DE69943296D1 - Makrocyclische analoga und verfahren zu ihrer verwendung und herstellung - Google Patents

Makrocyclische analoga und verfahren zu ihrer verwendung und herstellung

Info

Publication number
DE69943296D1
DE69943296D1 DE69943296T DE69943296T DE69943296D1 DE 69943296 D1 DE69943296 D1 DE 69943296D1 DE 69943296 T DE69943296 T DE 69943296T DE 69943296 T DE69943296 T DE 69943296T DE 69943296 D1 DE69943296 D1 DE 69943296D1
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DE
Germany
Prior art keywords
manufacture
macrocyclic analogues
macrocyclic
analogues
useful
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69943296T
Other languages
German (de)
English (en)
Inventor
Bruce A Littlefield
Monica Palme
Boris M Seletsky
Murray J Towle
Melvin J Yu
Wanjun Zheng
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eisai R&D Management Co Ltd
Original Assignee
Eisai R&D Management Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22219026&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE69943296(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Eisai R&D Management Co Ltd filed Critical Eisai R&D Management Co Ltd
Application granted granted Critical
Publication of DE69943296D1 publication Critical patent/DE69943296D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Steroid Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
DE69943296T 1998-06-17 1999-06-16 Makrocyclische analoga und verfahren zu ihrer verwendung und herstellung Expired - Lifetime DE69943296D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8968298P 1998-06-17 1998-06-17
PCT/US1999/013677 WO1999065894A1 (en) 1998-06-17 1999-06-16 Macrocyclic analogs and methods of their use and preparation

Publications (1)

Publication Number Publication Date
DE69943296D1 true DE69943296D1 (de) 2011-05-05

Family

ID=22219026

Family Applications (2)

Application Number Title Priority Date Filing Date
DE69943296T Expired - Lifetime DE69943296D1 (de) 1998-06-17 1999-06-16 Makrocyclische analoga und verfahren zu ihrer verwendung und herstellung
DE201112100031 Pending DE122011100031I1 (de) 1998-06-17 1999-06-16 Makrocyclische analoga und verfahren zu ihrer verwendung und herstellung.

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE201112100031 Pending DE122011100031I1 (de) 1998-06-17 1999-06-16 Makrocyclische analoga und verfahren zu ihrer verwendung und herstellung.

Country Status (22)

Country Link
US (4) US6214865B1 (https=)
EP (4) EP2272839B1 (https=)
JP (1) JP4454151B2 (https=)
KR (1) KR100798600B1 (https=)
CN (1) CN1216051C (https=)
AT (1) ATE502932T1 (https=)
AU (1) AU762998B2 (https=)
BE (1) BE2011C028I2 (https=)
BR (1) BRPI9911326B8 (https=)
CA (3) CA2335300C (https=)
CY (2) CY1111516T1 (https=)
DE (2) DE69943296D1 (https=)
DK (1) DK1087960T3 (https=)
FR (1) FR11C0038I2 (https=)
HU (1) HU227912B1 (https=)
IL (1) IL139960A0 (https=)
LU (1) LU91854I2 (https=)
NO (5) NO328280B1 (https=)
NZ (1) NZ508597A (https=)
PT (1) PT1087960E (https=)
WO (1) WO1999065894A1 (https=)
ZA (1) ZA200007159B (https=)

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RU2579511C2 (ru) 2010-01-26 2016-04-10 Эйсай Ар Энд Ди Менеджмент Ко., Лтд. Производные фуро[3,2-в]пирана, применимые в синтезе аналогов

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JP4454151B2 (ja) 2010-04-21
NO2011026I2 (no) 2012-06-11
US6365759B1 (en) 2002-04-02
BE2011C028I2 (en) 2018-08-24
AU762998B2 (en) 2003-07-10
EP2277873A1 (en) 2011-01-26
NO20006316L (no) 2001-02-15
BR9911326A (pt) 2001-04-03
CA2632433A1 (en) 1999-12-23
HUP0103357A2 (hu) 2002-01-28
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CA2335300A1 (en) 1999-12-23
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KR100798600B1 (ko) 2008-01-28
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EP2272839B1 (en) 2012-08-22
LU91854I2 (fr) 2011-10-17
ATE502932T1 (de) 2011-04-15
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