904C2 (ru) 2002-03-27
AU721102B2 (en) 2000-06-22
EP0934319A1 (fr) 1999-08-11
CN1089765C (zh) 2002-08-28
KR20000048992A (ko) 2000-07-25
EP0934319B1 (fr) 2002-06-05
JP4227197B2 (ja) 2009-02-18
AR009112A1 (es) 2000-03-08
NO991624D0 (no) 1999-04-06
SK282970B6 (sk) 2003-01-09
PL188244B1 (pl) 2005-01-31
CY2291B1 (en) 2003-07-04
SK45199A3 (en) 2000-02-14
BG63751B1 (bg) 2002-11-29
ATE218567T1 (de) 2002-06-15
UA57037C2 (ru) 2003-06-16
CZ298906B6 (cs) 2008-03-12
DE69713124D1 (de) 2002-07-11
PT934319E (pt) 2002-10-31
AU4559497A (en) 1998-05-05
BR9711879A (pt) 1999-08-24
HUP9904623A2 (hu) 2000-06-28
DE69713124T2 (de) 2003-01-30
HUP9904623A3 (en) 2001-03-28
FR2754262B1 (fr) 1998-10-30
NO991624L (no) 1999-06-07
CN1233248A (zh) 1999-10-27
CZ119399A3 (cs) 1999-07-14
PL332643A1 (en) 1999-09-27
EE9900155A (et) 1999-12-15
ZA978970B (en) 1998-04-20
TW461889B (en) 2001-11-01

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