DK0868420T3 - 3-pyrazolcarboxamid-derivater med cannabinoidreceptor-affinitet - Google Patents

3-pyrazolcarboxamid-derivater med cannabinoidreceptor-affinitet

Info

Publication number
DK0868420T3
DK0868420T3 DK96941716T DK96941716T DK0868420T3 DK 0868420 T3 DK0868420 T3 DK 0868420T3 DK 96941716 T DK96941716 T DK 96941716T DK 96941716 T DK96941716 T DK 96941716T DK 0868420 T3 DK0868420 T3 DK 0868420T3
Authority
DK
Denmark
Prior art keywords
cannabinoid receptor
carboxamide derivatives
receptor affinity
pyrazole carboxamide
pyrazole
Prior art date
Application number
DK96941716T
Other languages
Danish (da)
English (en)
Inventor
Francis Barth
Pierre Casellas
Joseph Millan
Didier Oustric
Murielle Rinaldi
Martine Sarran
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Application granted granted Critical
Publication of DK0868420T3 publication Critical patent/DK0868420T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK96941716T 1995-12-08 1996-12-06 3-pyrazolcarboxamid-derivater med cannabinoidreceptor-affinitet DK0868420T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9514547A FR2742148B1 (fr) 1995-12-08 1995-12-08 Nouveaux derives du pyrazole-3-carboxamide, procede pour leur preparation et compositions pharmaceutiques les contenant
PCT/FR1996/001953 WO1997021682A1 (fr) 1995-12-08 1996-12-06 Derives de 3-pyrazolecarboxamide avec une affinite pour le recepteur des cannabinoides

Publications (1)

Publication Number Publication Date
DK0868420T3 true DK0868420T3 (da) 2000-08-21

Family

ID=9485291

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96941716T DK0868420T3 (da) 1995-12-08 1996-12-06 3-pyrazolcarboxamid-derivater med cannabinoidreceptor-affinitet

Country Status (34)

Country Link
US (1) US5925768A (tr)
EP (2) EP0868420B1 (tr)
JP (1) JP3510270B2 (tr)
KR (1) KR100488610B1 (tr)
CN (1) CN1101813C (tr)
AR (1) AR004364A1 (tr)
AT (1) ATE191211T1 (tr)
AU (1) AU718763B2 (tr)
BR (1) BR9611986A (tr)
CA (1) CA2239489C (tr)
CZ (1) CZ294307B6 (tr)
DE (1) DE69607484T2 (tr)
DK (1) DK0868420T3 (tr)
EE (1) EE04674B1 (tr)
ES (1) ES2148820T3 (tr)
FR (1) FR2742148B1 (tr)
GR (1) GR3033626T3 (tr)
HU (1) HUP9901244A3 (tr)
IL (1) IL124801A (tr)
IS (1) IS4765A (tr)
MX (1) MX9804565A (tr)
MY (1) MY115228A (tr)
NO (1) NO310683B1 (tr)
NZ (1) NZ323962A (tr)
PL (1) PL186466B1 (tr)
PT (1) PT868420E (tr)
RU (1) RU2170230C2 (tr)
SI (1) SI0868420T1 (tr)
SK (1) SK283706B6 (tr)
TR (1) TR199801041T2 (tr)
TW (1) TW402594B (tr)
UA (1) UA44913C2 (tr)
WO (1) WO1997021682A1 (tr)
ZA (1) ZA9610299B (tr)

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US7276613B1 (en) 1998-11-24 2007-10-02 University Of Connecticut Retro-anandamides, high affinity and stability cannabinoid receptor ligands
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FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
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Also Published As

Publication number Publication date
NO310683B1 (no) 2001-08-13
SK75898A3 (en) 1999-01-11
PL327177A1 (en) 1998-11-23
AU1101097A (en) 1997-07-03
EP0885889A2 (fr) 1998-12-23
DE69607484T2 (de) 2000-10-26
EP0868420B1 (fr) 2000-03-29
EE04674B1 (et) 2006-08-15
ES2148820T3 (es) 2000-10-16
CN1207731A (zh) 1999-02-10
BR9611986A (pt) 1999-02-17
FR2742148B1 (fr) 1999-10-22
FR2742148A1 (fr) 1997-06-13
ATE191211T1 (de) 2000-04-15
EE9800171A (et) 1998-12-15
CZ177598A3 (cs) 1998-10-14
MX9804565A (es) 1998-09-30
KR100488610B1 (ko) 2005-09-26
CZ294307B6 (cs) 2004-11-10
NO982589D0 (no) 1998-06-05
ZA9610299B (en) 1997-06-18
IS4765A (is) 1998-06-08
PL186466B1 (pl) 2004-01-30
NO982589L (no) 1998-08-03
KR19990072004A (ko) 1999-09-27
AR004364A1 (es) 1998-11-04
NZ323962A (en) 1999-05-28
DE69607484D1 (de) 2000-05-04
HUP9901244A2 (hu) 1999-08-30
CA2239489C (en) 2006-05-09
MY115228A (en) 2003-04-30
RU2170230C2 (ru) 2001-07-10
TW402594B (en) 2000-08-21
WO1997021682A1 (fr) 1997-06-19
EP0868420A1 (fr) 1998-10-07
IL124801A (en) 2004-07-25
IL124801A0 (en) 1999-01-26
PT868420E (pt) 2000-08-31
JP3510270B2 (ja) 2004-03-22
TR199801041T2 (tr) 1998-08-21
UA44913C2 (uk) 2002-03-15
AU718763B2 (en) 2000-04-20
SI0868420T1 (en) 2000-10-31
JP2000502080A (ja) 2000-02-22
HUP9901244A3 (en) 2000-12-28
SK283706B6 (sk) 2003-12-02
EP0885889A3 (fr) 1999-01-27
GR3033626T3 (en) 2000-10-31
CN1101813C (zh) 2003-02-19
US5925768A (en) 1999-07-20
CA2239489A1 (en) 1997-06-19

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