HUP9901244A3 - 3-pyrazolecarboxamide derivatives having cannabinoid receptor affinity, intermediates, preparation and use thereof, pharmaceutical compositions containing these compounds - Google Patents

3-pyrazolecarboxamide derivatives having cannabinoid receptor affinity, intermediates, preparation and use thereof, pharmaceutical compositions containing these compounds

Info

Publication number
HUP9901244A3
HUP9901244A3 HU9901244A HUP9901244A HUP9901244A3 HU P9901244 A3 HUP9901244 A3 HU P9901244A3 HU 9901244 A HU9901244 A HU 9901244A HU P9901244 A HUP9901244 A HU P9901244A HU P9901244 A3 HUP9901244 A3 HU P9901244A3
Authority
HU
Hungary
Prior art keywords
intermediates
compounds
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
HU9901244A
Other languages
English (en)
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of HUP9901244A2 publication Critical patent/HUP9901244A2/hu
Publication of HUP9901244A3 publication Critical patent/HUP9901244A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HU9901244A 1995-12-08 1996-12-06 3-pyrazolecarboxamide derivatives having cannabinoid receptor affinity, intermediates, preparation and use thereof, pharmaceutical compositions containing these compounds HUP9901244A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9514547A FR2742148B1 (fr) 1995-12-08 1995-12-08 Nouveaux derives du pyrazole-3-carboxamide, procede pour leur preparation et compositions pharmaceutiques les contenant

Publications (2)

Publication Number Publication Date
HUP9901244A2 HUP9901244A2 (hu) 1999-08-30
HUP9901244A3 true HUP9901244A3 (en) 2000-12-28

Family

ID=9485291

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9901244A HUP9901244A3 (en) 1995-12-08 1996-12-06 3-pyrazolecarboxamide derivatives having cannabinoid receptor affinity, intermediates, preparation and use thereof, pharmaceutical compositions containing these compounds

Country Status (34)

Country Link
US (1) US5925768A (hu)
EP (2) EP0868420B1 (hu)
JP (1) JP3510270B2 (hu)
KR (1) KR100488610B1 (hu)
CN (1) CN1101813C (hu)
AR (1) AR004364A1 (hu)
AT (1) ATE191211T1 (hu)
AU (1) AU718763B2 (hu)
BR (1) BR9611986A (hu)
CA (1) CA2239489C (hu)
CZ (1) CZ294307B6 (hu)
DE (1) DE69607484T2 (hu)
DK (1) DK0868420T3 (hu)
EE (1) EE04674B1 (hu)
ES (1) ES2148820T3 (hu)
FR (1) FR2742148B1 (hu)
GR (1) GR3033626T3 (hu)
HU (1) HUP9901244A3 (hu)
IL (1) IL124801A (hu)
IS (1) IS4765A (hu)
MX (1) MX9804565A (hu)
MY (1) MY115228A (hu)
NO (1) NO310683B1 (hu)
NZ (1) NZ323962A (hu)
PL (1) PL186466B1 (hu)
PT (1) PT868420E (hu)
RU (1) RU2170230C2 (hu)
SI (1) SI0868420T1 (hu)
SK (1) SK283706B6 (hu)
TR (1) TR199801041T2 (hu)
TW (1) TW402594B (hu)
UA (1) UA44913C2 (hu)
WO (1) WO1997021682A1 (hu)
ZA (1) ZA9610299B (hu)

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US20010009965A1 (en) * 1998-05-04 2001-07-26 Alexandros Makriyannis Novel analgesic and immunomodulatory cannabinoids
US7589220B2 (en) * 1998-06-09 2009-09-15 University Of Connecticut Inhibitors of the anandamide transporter
US7897598B2 (en) * 1998-06-09 2011-03-01 Alexandros Makriyannis Inhibitors of the anandamide transporter
US7161016B1 (en) 1998-11-24 2007-01-09 University Of Connecticut Cannabimimetic lipid amides as useful medications
US7276613B1 (en) 1998-11-24 2007-10-02 University Of Connecticut Retro-anandamides, high affinity and stability cannabinoid receptor ligands
HUP0203437A3 (en) 1999-03-22 2003-07-28 Immugen Pharmaceuticals Inc So Use of resorcinol derivatives for producing pharmaceutical compositions for treatment of immune diseases
US6566560B2 (en) 1999-03-22 2003-05-20 Immugen Pharmaceuticals, Inc. Resorcinolic compounds
US6900236B1 (en) 1999-10-18 2005-05-31 University Of Connecticut Cannabimimetic indole derivatives
US8084467B2 (en) * 1999-10-18 2011-12-27 University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
JP2003511469A (ja) 1999-10-18 2003-03-25 ユニバーシティ オブ コネチカット 抹消カンナビノイド受容体（ｃｂ２）選択的配位子
US6943266B1 (en) 1999-10-18 2005-09-13 University Of Connecticut Bicyclic cannabinoid agonists for the cannabinoid receptor
US7119108B1 (en) 1999-10-18 2006-10-10 University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
US7393842B2 (en) * 2001-08-31 2008-07-01 University Of Connecticut Pyrazole analogs acting on cannabinoid receptors
US7741365B2 (en) * 1999-10-18 2010-06-22 University Of Connecticut Peripheral cannabinoid receptor (CB2) selective ligands
JP2003512357A (ja) * 1999-10-18 2003-04-02 ユニバーシティ オブ コネチカット カンナビノイドレセプタ拮抗物質としてのピラゾール誘導体
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US5015651A (en) * 1988-01-07 1991-05-14 E. I. Du Pont De Nemours And Company Treatment of hypertension with 1,2,4-angiotensin II antagonists
FR2665898B1 (fr) * 1990-08-20 1994-03-11 Sanofi Derives d'amido-3 pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2713225B1 (fr) * 1993-12-02 1996-03-01 Sanofi Sa N-pipéridino-3-pyrazolecarboxamide substitué.
FR2714057B1 (fr) * 1993-12-17 1996-03-08 Sanofi Elf Nouveaux dérivés du 3-pyrazolecarboxamide, procédé pour leur préparation et compositions pharmaceutiques les contenant.

Also Published As

Publication number Publication date
NO310683B1 (no) 2001-08-13
SK75898A3 (en) 1999-01-11
PL327177A1 (en) 1998-11-23
AU1101097A (en) 1997-07-03
EP0885889A2 (fr) 1998-12-23
DE69607484T2 (de) 2000-10-26
EP0868420B1 (fr) 2000-03-29
EE04674B1 (et) 2006-08-15
ES2148820T3 (es) 2000-10-16
CN1207731A (zh) 1999-02-10
BR9611986A (pt) 1999-02-17
FR2742148B1 (fr) 1999-10-22
FR2742148A1 (fr) 1997-06-13
ATE191211T1 (de) 2000-04-15
EE9800171A (et) 1998-12-15
CZ177598A3 (cs) 1998-10-14
MX9804565A (es) 1998-09-30
KR100488610B1 (ko) 2005-09-26
CZ294307B6 (cs) 2004-11-10
NO982589D0 (no) 1998-06-05
ZA9610299B (en) 1997-06-18
IS4765A (is) 1998-06-08
PL186466B1 (pl) 2004-01-30
NO982589L (no) 1998-08-03
KR19990072004A (ko) 1999-09-27
AR004364A1 (es) 1998-11-04
NZ323962A (en) 1999-05-28
DE69607484D1 (de) 2000-05-04
HUP9901244A2 (hu) 1999-08-30
CA2239489C (en) 2006-05-09
MY115228A (en) 2003-04-30
RU2170230C2 (ru) 2001-07-10
TW402594B (en) 2000-08-21
DK0868420T3 (da) 2000-08-21
WO1997021682A1 (fr) 1997-06-19
EP0868420A1 (fr) 1998-10-07
IL124801A (en) 2004-07-25
IL124801A0 (en) 1999-01-26
PT868420E (pt) 2000-08-31
JP3510270B2 (ja) 2004-03-22
TR199801041T2 (xx) 1998-08-21
UA44913C2 (uk) 2002-03-15
AU718763B2 (en) 2000-04-20
SI0868420T1 (en) 2000-10-31
JP2000502080A (ja) 2000-02-22
SK283706B6 (sk) 2003-12-02
EP0885889A3 (fr) 1999-01-27
GR3033626T3 (en) 2000-10-31
CN1101813C (zh) 2003-02-19
US5925768A (en) 1999-07-20
CA2239489A1 (en) 1997-06-19

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